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1
المؤلفون: Yoko Shimizu, S.-H. Sheldon Tai, Nag S. Kumar, Michel Roberge, Elyse Bourque, Masahiro Niikura, Olga Agafitei, James Brian Jaquith, Fahimeh S. Shidmoossavee, Steve Arns, Aruna D. Balgi, Tom A. Pfeifer, Sharon Sun
المصدر: European Journal of Medicinal Chemistry. 120:64-73
مصطلحات موضوعية: 0301 basic medicine, Mutant, 010402 general chemistry, Antiviral Agents, 01 natural sciences, Virus, Microbiology, Small Molecule Libraries, Viral Matrix Proteins, Structure-Activity Relationship, 03 medical and health sciences, Influenza, Human, Drug Discovery, Amantadine, medicine, Humans, Potency, Pharmacology, biology, Chemistry, Organic Chemistry, Influenza a, General Medicine, Yeast, 0104 chemical sciences, 030104 developmental biology, M2 proton channel, Influenza A virus, Mutation, biology.protein, Protons, medicine.drug, Cell based
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2
المؤلفون: Renato Skerlj, Tuya Ba, Ernest J. McEachern, Elyse Bourque, Ian Baird, Dominique Schols, Wilson Trevor R, Renee Mosi, Jonathan Langille, Yuanxi Zhou, Bryon Carpenter, Michael Bey, Simon P. Fricker, Dana Huskens, Duane Veale, Rebecca S.Y. Wong, Gary Bridger, Curtis Harwig, Veronique Bodart, Ron MacFarland, Markus Metz, Sanjay Danthi
المصدر: ACS Medicinal Chemistry Letters. 3:216-221
مصطلحات موضوعية: congenital, hereditary, and neonatal diseases and abnormalities, biology, business.industry, Purkinje fibers, Organic Chemistry, hERG, Human immunodeficiency virus (HIV), Pharmacology, medicine.disease_cause, Biochemistry, Bioavailability, Chemokine receptor, medicine.anatomical_structure, Drug Discovery, Lipophilicity, biology.protein, Medicine, Action potential duration, cardiovascular diseases, business, Ion channel
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3
المؤلفون: Renato Skerlj, Gary Bridger, Yuanxi Zhou, Elyse Bourque, Ernest McEachern, Jonathan Langille, Curtis Harwig, Duane Veale, Wen Yang, Tongshong Li, Yongbao Zhu, Michael Bey, Ian Baird, Michael Sartori, Markus Metz, Renee Mosi, Kim Nelson, Veronique Bodart, Rebecca Wong, Simon Fricker, Ron Mac Farland, Dana Huskens, Dominique Schols
المصدر: Bioorganic & Medicinal Chemistry Letters. 21:6950-6954
مصطلحات موضوعية: Tertiary amine, Anti-HIV Agents, Pyridines, medicine.drug_class, Stereochemistry, Clinical Biochemistry, Pharmaceutical Science, Carboxamide, CCR5 receptor antagonist, Pharmacology, Virus Replication, Biochemistry, Peripheral blood mononuclear cell, Chemical synthesis, Inhibitory Concentration 50, Dogs, Piperidines, Drug Discovery, medicine, Animals, Humans, Structure–activity relationship, Molecular Biology, Molecular Structure, Chemistry, Organic Chemistry, virus diseases, Amides, In vitro, Rats, Viral replication, Drug Design, CCR5 Receptor Antagonists, HIV-1, Leukocytes, Mononuclear, Molecular Medicine
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4
المؤلفون: Zefferino Santucci, Gary Bridger, Gloria Lau, Dominique Schols, Elyse Bourque, Wen Yang, Simon P. Fricker, Markus Metz, Curtis Harwig, Marilyn C. Darkes, Renato T. Skerlj, Jonathan Langille, Jean Labrecque, Sanjay Danthi
المصدر: Journal of the American Chemical Society. 133:16477-16485
مصطلحات موضوعية: Models, Molecular, Anti-HIV Agents, Stereochemistry, hERG, Allosteric regulation, Mutagenesis (molecular biology technique), Microbial Sensitivity Tests, Computational biology, CCR5 receptor antagonist, Biochemistry, Catalysis, Structure-Activity Relationship, Colloid and Surface Chemistry, medicine, Humans, Urea, Structure–activity relationship, Dose-Response Relationship, Drug, Molecular Structure, biology, Chemistry, Stereoisomerism, General Chemistry, Small molecule, Ether-A-Go-Go Potassium Channels, Entry inhibitor, Molecular Weight, Mutagenesis, Drug Design, CCR5 Receptor Antagonists, HIV-1, Leukocytes, Mononuclear, biology.protein, Pharmacophore, medicine.drug
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5
المؤلفون: Renato Skerlj, Gary Bridger, Yuanxi Zhou, Elyse Bourque, Jonathan Langille, Maria Di Fluri, David Bogucki, Wen Yang, Tongshuang Li, Letian Wang, Susan Nan, Ian Baird, Markus Metz, Marilyn Darkes, Jean Labrecque, Gloria Lau, Simon Fricker, Dana Huskens, Dominique Schols
المصدر: Bioorganic & Medicinal Chemistry Letters. 21:2450-2455
مصطلحات موضوعية: Receptors, CCR5, Pyridines, Organic Chemistry, Clinical Biochemistry, Pharmaceutical Science, Virus Replication, Amides, Biochemistry, Rats, Cyclic N-Oxides, Structure-Activity Relationship, Dogs, Piperidines, Drug Design, CCR5 Receptor Antagonists, Oximes, Drug Discovery, HIV-1, Animals, Humans, Molecular Medicine, Molecular Biology
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6
المؤلفون: Adam Galey, Stephen G. Withers, Natalia Zisman, Jenna Udechukwu, Jay Paquette, Jason Samuel Tan, Elyse Bourque, Samantha Dercho, Richard Liggins, Fiona C. Ross, Sharon Sun, Murray S. Webb, Vionarica Gusti, Steve Arns
المصدر: Bioorganicmedicinal chemistry letters. 25(12)
مصطلحات موضوعية: Oseltamivir, medicine.drug_class, Clinical Biochemistry, Pharmaceutical Science, Administration, Oral, Biological Availability, Neuraminidase, Pharmacology, 010402 general chemistry, 01 natural sciences, Biochemistry, chemistry.chemical_compound, Mice, Viral Proteins, Pharmacokinetics, Drug Discovery, medicine, Viral neuraminidase, Animals, Prodrugs, Enzyme Inhibitors, Molecular Biology, Neuraminidase inhibitor, biology, 010405 organic chemistry, Organic Chemistry, Screening assay, Prodrug, 0104 chemical sciences, 3. Good health, Bioavailability, chemistry, biology.protein, Sialic Acids, Molecular Medicine, Half-Life
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7
المؤلفون: Josephine Yuen, Philip J. Kocienski, Elyse Bourque, Michael J. Stocks
المصدر: Synthesis. :3219-3224
مصطلحات موضوعية: Stereochemistry, Fragment (computer graphics), Organic Chemistry, Tetronasin, Cationic polymerization, chemistry.chemical_element, General Medicine, Combinatorial chemistry, Copper, Catalysis, chemistry.chemical_compound, Fragment (logic), chemistry, Molybdenum, Tetrahydrofuran
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::c4167c3f1b44acaccf9201cc317433c5
https://doi.org/10.1055/s-2005-918486 -
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المؤلفون: Elyse Bourque, Yves L. Dory, Pierre Deslongchamps
المصدر: The Journal of Organic Chemistry. 68:2390-2397
مصطلحات موضوعية: chemistry.chemical_classification, chemistry.chemical_compound, Ketone, chemistry, Computational chemistry, Organic Chemistry, Photochemistry, Enone, Diels–Alder reaction
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9
المؤلفون: Tom Wennekes, Jay Paquette, Richard Liggins, Natalia Zisman, Adam Galey, Steve Arns, Stephen G. Withers, Elyse Bourque, Murray S. Webb, Samantha Dercho, Vionarica Gusti, Fiona C. Ross, Sharon Sun, Jason Samuel Tan, Jenna Udechukwu
المصدر: Bioorganic & Medicinal Chemistry Letters. 26:3830
مصطلحات موضوعية: Chemistry, Organic Chemistry, Clinical Biochemistry, Pharmaceutical Science, Screening assay, Prodrug, Pharmacology, Biochemistry, Clinical biochemistry, Bioavailability, Drug Discovery, Viral neuraminidase, Molecular Medicine, Molecular Biology
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10
المؤلفون: Curtis Harwig, Dominique Schols, Gang Chen, Wen Yang, Duane Veale, Susan Nan, Simon P. Fricker, Alan Kaller, Danielle Guay, Jason M. Crawford, Michael Satori, Markus Metz, Yongbao Zhu, Helen Yee, Maria Krumpak, Elyse Bourque, Wilson Trevor R, David Bogucki, Bryon Carpenter, Michael Bey, David C. Leitch, Ron MacFarland, David Gauthier, Ian Baird, Rebecca Wong, Renato T. Skerlj, Jonathan Langille, Yuanxi Zhou, Gary Bridger, Renee Mosi, Ernest J. McEachern, Tuya Ba, Tong-Shuang Li, Krystyna Vocadlo, Veronique Bodart
المصدر: Journal of medicinal chemistry. 56(20)
مصطلحات موضوعية: Receptors, CCR5, Anti-HIV Agents, Cell Survival, hERG, Human immunodeficiency virus (HIV), CHO Cells, Pharmacology, medicine.disease_cause, Imidazolidines, Virus Replication, Benzoates, Chemokine receptor, Structure-Activity Relationship, Cricetulus, Piperidines, In vivo, Cricetinae, Drug Discovery, medicine, Animals, Humans, Cells, Cultured, Cardiotoxicity, biology, Molecular Structure, Chemistry, Imidazoles, In vitro, Receptor selectivity, HEK293 Cells, Biochemistry, Models, Chemical, Drug Design, Lipophilicity, CCR5 Receptor Antagonists, Host-Pathogen Interactions, biology.protein, HIV-1, Leukocytes, Mononuclear, Molecular Medicine