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1دورية أكاديمية
المؤلفون: Christopher C. Presley, Charles K. Perry, Elizabeth S. Childress, Matthew J. Mulder, Vincent B. Luscombe, Alice L. Rodriguez, Colleen M. Niswender, P. Jeffrey Conn, Craig W. Lindsley
المصدر: ACS Omega, Vol 4, Iss 7, Pp 12782-12789 (2019)
وصف الملف: electronic resource
Relation: https://doaj.org/toc/2470-1343
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2
المؤلفون: Stefan R. Hargett, Elizabeth S. Childress, Joseph M. Salamoun, Jose A Santiago-Rivera, Divya P. Shah, Christopher J Garcia, Webster L. Santos, Sing-Young Chen, Kyle L. Hoehn, Stephanie J. Alexopoulos, Yumin Dai, Simon P. Tucker
المصدر: J Med Chem
مصطلحات موضوعية: Male, Pyrazine, Protonophore, Mitochondria, Liver, Diamines, Mitochondrion, 01 natural sciences, Article, 03 medical and health sciences, chemistry.chemical_compound, Oxygen Consumption, Aniline, Non-alcoholic Fatty Liver Disease, In vivo, Drug Discovery, Animals, 030304 developmental biology, Oxadiazoles, 0303 health sciences, Uncoupling Agents, Depolarization, Small molecule, 0104 chemical sciences, Mice, Inbred C57BL, 010404 medicinal & biomolecular chemistry, Liver, chemistry, Biochemistry, Pyrazines, Molecular Medicine, Lead compound
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3
المؤلفون: Colleen M. Niswender, Christopher C Presley, P. Jeffrey Conn, Vincent B. Luscombe, Alice L. Rodriguez, Charles K. Perry, Craig W. Lindsley, Matthew J. Mulder, Elizabeth S. Childress
المصدر: ACS Omega, Vol 4, Iss 7, Pp 12782-12789 (2019)
مصطلحات موضوعية: Molecular switch, Cytochrome, biology, Ligand, General Chemical Engineering, Metabolite, Allosteric regulation, General Chemistry, Combinatorial chemistry, lcsh:Chemistry, chemistry.chemical_compound, lcsh:QD1-999, chemistry, Biotransformation, In vivo, biology.protein, G protein-coupled receptor
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4
المؤلفون: Colleen M. Niswender, Craig W. Lindsley, Andrew S. Felts, Vincent B. Luscombe, P. Jeffrey Conn, Hyekyung P. Cho, Elizabeth S. Childress, Megan M. Breiner, Joshua M. Wieting, Kyle A. Emmitte, Madeline F. Long, Alice L. Rodriguez, Anna L. Blobaum
المصدر: Journal of Medicinal Chemistry. 62:378-384
مصطلحات موضوعية: 0303 health sciences, Pyrimidine, medicine.drug_class, Stereochemistry, Allosteric regulation, Carboxamide, 01 natural sciences, 0104 chemical sciences, 010404 medicinal & biomolecular chemistry, 03 medical and health sciences, chemistry.chemical_compound, chemistry, Metabotropic glutamate receptor, Drug Discovery, Pyridine, medicine, Molecular Medicine, Structure–activity relationship, Selectivity, Receptor, 030304 developmental biology
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5
المؤلفون: Sing-Young Chen, Simon P. Tucker, Stefan R. Hargett, Elizabeth S. Childress, Martina Beretta, Kyle L. Hoehn, Kate G. R. Quinlan, Stephanie J. Alexopoulos, Webster L. Santos, Isabella Aleksovska, Charles G. Cranfield, Divya P. Shah, Ellen M. Olzomer, Joseph M. Salamoun, Tristan Rawling, Ariane Roseblade, Margaret J. Morris
المصدر: Metabolism: clinical and experimental. 117
مصطلحات موضوعية: 0301 basic medicine, Male, medicine.medical_specialty, Food intake, Endocrinology, Diabetes and Metabolism, medicine.medical_treatment, 030209 endocrinology & metabolism, Diet, High-Fat, Small Molecule Libraries, 03 medical and health sciences, chemistry.chemical_compound, Eating, Mice, 0302 clinical medicine, Endocrinology, Metabolic Diseases, In vivo, Internal medicine, medicine, Animals, Insulin, Obesity, Adiposity, business.industry, Cholesterol, Body Weight, Calorimetry, Indirect, Metabolism, medicine.disease, Lipid Metabolism, Mitochondria, Respiratory quotient, Mice, Inbred C57BL, 030104 developmental biology, Glucose, chemistry, Diet, Western, Lean body mass, Insulin Resistance, business, Energy Metabolism
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6
المؤلفون: Anna L. Blobaum, Jerri M. Rook, Jonathan W. Dickerson, Colleen M. Niswender, Julie L. Engers, Hekyung P Cho, Elizabeth S. Childress, Darren W. Engers, Rory A. Capstick, P. Jeffrey Conn, Craig W. Lindsley, Vincent B. Luscombe, Madeline F. Long
المصدر: ACS Medicinal Chemistry Letters. 9:917-922
مصطلحات موضوعية: 0301 basic medicine, Agonist, medicine.drug_class, Organic Chemistry, Allosteric regulation, Carboxamide, Pharmacology, Biochemistry, 03 medical and health sciences, chemistry.chemical_compound, 030104 developmental biology, 0302 clinical medicine, chemistry, Drug Discovery, Pyridine, Toxicity, medicine, Potency, Cholinergic, 030217 neurology & neurosurgery, EC50
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7
المصدر: Journal of Medicinal Chemistry. 61:4641-4655
مصطلحات موضوعية: 0301 basic medicine, ATP synthase, biology, Chemistry, Metabolism, Small molecule, Drug synergism, Cell biology, 03 medical and health sciences, 030104 developmental biology, Biochemistry, Mitochondrial matrix, Drug Discovery, biology.protein, Molecular Medicine, Inner mitochondrial membrane
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8
المؤلفون: Kevin R. Lynch, Yugesh Kharel, Webster L. Santos, Anne M. Brown, David R. Bevan, Elizabeth S. Childress
المصدر: Journal of Medicinal Chemistry. 60:3933-3957
مصطلحات موضوعية: 0301 basic medicine, Sphingosine kinase, In Vitro Techniques, Article, Mice, 03 medical and health sciences, chemistry.chemical_compound, 0302 clinical medicine, Aminothiazole, Drug Discovery, Animals, Humans, Enzyme Inhibitors, Receptor, biology, Sphingosine, Cell growth, Sphingosine Kinase 2, Rats, Phosphotransferases (Alcohol Group Acceptor), SPHK2, 030104 developmental biology, Biochemistry, Sphingosine kinase 1, chemistry, Drug Design, 030220 oncology & carcinogenesis, Cancer research, biology.protein, Molecular Medicine
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9
المصدر: The Journal of organic chemistry. 84(9)
مصطلحات موضوعية: 010405 organic chemistry, Chemistry, Organic Chemistry, Regioselectivity, chemistry.chemical_element, 010402 general chemistry, 01 natural sciences, Combinatorial chemistry, Microwave assisted, High yielding, 0104 chemical sciences, Catalysis, chemistry.chemical_compound, Pyridine, Palladium
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10
المؤلفون: Elizabeth S. Childress, Webster L. Santos, Frank Gillam, Jeannine S. Strobl, Masoud Agah, Chenming Zhang, Vaishnavi Srinivasaraghavan, Hesam Babahosseini, Zongmin Zhao
المصدر: Lab on a Chip
مصطلحات موضوعية: Cell, Biomedical Engineering, Sphingosine kinase, Antineoplastic Agents, Breast Neoplasms, Bioengineering, 02 engineering and technology, Electric Capacitance, 01 natural sciences, Biochemistry, Structure-Activity Relationship, chemistry.chemical_compound, Drug Delivery Systems, Polylactic Acid-Polyglycolic Acid Copolymer, Single-cell analysis, Cell Line, Tumor, medicine, Humans, Lactic Acid, Protein Kinase Inhibitors, Cell Proliferation, Membrane potential, Molecular Structure, Cell growth, Chemistry, 010401 analytical chemistry, technology, industry, and agriculture, General Chemistry, Microfluidic Analytical Techniques, 021001 nanoscience & nanotechnology, Biomechanical Phenomena, 0104 chemical sciences, 3. Good health, Phosphotransferases (Alcohol Group Acceptor), PLGA, medicine.anatomical_structure, Cancer cell, Drug delivery, Disease Progression, Biophysics, Nanoparticles, Female, Single-Cell Analysis, 0210 nano-technology, Polyglycolic Acid, Biomedical engineering
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::c152e246c298a2b5665c486b5e372f9b
https://doi.org/10.1039/c5lc01201e