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المؤلفون: Thomas J. Connors, Jie Qian, Zeck Huang, Joanne R. Mathiasen, Edward R. Bacon, Thelma S. Angeles, Mark J. Huffman, Emir Duzic, Joseph M. Salvino, Beth Ann McKenna, Hervé Schaffhauser, Robert J. McHugh, Lily D. Lu, George C. Morton, Beverly P. Holskin, Karla Kopec, Amy DiCamillo, Gerard C. Rosse, Chrysanthe Spais, Rabindranath Tripathy, Lisa D. Aimone
المصدر: Bioorganic & Medicinal Chemistry Letters. 22:1421-1426
مصطلحات موضوعية: Stereochemistry, Chemistry, Organic Chemistry, Clinical Biochemistry, Antagonist, Pharmaceutical Science, Stereoisomerism, Biochemistry, Sulfone, chemistry.chemical_compound, In vivo, Drug Discovery, 5-HT6 receptor, Molecular Medicine, Pharmacophore, Receptor, Molecular Biology, 5-HT receptor
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المؤلفون: Beverly P. Holskin, Karla Kopec, Joanne R. Mathiasen, Amy DiCamillo, Babu G. Sundar, Thomas J. Connors, Emir Duzic, Edward R. Bacon, Gerard C. Rosse, Chrysanthe Spais, Thomas R. Bailey, Beth Ann McKenna, Rebecca A. Brown, Jie Qian, Derek Dunn, Mark J. Huffman, Joseph M. Salvino, Huang Zeqi, Lisa D. Aimone, Hervé Schaffhauser, Deborah Galinis, Thelma S. Angeles, Lily D. Lu, George C. Morton
المصدر: Bioorganic & Medicinal Chemistry Letters. 22:120-123
مصطلحات موضوعية: biology, Organic Chemistry, Clinical Biochemistry, hERG, Pharmaceutical Science, Pharmacology, Biochemistry, Social recognition, chemistry.chemical_compound, chemistry, Drug Discovery, biology.protein, 5-HT6 receptor, Molecular Medicine, Structure–activity relationship, Serotonin Antagonists, Penetrant (biochemical), Receptor, Molecular Biology, 5-HT receptor
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المؤلفون: Emir Duzic, Edward R. Bacon, Joanne R. Mathiasen, Michael J. Marino, Donna Bozyczko-Coyne, John A. Gruner, John P. Mallamo, Rita Raddatz, Dorothy G. Flood, Lisa D. Aimone, Hervé Schaffhauser, Siyuan Le, Maciej Gasior, Michael Williams, Mark A. Ator, Robert L. Hudkins
المصدر: Journal of Pharmacology and Experimental Therapeutics. 340:124-133
مصطلحات موضوعية: Pharmacology, Agonist, Chemistry, medicine.drug_class, Antagonist, Receptor antagonist, Dose–response relationship, chemistry.chemical_compound, medicine, Molecular Medicine, Inverse agonist, Receptor, Ex vivo, Histamine
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_________::d821744703207b55845570e2612fea8e
https://doi.org/10.1124/jpet.111.186585 -
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المؤلفون: Michael Williams, Emir Duzic, Michael J. Marino
المصدر: Burger's Medicinal Chemistry and Drug Discovery. :499-548
مصطلحات موضوعية: Chemistry, Drug discovery, Computational biology, Receptor
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_________::8a3bba92664cb3ff3510fc7cac14c559
https://doi.org/10.1002/0471266949.bmc029.pub2 -
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المؤلفون: Beverly P. Holskin, Sheryl L. Meyer, Emmanuel Burgeon, Bruce Jones, Thao Ung, Emir Duzic, Sandra Y. Flores, Mark A. Ator, Vincent J. Dupriez
المصدر: Analytical Biochemistry. 400:184-189
مصطلحات موضوعية: Biophysics, Aequorin, Photoprotein, Digitonin, CHO Cells, Transfection, Biochemistry, Receptors, G-Protein-Coupled, law.invention, Cricetulus, law, Cricetinae, Animals, Humans, Receptor, Molecular Biology, G protein-coupled receptor, Cryopreservation, biology, Oxotremorine, Receptor, Muscarinic M1, Cell Biology, Acetylcholine, Cell biology, Cell culture, biology.protein, Recombinant DNA, Calcium, Function (biology)
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المؤلفون: Aya Takesono, Stephen M. Lanier, Mary Cismowski, Mark W. Nowak, Emir Duzic
المصدر: Journal of Biological Chemistry. 277:13827-13830
مصطلحات موضوعية: GTP-binding protein regulators, G protein, Heterotrimeric G protein, Cell Biology, G protein-coupled inwardly-rectifying potassium channel, Signal transduction, Biology, Receptor, Molecular Biology, Biochemistry, Muscarinic agonist, Cell biology, G protein-coupled receptor
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_________::650e900fd3c54829e3948acc58637b6d
https://doi.org/10.1074/jbc.m201064200 -
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المؤلفون: Glenn E. Kirsch, Arthur Brown, Emir Duzic, Yuri A. Kuryshev
المصدر: Assay and Drug Development Technologies
مصطلحات موضوعية: CHO Cells, Biology, Pharmacology, Membrane Potentials, Cricetulus, Automated patch clamp, Cricetinae, Drug Discovery, medicine, Animals, Humans, Membrane potential, Voltage-dependent calcium channel, Dose-Response Relationship, Drug, Calcium channel, HEK 293 cells, Original Articles, Calcium Channel Blockers, Electrophysiological Phenomena, Electrophysiology, HEK293 Cells, Mechanism of action, cardiovascular system, Molecular Medicine, Drug Evaluation, Calcium Channels, medicine.symptom, Muscle contraction
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::1ed5d140febc1782333336fa9f36cfce
https://pubmed.ncbi.nlm.nih.gov/24579774 -
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المؤلفون: Michael Spruyt, Stephen M. Lanier, Jeffrey S. Lizano, Mary J. Cismowski, Xiaobing Xie, Catalina Ribas, Chienling Ma, Emir Duzic
المصدر: Journal of Biological Chemistry. 275:23421-23424
مصطلحات موضوعية: Gs alpha subunit, Activator (genetics), Gi alpha subunit, macromolecular substances, Cell Biology, Biology, Biochemistry, Yeast, Cell biology, Heterotrimeric G protein, Guanine nucleotide exchange factor, Signal transduction, Ras superfamily, Molecular Biology
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_________::96cc7c3e2e77a10fae6d8031d774ad74
https://doi.org/10.1074/jbc.c000322200 -
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المؤلفون: Karl E.O. Åkerman, Stephen M. Lanier, Sanna Soini, Emir Duzic
المصدر: Pfl�gers Archiv European Journal of Physiology. 435:280-285
مصطلحات موضوعية: Agonist, Patch-Clamp Techniques, Nifedipine, Physiology, medicine.drug_class, Clinical Biochemistry, Rauwolscine, 8-Bromo Cyclic Adenosine Monophosphate, Pharmacology, Transfection, Pertussis toxin, PC12 Cells, chemistry.chemical_compound, GTP-Binding Proteins, Physiology (medical), Cyclic AMP, medicine, Animals, Channel blocker, Virulence Factors, Bordetella, Patch clamp, Adrenergic alpha-Antagonists, Neurons, Calcium channel, Electric Conductivity, Imidazoles, T-type calcium channel, Dihydropyridine, Yohimbine, Medetomidine, Receptors, Adrenergic, alpha, Calcium Channel Blockers, Recombinant Proteins, Rats, Pertussis Toxin, chemistry, Biophysics, Calcium Channels, Adrenergic alpha-Agonists, medicine.drug
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المؤلفون: Emir Duzic, Toshiaki Ebina, Naoki Oka, Jun-ichi Kawabe, Yoshihiro Ishikawa, Carsten Schwencke, Yoshiyuki Toya
المصدر: FEBS Letters. 384:273-276
مصطلحات موضوعية: Phorbol ester, Time Factors, Molecular Sequence Data, Biophysics, Kidney, Transfection, Biochemistry, ADCY10, Adenylyl cyclase, chemistry.chemical_compound, Alkaloids, Structural Biology, Cyclic AMP, Genetics, medicine, Humans, Insulin, Staurosporine, Enzyme Inhibitors, Protein kinase A, Adenylylcyclase, Molecular Biology, Cells, Cultured, Protein Kinase C, Protein kinase C, Dose-Response Relationship, Drug, Kinase, Activator (genetics), ADCY9, Cell Biology, Molecular biology, Enzyme Activation, Isoenzymes, chemistry, Tetradecanoylphorbol Acetate, Adenylyl Cyclases, medicine.drug