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1دورية أكاديمية
المؤلفون: Panagiotis Kanellopoulos, Emmanouil Lymperis, Aikaterini Kaloudi, Marion de Jong, Eric P. Krenning, Berthold A. Nock, Theodosia Maina
المصدر: Molecules, Vol 25, Iss 15, p 3418 (2020)
مصطلحات موضوعية: gastrin-releasing peptide receptor targeting, [99mTc]Tc-radiotracer, tumor targeting, [99mTc]Tc-DB1 mimic, PEGx-spacer, neprilysin-inhibition, Organic chemistry, QD241-441
وصف الملف: electronic resource
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2دورية أكاديمية
المؤلفون: Emmanouil Lymperis, Aikaterini Kaloudi, Panagiotis Kanellopoulos, Marion de Jong, Eric P. Krenning, Berthold A. Nock, Theodosia Maina
المصدر: Molecules, Vol 24, Iss 6, p 1015 (2019)
مصطلحات موضوعية: GRPR-antagonist, bombesin-like radioligand, tumor targeting, tumor imaging, neprilysin-inhibition, phosphoramidon, in vivo stability, Organic chemistry, QD241-441
وصف الملف: electronic resource
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3دورية أكاديمية
المؤلفون: Aikaterini Kaloudi, Emmanouil Lymperis, Panagiotis Kanellopoulos, Beatrice Waser, Marion de Jong, Eric P. Krenning, Jean Claude Reubi, Berthold A. Nock, Theodosia Maina
المصدر: Pharmaceuticals, Vol 12, Iss 1, p 42 (2019)
مصطلحات موضوعية: bombesin, gastrin-releasing peptide, gastrin-releasing peptide receptor, tumor targeting, 99mTc-radioligand, metabolic stability, neprilysin-inhibition, phosphoramidon, Medicine, Pharmacy and materia medica, RS1-441
وصف الملف: electronic resource
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4دورية أكاديمية
المؤلفون: Aikaterini Kaloudi, Emmanouil Lymperis, Athina Giarika, Simone Dalm, Francesca Orlandi, Donato Barbato, Mattia Tedesco, Theodosia Maina, Marion de Jong, Berthold A. Nock
المصدر: Molecules, Vol 22, Iss 11, p 1950 (2017)
مصطلحات موضوعية: GRPR-antagonist, theragnostics, targeted tumor imaging, PET-imaging, breast cancer, Organic chemistry, QD241-441
وصف الملف: electronic resource
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5
المؤلفون: Theodosia Maina, Berthold A. Nock, Aikaterini Kaloudi, Panagiotis Kanellopoulos, Eric P. Krenning, Marion de Jong, Emmanouil Lymperis
المساهمون: Radiology & Nuclear Medicine
المصدر: Journal of Labelled Compounds & Radiopharmaceuticals, 62(10), 646-655. John Wiley & Sons Ltd.
مصطلحات موضوعية: Agonist, medicine.drug_class, Pharmacology, 01 natural sciences, Biochemistry, 030218 nuclear medicine & medical imaging, Analytical Chemistry, 03 medical and health sciences, chemistry.chemical_compound, 0302 clinical medicine, SDG 3 - Good Health and Well-being, In vivo, Drug Discovery, medicine, Radioligand, Radiology, Nuclear Medicine and imaging, Receptor, Neprilysin, Spectroscopy, 010405 organic chemistry, Chemistry, Organic Chemistry, Phosphoramidon, Antagonist, Bombesin, 0104 chemical sciences
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6
المؤلفون: Theodosia Maina, Panagiotis Kanellopoulos, Eric P. Krenning, Emmanouil Lymperis, Aikaterini Kaloudi, Berthold A. Nock, Marion de Jong
المساهمون: Radiology & Nuclear Medicine, Erasmus MC other
المصدر: Molecules
Volume 25
Issue 15
Molecules, 25(15):3418. Multidisciplinary Digital Publishing Institute (MDPI)
Molecules, Vol 25, Iss 3418, p 3418 (2020)مصطلحات موضوعية: Male, Cell, Pharmaceutical Science, Peptide, Mice, SCID, Pharmacology, 030218 nuclear medicine & medical imaging, Analytical Chemistry, gastrin-releasing peptide receptor targeting, Mice, chemistry.chemical_compound, 0302 clinical medicine, Biomimetic Materials, Drug Discovery, Receptor, Neprilysin, chemistry.chemical_classification, [99mTc]Tc-radiotracer, PEGx-spacer, Organotechnetium Compounds, Neoplasm Proteins, medicine.anatomical_structure, Chemistry (miscellaneous), 030220 oncology & carcinogenesis, PC-3 Cells, Molecular Medicine, phosphoramidon, Biodistribution, [99mTc]Tc-DB1 mimic, Antineoplastic Agents, Article, lcsh:QD241-441, 03 medical and health sciences, lcsh:Organic chemistry, In vivo, PEG ratio, medicine, Animals, Humans, Physical and Theoretical Chemistry, tumor targeting, Organic Chemistry, Phosphoramidon, Prostatic Neoplasms, Xenograft Model Antitumor Assays, Receptors, Bombesin, chemistry, Peptides, neprilysin-inhibition
وصف الملف: application/pdf
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7
المؤلفون: Aikaterini, Kaloudi, Emmanouil, Lymperis, Panagiotis, Kanellopoulos, Beatrice, Waser, Marion, de Jong, Eric P, Krenning, Jean Claude, Reubi, Berthold A, Nock, Theodosia, Maina
المصدر: Pharmaceuticals
مصطلحات موضوعية: phosphoramidon, bombesin, 99mTc-radioligand, tumor targeting, gastrin-releasing peptide receptor, hormones, hormone substitutes, and hormone antagonists, Article, gastrin-releasing peptide, metabolic stability, neprilysin-inhibition
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8
المؤلفون: Theodosia Maina, Eric P. Krenning, Panagiotis Kanellopoulos, Marion de Jong, Aikaterini Kaloudi, Berthold A. Nock, Emmanouil Lymperis
المساهمون: Radiology & Nuclear Medicine
المصدر: Molecules, 24(6):1015. Multidisciplinary Digital Publishing Institute (MDPI)
Molecules
Volume 24
Issue 6
Molecules, Vol 24, Iss 6, p 1015 (2019)مصطلحات موضوعية: Male, Cell, in vivo stability, Pharmaceutical Science, Peptide, Pharmacology, 030218 nuclear medicine & medical imaging, Analytical Chemistry, chemistry.chemical_compound, Prostate cancer, Mice, 0302 clinical medicine, Drug Stability, Drug Discovery, Tissue Distribution, Neprilysin, bombesin-like radioligand, chemistry.chemical_classification, Chemistry, Indium Radioisotopes, Glycopeptides, medicine.anatomical_structure, Chemistry (miscellaneous), 030220 oncology & carcinogenesis, Molecular Medicine, Bombesin, phosphoramidon, Article, lcsh:QD241-441, 03 medical and health sciences, lcsh:Organic chemistry, In vivo, Cell Line, Tumor, medicine, Pi, Animals, Humans, Physical and Theoretical Chemistry, IC50, Biosimilar Pharmaceuticals, GRPR-antagonist, tumor targeting, tumor imaging, Organic Chemistry, Phosphoramidon, Prostatic Neoplasms, Trastuzumab, medicine.disease, Receptors, Bombesin, neprilysin-inhibition
وصف الملف: application/pdf
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9
المؤلفون: Jean Claude Reubi, Eric P. Krenning, Theodosia Maina, Berthold A. Nock, Aikaterini Kaloudi, Beatrice Waser, Marion de Jong, Panagiotis Kanellopoulos, Emmanouil Lymperis
المساهمون: Radiology & Nuclear Medicine
المصدر: Pharmaceuticals, Vol 12, Iss 1, p 42 (2019)
Pharmaceuticals
Volume 12
Issue 1
Kaloudi, Aikaterini; Lymperis, Emmanouil; Kanellopoulos, Panagiotis; Waser, Beatrice; de Jong, Marion; Krenning, Eric P; Reubi, Jean Claude; Nock, Berthold A; Maina, Theodosia (2019). Localization of 99mTc-GRP Analogs in GRPR-Expressing Tumors: Effects of Peptide Length and Neprilysin Inhibition on Biological Responses. Pharmaceuticals, 12(1) MDPI 10.3390/ph12010042 <http://dx.doi.org/10.3390/ph12010042>
Pharmaceuticals, 12(1):Unsp 42. Multidisciplinary Digital Publishing Institute (MDPI)مصطلحات موضوعية: 0301 basic medicine, phosphoramidon, gastrin-releasing peptide receptor, Pharmaceutical Science, lcsh:Medicine, lcsh:RS1-441, 610 Medicine & health, gastrin-releasing peptide, metabolic stability, lcsh:Pharmacy and materia medica, 03 medical and health sciences, chemistry.chemical_compound, 0302 clinical medicine, In vivo, Spect imaging, Gastrin-releasing peptide, Drug Discovery, Gastrin-releasing peptide receptor, Receptor, Neprilysin, Chemistry, tumor targeting, Phosphoramidon, lcsh:R, Bombesin, 99mTc-radioligand, 030104 developmental biology, bombesin, 030220 oncology & carcinogenesis, Cancer research, Molecular Medicine, 570 Life sciences, biology, hormones, hormone substitutes, and hormone antagonists, neprilysin-inhibition
وصف الملف: application/pdf
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10
المؤلفون: Emmanouil, Lymperis, Aikaterini, Kaloudi, Panagiotis, Kanellopoulos, Eric P, Krenning, Marion, de Jong, Theodosia, Maina, Berthold A, Nock
المصدر: Journal of labelled compoundsradiopharmaceuticalsREFERENCES. 62(10)
مصطلحات موضوعية: Male, Receptors, Bombesin, Heterocyclic Compounds, 1-Ring, Mice, Drug Stability, Indium Radioisotopes, PC-3 Cells, Animals, Humans, Prostatic Neoplasms, Biological Transport, Tissue Distribution, Oligopeptides