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1
المؤلفون: Maria Rosalia Pasca, Marco Pieroni, Giannamaria Annunziato, Giorgia Mori, Marialaura Pavone, Gabriele Costantino, Federica Vacondio, Elisa Azzali, Miriam Girardini
المصدر: ACS Med Chem Lett
مصطلحات موضوعية: Scaffold, 010405 organic chemistry, Drug discovery, Computer science, Isostere, Organic Chemistry, 2-aminothiazole, 01 natural sciences, Biochemistry, Medicinal chemistry, 0104 chemical sciences, 010404 medicinal & biomolecular chemistry, Chemical agents, Drug Discovery
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2
المؤلفون: Marco Pieroni, Federica Vacondio, Michal Zolkiewski, Gabriele Costantino, Elisa Azzali, Nicoletta Basilico, Silvia Parapini, Giannamaria Annunziato, Claudia Beato, Agostino Bruno
المصدر: Journal of Medicinal Chemistry. 60:1959-1970
مصطلحات موضوعية: 0301 basic medicine, Combination therapy, Phenotypic screening, Drug Evaluation, Preclinical, Thiophenes, Pharmacology, Biology, 01 natural sciences, Antimalarials, Structure-Activity Relationship, 03 medical and health sciences, parasitic diseases, Drug Discovery, medicine, Humans, Structure–activity relationship, Antimalarial Agent, Artemisinin, Biological evaluation, 010405 organic chemistry, Drug discovery, medicine.disease, Amides, 0104 chemical sciences, 030104 developmental biology, Molecular Medicine, Malaria, medicine.drug
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3
المؤلفون: Diana Machado, Tatiane S. Coelho, Elizeth Lopes, Sofia Santos Costa, Miguel Viveiros, Elisa Azzali, Pedro Eduardo Almeida da Silva, Isabel Couto, Marco Pieroni
المصدر: ASSAY and Drug Development Technologies. 14:524-534
مصطلحات موضوعية: 0301 basic medicine, medicine.medical_specialty, Tuberculosis, medicine.drug_class, medicine.medical_treatment, Mycobacterium smegmatis, 030106 microbiology, Antibiotics, Microbial Sensitivity Tests, Antimycobacterial, Mycobacterium tuberculosis, 03 medical and health sciences, Drug Discovery, medicine, Humans, Intensive care medicine, Therapeutic regimen, biology, Experimental model, Models, Theoretical, biology.organism_classification, medicine.disease, Anti-Bacterial Agents, High-Throughput Screening Assays, 030104 developmental biology, Immunology, Molecular Medicine, Adjuvant
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::090ab5bcfb1de5d3d674f966ace8a353
https://doi.org/10.1089/adt.2016.752 -
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المصدر: RSC advances. 9(35)
مصطلحات موضوعية: chemistry.chemical_classification, Chemistry, General Chemical Engineering, Protide, 02 engineering and technology, General Chemistry, Prodrug, 010402 general chemistry, 021001 nanoscience & nanotechnology, Ribonucleoside, 01 natural sciences, Combinatorial chemistry, Microwave assisted, 0104 chemical sciences, chemistry.chemical_compound, Nucleotide, Organic synthesis, 0210 nano-technology, Nucleoside, Microwave
وصف الملف: application/pdf
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::82a1547922f799fdcbfd43601df1def2
https://pubmed.ncbi.nlm.nih.gov/35514718 -
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المؤلفون: Marco Pieroni, Elisa Azzali, Gabriele Costantino, Diana Machado, Miguel Viveiros, Isabel Couto
المصدر: Future microbiology. 13
مصطلحات موضوعية: 0301 basic medicine, Microbiology (medical), Tuberculosis, medicine.medical_treatment, 030106 microbiology, Antitubercular Agents, Microbial Sensitivity Tests, Pharmacology, Microbiology, Membrane Potentials, Mycobacterium tuberculosis, 03 medical and health sciences, Adenosine Triphosphate, medicine, Humans, Membrane potential, biology, Chemistry, Chemiosmosis, Macrophages, Biological Transport, medicine.disease, biology.organism_classification, Thiazoles, Lipophilicity, Efflux, Adjuvant, Intracellular
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المؤلفون: Sanja Glisic, Elisa Azzali, Vladimir Perovic, Jelica Vucicevic, Nevena Veljkovic, Tatjana Srdic-Rajic, Sabrina Tassini, Marco Pieroni, Katarina Nikolic, Marco Radi, Gabriele Costantino, Jonne M. Laurila, Mika Scheinin, Danica Agbaba
المصدر: Bioorganic and Medicinal Chemistry
Bioorganic & Medicinal Chemistryمصطلحات موضوعية: 0301 basic medicine, Drug, medicine.medical_treatment, media_common.quotation_subject, Clinical Biochemistry, Pharmaceutical Science, Imidazoline receptor, Apoptosis, Pharmacology, Ligands, Rilmenidine, ta3111, Biochemistry, Drug design, Synthesis, 03 medical and health sciences, 0302 clinical medicine, Receptors, Adrenergic, alpha-2, Drug Discovery, medicine, Humans, Cytotoxic T cell, Doxorubicin, Oxazoles, Molecular Biology, media_common, Antibiotics, Antineoplastic, Molecular Structure, Cytotoxic activity, Chemistry, Organic Chemistry, Drug Synergism, Ligand (biochemistry), ta3122, 3. Good health, 030104 developmental biology, alpha(2)-Adrenoceptors, 030220 oncology & carcinogenesis, Doxorubicin synergism, Molecular Medicine, K562 Cells, Adrenergic alpha-Agonists, Adjuvant, medicine.drug
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7
المؤلفون: Giannamaria Annunziato, Manuela Villa, Claudia Beato, Gabriele Costantino, Marco Pieroni, Elisa Azzali, Mario Varasi, Paolo Trifiro, Paola Vianello, Paola Dessanti, Ciro Mercurio, Giuseppe Meroni
المصدر: European Journal of Medicinal Chemistry. 92:377-386
مصطلحات موضوعية: Cyclopropanes, Models, Molecular, Stereochemistry, Structure-Activity Relationship, Drug Discovery, Histone methylation, medicine, Humans, Epigenetics, Histone Demethylases, Pharmacology, Dose-Response Relationship, Drug, Molecular Structure, biology, Chemistry, Organic Chemistry, Tranylcypromine, KDM1A, General Medicine, Recombinant Proteins, Histone, Biochemistry, Acetylation, DNA methylation, biology.protein, Demethylase, medicine.drug
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8دورية أكاديمية
المؤلفون: Marco Pieroni, Diana Machado, Elisa Azzali, Sofia Santos Costa, Isabel Couto, Gabriele Costantino, Miguel Viveiros
المصدر: Journal of Medicinal Chemistry; Aug2015, Vol. 58 Issue 15, p5842-5853, 12p
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9Rational design and synthesis of thioridazine analogues as enhancers of the antituberculosis therapy
المؤلفون: Gabriele Costantino, Diana Machado, Sofia Santos Costa, Marco Pieroni, Miguel Viveiros, Elisa Azzali, Isabel Couto
المصدر: Universidade Nova de Lisboa
CIÊNCIAVITAEمصطلحات موضوعية: Tuberculosis, Mycobacterium smegmatis, Antitubercular Agents, Drug resistance, Thioridazine, Microbial Sensitivity Tests, Pharmacology, Mycobacterium tuberculosis, In vivo, Drug Discovery, medicine, Humans, biology, Chemistry, Macrophages, Rational design, Drug Synergism, medicine.disease, biology.organism_classification, Drug Design, Molecular Medicine, Efflux, Ex vivo, medicine.drug
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::1edef3c31ba4558786b3348a116bb350
https://novaresearch.unl.pt/en/publications/1b149d07-7a7c-46ad-9901-aac342941551 -
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المؤلفون: Diana Machado, Elisa Azzali, Isabel Couto, Gabriele Costantino, Marco Pieroni, Miguel Viveiros
المصدر: Universidade Nova de Lisboa
CIÊNCIAVITAEURL الوصول: https://explore.openaire.eu/search/publication?articleId=dedup_wf_001::478be6d0e7ef78a551ba85a6dd098529
https://novaresearch.unl.pt/en/publications/0b4334d0-69cc-4a75-9419-fc7f8d8370bb