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1
المؤلفون: Jay A. Grobler, Meizhen Feng, Yuan Li, Yves Ducharme, Jean-Pierre Falgueyret, Bernard Cote, Youwei Yan, Louis-Charles Campeau, Ernest Asante-Appiah, Ming-Tain Lai, Jason Burch, Marc V. Witmer, Daria J. Hazuda, Michael D. Miller, Nancy A. Sachs, Elizabeth Cauchon, Paul Tawa, Daniel J. DiStefano, Meiqing Lu
المصدر: Antimicrobial Agents and Chemotherapy. 58:1652-1663
مصطلحات موضوعية: Efavirenz, Anti-HIV Agents, Pyridones, Etravirine, HIV Infections, In Vitro Techniques, Biology, Virus Replication, Antiviral Agents, Monocytes, Virus, chemistry.chemical_compound, Doravirine, medicine, Humans, Pharmacology (medical), Pharmacology, Reverse-transcriptase inhibitor, Macrophages, virus diseases, Drug Synergism, Triazoles, Virology, HIV Reverse Transcriptase, Reverse transcriptase, Infectious Diseases, chemistry, Viral replication, Rilpivirine, HIV-1, medicine.drug
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::031e80e91b45808e18f50cd354a2ad72
https://doi.org/10.1128/aac.02403-13 -
2
المؤلفون: Sébastien Gagné, Amandine Chefson, Sylvie Toulmond, Patrick Lacombe, Mélissa Arbour, Austin Chen, Dan McKay, Elizabeth Cauchon, Erich L. Grimm, Yeeman K. Ramtohul, M. David Percival, Jean-François Lévesque, Yves Ducharme, Dwight Macdonald, Yongxin Han, René St-Jacques, Robert Houle, Bruce Mackay, Jean-Pierre Falgueyret, Pierre-André Fournier
المصدر: Bioorganic & Medicinal Chemistry Letters. 22:2670-2674
مصطلحات موضوعية: Dependent manner, medicine.drug_class, Clinical Biochemistry, Administration, Oral, Pharmaceutical Science, Pharmacology, Biochemistry, Renin inhibitor, Structure-Activity Relationship, Enzyme activator, chemistry.chemical_compound, Catalytic Domain, Renin, Drug Discovery, Renin–angiotensin system, medicine, Animals, Humans, Structure–activity relationship, Isoxazole, Molecular Biology, Antihypertensive Agents, Molecular Structure, CYP3A4, Chemistry, Organic Chemistry, Isoxazoles, Rats, Enzyme Activation, Drug Design, Molecular Medicine, Linker
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3
المؤلفون: Stephen M. Soisson, Tom Y.-H. Wu, Michel Gallant, Austin Chen, Dwight Macdonald, Daniel Dube, Robert Houle, Jean-Pierre Falgueyret, Renee Aspiotis, Dan McKay, Jean-François Lévesque, Patrick Roy, Helene Juteau, Sébastien Gagné, M. David Percival, Erich L. Grimm, Sebastien Laliberte, Patrick Lacombe, Elizabeth Cauchon
المصدر: Bioorganic & Medicinal Chemistry Letters. 21:2430-2436
مصطلحات موضوعية: Stereochemistry, Carboxylic acid, Clinical Biochemistry, hERG, Drug Evaluation, Preclinical, Administration, Oral, Pharmaceutical Science, Biochemistry, Chemical synthesis, Rats, Sprague-Dawley, Structure-Activity Relationship, chemistry.chemical_compound, Dogs, Piperidines, Catalytic Domain, Renin, Drug Discovery, Animals, Humans, Structure–activity relationship, Computer Simulation, Protease Inhibitors, Molecular Biology, chemistry.chemical_classification, biology, Organic Chemistry, Prodrug, Rats, Enzyme, chemistry, Enzyme inhibitor, Zwitterion, biology.protein, Molecular Medicine
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4
المؤلفون: Bruno Roy, Claudio Sturino, Nicolas Lachance, Robert Zamboni, Kathleen M. Metters, Christine Brideau, Lianhai Li, John Scheigetz, Danielle Denis, Deborah Slipetz, Marie-Claude Carrière, Elizabeth Cauchon, Gillian Greig, Gary P. O'Neill, Carl Berthelette, Michael J. Boyd, Marie-Claude Mathieu, Sonia Lamontagne, Nicole Sawyer, Robert N. Young, Nancy N. Tsou, Zhaoyin Wang, Stacia Kargman, Marc Labelle
المصدر: Bioorganic & Medicinal Chemistry Letters. 16:3043-3048
مصطلحات موضوعية: Indole test, Indoles, Molecular Structure, Chemistry, Receptors, Prostaglandin, Organic Chemistry, Clinical Biochemistry, Antagonist, Pharmaceutical Science, Biochemistry, Chemical synthesis, In vitro, Structure-Activity Relationship, chemistry.chemical_compound, Safrole, Drug Discovery, Molecular Medicine, Prostaglandin D2, Receptors, Immunologic, Receptor, Molecular Biology, Prostaglandin G2, Prostaglandin D2 receptor
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5
المؤلفون: Elizabeth Cauchon, Nicole Sawyer, François G. Gervais, Rani P.G. Cruz, Gary P. O'Neill, Donald W. Nicholson, Kathleen M. Metters, Anne Chateauneuf
المصدر: British Journal of Pharmacology. 137:1163-1172
مصطلحات موضوعية: Pharmacology, education.field_of_study, Ligand binding assay, Population, respiratory system, Biology, Molecular biology, Dissociation constant, chemistry.chemical_compound, chemistry, Biochemistry, Potency, lipids (amino acids, peptides, and proteins), Prostaglandin D2, Binding site, Receptor, education, Prostaglandin D2 receptor
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6
المؤلفون: Nguyen Natalie, Ernest Asante-Appiah, Manuel Chan, Nathalie Coulombe, Yves Ducharme, Mark Wrona, C. Bayly, Paul Tawa, Serge Plamondon, Kristina Dupont-Gaudet, Amandine Chefson, Jean-François Truchon, Sébastien Guiral, Louis-Charles Campeau, Joe Vacca, Sébastien Gagné, Rob Papp, Elizabeth Cauchon, Leanne Bedard, Eric Langlois, Robert Forget, Stéphane G. Ouellet, Stephanie Roy, Mélina Girardin, Jason Burch, Jean-Pierre Falgueyret, Bernard Cote, Danny Gauvreau, St-Onge Miguel, Marc Blouin, Ria Seliniotakis, Wanda Cromlish, Chun Sing Li, Amélie Roy, Smita Debnath, Youwei Yan, Denis Deschenes
المصدر: Bioorganicmedicinal chemistry letters. 24(3)
مصطلحات موضوعية: Anti-HIV Agents, Pyridones, viruses, Clinical Biochemistry, Mutant, Pharmaceutical Science, Pharmacology, Crystallography, X-Ray, Biochemistry, Nucleoside Reverse Transcriptase Inhibitor, Rats, Sprague-Dawley, chemistry.chemical_compound, Inhibitory Concentration 50, Dogs, Pharmacokinetics, immune system diseases, Doravirine, Drug Discovery, Drug Resistance, Viral, Potency, Animals, Humans, Molecular Biology, Cells, Cultured, Molecular Structure, Chemistry, Organic Chemistry, Wild type, virus diseases, Triazoles, Virology, Reverse transcriptase, Rats, Regimen, Mutation, HIV-1, Molecular Medicine, Reverse Transcriptase Inhibitors
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7
المصدر: European Journal of Pharmacology. 400:145-153
مصطلحات موضوعية: Cell Survival, Basic fibroblast growth factor, Dermatan Sulfate, Dermatan sulfate, Dermal fibroblast, Glycosaminoglycan, chemistry.chemical_compound, Cell Adhesion, medicine, Humans, Drug Interactions, Chondroitin sulfate, Fibroblast, Cells, Cultured, Polysaccharide-Lyases, Skin, Pharmacology, Chondroitin Lyases, biology, Fibroblasts, Molecular biology, carbohydrates (lipids), medicine.anatomical_structure, Chondroitin Sulfate Proteoglycans, Proteoglycan, chemistry, Biochemistry, cardiovascular system, biology.protein, Fibroblast Growth Factor 2, Cell Division, Chondroitin AC lyase
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8
المؤلفون: Mélissa Arbour, Gavin Chit Tsui, Jean-Pierre Falgueyret, Pierre-André Fournier, Yongxin Han, Michel Gallant, Patrick Lacombe, Daniel Dube, Daniel Simard, Elizabeth Cauchon, Austin Chen, Renee Aspiotis, Suzanna Liu, René St-Jacques, Christophe Mellon, Erich L. Grimm, Yeeman K. Ramtohul, Helene Juteau
المصدر: Bioorganicmedicinal chemistry letters. 22(5)
مصطلحات موضوعية: Transgene, Clinical Biochemistry, hERG, Pharmaceutical Science, Biological Availability, Pharmacology, Biochemistry, Plasma renin activity, Rats, Sprague-Dawley, Structure-Activity Relationship, Dogs, Piperidines, Drug Discovery, Renin–angiotensin system, Renin, Structure–activity relationship, Animals, Cytochrome P-450 CYP3A, Humans, Animal species, Molecular Biology, Antihypertensive Agents, Cytochrome P-450 CYP3A Inhibitors, biology, Chemistry, Organic Chemistry, Ether-A-Go-Go Potassium Channels, Bioavailability, Rats, Hypertension, biology.protein, Molecular Medicine, Rats, Transgenic
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9
المؤلفون: Renee Aspiotis, Amadine Chefson, Jean-François Lévesque, Yongxin Han, Louis-Charles Campeau, Dan McKay, Guillaume Larouche, Jean-Pierre Falgueyret, Robert Houle, Elizabeth Cauchon, David Percival, Austin Chen, Sébastien Gagné, Yves Ducharme, Sebastien Laliberte
المصدر: Bioorganicmedicinal chemistry letters. 21(24)
مصطلحات موضوعية: medicine.drug_class, Stereochemistry, Clinical Biochemistry, hERG, Pharmaceutical Science, Biochemistry, Renin inhibitor, Structure-Activity Relationship, Dogs, Piperidines, Catalytic Domain, Drug Discovery, Renin–angiotensin system, Renin, medicine, Animals, Cytochrome P-450 CYP3A, Humans, Computer Simulation, Protease Inhibitors, Spiro Compounds, Molecular Biology, Antihypertensive Agents, Binding Sites, biology, CYP3A4, Chemistry, Organic Chemistry, Macaca mulatta, Rats, Drug Design, Hypertension, biology.protein, Molecular Medicine, Cytochrome P-450 CYP3A Inhibitors
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10
المؤلفون: Jean-Pierre Falgueyret, Greg L. Beilhartz, Maryam Ehteshami, Siqi Zhu, Jay A. Grobler, Anick Auger, Roman A. Melnyk, Elizabeth Cauchon, Matthias Götte
المصدر: The Journal of biological chemistry. 286(34)
مصطلحات موضوعية: Indoles, DNA polymerase, Pyridones, Allosteric regulation, Biochemistry, Catalysis, chemistry.chemical_compound, Nitriles, Molecular Biology, Polymerase, DNA Primers, chemistry.chemical_classification, biology, Cell Biology, Reverse Transcription, Molecular biology, Footprinting, Reverse transcriptase, HIV Reverse Transcriptase, Enzyme, chemistry, DNA, Viral, biology.protein, HIV-1, RNA, Viral, Primer (molecular biology), DNA, Allosteric Site, Molecular Biophysics
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::fa1097466738794c0e4ef994580df613
https://pubmed.ncbi.nlm.nih.gov/21737446