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1
المؤلفون: Alessandro Poffe, Simone Spada, Carla Marchioro, Mauro Corsi, Romano Di Fabio, Michael Trower, Philip Gerrard, Giuseppe Alvaro, Simone Braggio, Cristiana Griffante, Laura Piccoli, Elvira Tranquillini, Sergio Melotto, Alfonso Pozzan, Emiliangelo Ratti, Renzo Carletti
المصدر: Bioorganic & Medicinal Chemistry. 21:6264-6273
مصطلحات موضوعية: Male, Models, Molecular, Orvepitant, Clinical Biochemistry, Molecular Conformation, Druggability, Pharmaceutical Science, CHO Cells, Pharmacology, Biology, Biochemistry, Piperazines, Cricetulus, Dogs, Neurokinin-1 Receptor Antagonists, Piperidines, Cricetinae, Drug Discovery, Casopitant, medicine, Animals, Humans, Receptor, Molecular Biology, Aprepitant, G protein-coupled receptor, Behavior, Animal, Organic Chemistry, Receptors, Neurokinin-1, Bridged Bicyclo Compounds, Heterocyclic, Antidepressive Agents, Rats, Molecular Medicine, Female, NK1 receptor antagonist, Pharmacophore, Gerbillinae, Half-Life, Protein Binding, medicine.drug
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2
المؤلفون: Aldo Feriani, Karen L Roberts, Beatrice Oliosi, Giovanna Tedesco, Robert J. Barnaby, Carla Marchioro, Maria Elvira Tranquillini, Paolo G. Cassarà, A. Ursini, Franciscus T.M. van Amsterdam, Angelo Reggiani, Mauro Corsi, S. Polinelli, Emiliangelo Ratti, Daniele Donati, Giovanni Curotto, David G. Trist, Daniela Niccolai, Gabriella Finizia
المصدر: Bioorganic & Medicinal Chemistry. 19:4257-4273
مصطلحات موضوعية: Stereochemistry, Guinea Pigs, Clinical Biochemistry, Pharmaceutical Science, Ring (chemistry), Biochemistry, Mice, Structure-Activity Relationship, Cholecystokinin-2 Receptor, chemistry.chemical_compound, Dogs, Drug Discovery, Animals, Structure–activity relationship, Tissue Distribution, Molecular Biology, Alkyl, Cholecystokinin, chemistry.chemical_classification, Benzodiazepinones, Molecular Structure, Chemistry, Organic Chemistry, Stereoisomerism, Receptor, Cholecystokinin B, Rats, Cholecystokinin B receptor, Molecular Medicine, Lead compound, Derivative (chemistry)
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3
المؤلفون: Fabio Maria Sabbatini, Daniele Donati, Stefania Faedo, Carla Marchioro, Fabrizio Micheli, Monica Viziano, Sylvie Gehanne, Giorgio Tarzia, Micaela Maffeis, Maria Elvira Tranquillini, Paolo Cavanni, Romano Di Fabio
المصدر: Il Farmaco. 58:1005-1009
مصطلحات موضوعية: Scaffold, Stereochemistry, Pharmaceutical Science, CHO Cells, Thiophenes, Receptors, Metabotropic Glutamate, Ring (chemistry), Binding, Competitive, Chemical synthesis, Inhibitory Concentration 50, Mice, Structure-Activity Relationship, chemistry.chemical_compound, Cricetinae, Drug Discovery, Benzene Derivatives, Animals, Pyrroles, Pain Measurement, Pyrrole, Nociceptors, Esters, Biological activity, Analgesics, Non-Narcotic, Rats, Spinal Cord, chemistry, Metabotropic glutamate receptor 1, Bioisostere, Selectivity
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4
المصدر: Il Farmaco. 53:49-54
مصطلحات موضوعية: Bicyclic molecule, Stereochemistry, Diastereomer, Pharmaceutical Science, Stereoisomerism, Receptor, Cholecystokinin B, Stereocenter, Benzodiazepines, Structure-Activity Relationship, chemistry.chemical_compound, Chain (algebraic topology), chemistry, Drug Discovery, Lactam, Receptors, Cholecystokinin, Enantiomer
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5
المؤلفون: Giorgio Pentassuglia, Stefano Polinelli, Daniele Donati, Gabriella Finizia, Giorgio Tarzia, Maria Elvira Tranquillini, Antonella Ursini
المصدر: Archiv der Pharmazie. 331:41-44
مصطلحات موضوعية: Bicyclic molecule, Chemistry, Stereochemistry, Guinea Pigs, Pharmaceutical Science, In Vitro Techniques, Ligands, Chemical synthesis, Receptor, Cholecystokinin B, Benzodiazepines, chemistry.chemical_compound, Drug Discovery, Lactam, Animals, Receptors, Cholecystokinin, Selectivity, Biological evaluation
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::4743a8a043b0fe7415ecdf7953f0dc70
https://doi.org/10.1002/(sici)1521-4184(199801)331:1<41::aid-ardp41>3.0.co;2-s -
6
المؤلفون: Gabriella Finizia, Daniele Donati, Paolo G. Cassarà, A. Ursini, Giovanni Curotto, S. Polinelli, Giorgio Tarzia, F. T. M. Van Amsterdam, Giorgio Pentassuglia, Mauro Corsi, Maria Elvira Tranquillini
المصدر: Archiv der Pharmazie. 330:353-357
مصطلحات موضوعية: Bicyclic molecule, Hydrocarbons, Halogenated, Chemistry, Ligand, Stereochemistry, Aryl, Guinea Pigs, Pharmaceutical Science, Stereoisomerism, Ligands, Ring (chemistry), Chemical synthesis, Receptor, Cholecystokinin B, Benzodiazepines, Kinetics, Structure-Activity Relationship, chemistry.chemical_compound, Drug Discovery, Halogen, Lactam, Animals, Receptors, Cholecystokinin
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7
المؤلفون: Beatrice Oliosi, Antonella Ursini, Daniele Donati, Maria Elvira Tranquillini, Gabriella Finizia
المصدر: Bioorganic & Medicinal Chemistry Letters. 6:2957-2962
مصطلحات موضوعية: chemistry.chemical_classification, Stereochemistry, Organic Chemistry, Clinical Biochemistry, Substitution (logic), Pharmaceutical Science, Biochemistry, chemistry, Drug Discovery, Molecular Medicine, Receptor, Molecular Biology, Alkyl, Biological evaluation
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8
المؤلفون: Gian Luca Araldi, Giorgio Pentassuglia, Antonella Ursini, Maria Elvira Tranquillini, A. Pezzoli, Daniele Donati
المصدر: Bioorganic & Medicinal Chemistry Letters. 6:1683-1688
مصطلحات موضوعية: chemistry.chemical_compound, chemistry, Organic Chemistry, Clinical Biochemistry, Drug Discovery, Pharmaceutical Science, Molecular Medicine, Epoxide, Organic chemistry, Antimicrobial, Molecular Biology, Biochemistry, Combinatorial chemistry
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9
المؤلفون: Gabriella Finizia, Beatrice Oliosi, Antonella Ursini, Maria Elvira Tranquillini, Daniele Donati
المصدر: ChemInform. 28
مصطلحات موضوعية: chemistry.chemical_classification, Stereochemistry, Chemistry, Substitution (logic), General Medicine, Receptor, Alkyl, Biological evaluation
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10
المؤلفون: Giorgio Tarzia, Antonella Ursini, Maria Elvira Tranquillini, Gabriella Finizia, Daniele Donati, Giorgio Pentassuglia, Stefano Polinelli
المصدر: ChemInform. 29
مصطلحات موضوعية: Chemistry, Stereochemistry, General Medicine, Receptor, Biological evaluation