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1
المؤلفون: Chun-wa Chung, Rab K. Prinjha, Rejbinder Kaur, Peter Ernest Soden, Ann Louise Walker, Van Loc Nguyen, Christophe Simon, Simon Taylor, Romain Luc Marie Gosmini, Jean-Marie Brusq, Antonia J. Lewis, Mark B. Schilling, Lionel Trottet, Matthew D. Walker, Leanne Cutler, Olivier Mirguet, Emmanuel Hubert Demont, Edwige Nicodeme, Eric Boursier, Jérôme Toum, Alizon M. Riou-Eymard, Gael Krysa, Hugh Clark, Paul Bamborough
المصدر: Journal of Medicinal Chemistry. 57:8111-8131
مصطلحات موضوعية: Anti-Inflammatory Agents, Regulator, Cell Cycle Proteins, Inflammation, Protein Serine-Threonine Kinases, Benzoates, Mice, Structure-Activity Relationship, Transcription (biology), Neuroblastoma, Drug Discovery, medicine, Animals, Humans, Histone code, Epigenetics, Gene, Genetics, Apolipoprotein A-I, Chemistry, Nuclear Proteins, medicine.disease, Bromodomain, Aminoquinolines, Quinolines, Cancer research, Molecular Medicine, medicine.symptom, Transcription Factors
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2
المؤلفون: Svetlana L. Belyanskaya, Chun-wa Chung, Eric Humphries, Christopher S. Kollmann, Nicolas Ancellin, Christopher C. Arico-Muendel, Hongfeng Deng, Ryan P. Bingham, Van Loc Nguyen, Jeffrey A. Messer, Yun Ding, Emily Blazensky, Arthur Beljean, Anne-Benedicte Boullay, Sarah E. Smith, Jingye Zhou, Edwige Nicodeme, Jing Chai, Flora S. Sundersingh, Clare I. Hobbs, Alain Claude-Marie Daugan, Myriam Ajakane, Donald O. Somers, Nerina Dodic, Kenny Herry, Paul S. Carter, Eric Boursier
مصطلحات موضوعية: 0301 basic medicine, chemistry.chemical_classification, Benzimidazole, biology, Stereochemistry, Aryl, Organic Chemistry, Active site, Biochemistry, Amino acid, 03 medical and health sciences, chemistry.chemical_compound, 030104 developmental biology, chemistry, In vivo, Drug Discovery, biology.protein, Transferase, DNA
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::19d2b0e96f6386d1d5d0d6f742324e42
https://europepmc.org/articles/PMC4834658/ -
3
المؤلفون: Jean-François Mirjolet, Florent Potvain, Raphaelle Guillard-Huet, Guillaume Serin, Didier Grillot, Akanksha Gangar, Eric Boursier
المصدر: Cancer Research. 78:782-782
مصطلحات موضوعية: Cancer Research, Programmed cell death, biology, business.industry, Cell, Cancer, medicine.disease, medicine.anatomical_structure, Immune system, Oncology, Antigen, Apoptosis, Cancer cell, biology.protein, medicine, Cancer research, business, Calreticulin
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_________::48a0828a0909a71a277e6ed10ad0c0cb
https://doi.org/10.1158/1538-7445.am2018-782 -
4
المؤلفون: Laura J Pothier Kaushansky, Jennifer L. DeLorey, Hongfeng Deng, Christopher P. Davie, Jingye Zhou, Sarah E. Smith, Katie L Sargent Bedard, Christopher S. Kollmann, Barry A. Morgan, Nicolas Ancellin, Kenny Herry, Matthew A. Clark, Eric Boursier, Paul S. Carter, Clare I. Hobbs, Quan Zhou, Alexander L. Satz, Don O. Somers, Svetlana L. Belyanskaya, Jeffrey A. Messer, Yun Ding, Flora S. Sundersingh, Arthur Beljean, Chun-wa Chung, Ryan P. Bingham, LaShadric C. Grady, Christopher C. Arico-Muendel, G Joseph Franklin, Paolo A. Centrella, Jennifer Summerfield
مصطلحات موضوعية: biology, Stereochemistry, Organic Chemistry, A protein, Biochemistry, Combinatorial chemistry, Cofactor, chemistry.chemical_compound, Protein structure, chemistry, Drug Discovery, biology.protein, Transferase, DNA
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::f1887eff01483569c140544dbed75f5c
https://europepmc.org/articles/PMC4538436/ -
5
المؤلفون: Ian Churcher, Sarah E. Smith, Ryan P. Bingham, Clare I. Hobbs, Donald O. Somers, Eric Boursier, Chun Wa Chung, Charlène Fournier, Yoshiaki Washio, Peter Francis, Claus Spitzfaden, Iain H. Reid, Stephen D. Pickett, Sophie M. Bertrand, Graham L. Simpson, Andrew N. Hobbs, Klára Valkó, Laura A. Gummer, Robert J. Young, Nicolas Ancellin, Craig Jamieson, Colin J. Suckling, Anne Bénédicte Boullay, Lisa A. Sloan, Kenny Herry, Paul S. Carter, Nerina Dodic, Paul Homes, Edwige Nicodeme, Jennifer A. Borthwick, Benjamin Beaufils, Marie Helene Fouchet
المصدر: Journal of medicinal chemistry. 58(18)
مصطلحات موضوعية: Models, Molecular, Branched chain aminotransferase, Pyrimidinones, Crystallography, X-Ray, Mitochondrial Proteins, Structure-Activity Relationship, Valine, Leucine, Drug Discovery, Adipocytes, Structure–activity relationship, Transferase, Animals, Humans, Isoleucine, Transaminases, chemistry.chemical_classification, Mice, Inbred BALB C, Ligand efficiency, Chemistry, Molecular biology, Amino acid, Mice, Inbred C57BL, Biochemistry, Molecular Medicine, Pyrazoles
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6
المؤلفون: Jean-Marie Brusq, Pascal Grondin, Benjamin Beaufils, Frédéric Donche, Stéphane Sautet, Celine Marques, Edwige Nicodeme, Yann Dudit, Catherine-Anne Clément, Pascal Huet, Yannick Saintillan, Eric Boursier, Jérôme Toum, Mathieu Pizzonero, Emilie Rondet, Lionel Trottet, Olivier Mirguet
مصطلحات موضوعية: chemistry.chemical_classification, medicine.medical_specialty, business.industry, Organic Chemistry, AMPK, Type 2 diabetes, medicine.disease, Biochemistry, Proinflammatory cytokine, Endocrinology, Enzyme, Pharmacokinetics, chemistry, Internal medicine, Drug Discovery, Hyperlipidemia, medicine, business, Protein kinase A, Beta oxidation
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::8260bf96114fc481fec9048186ad6416
https://europepmc.org/articles/PMC4027520/ -
7
المؤلفون: Delphine Delannée, Agnès Costaz, Jonathan Thomas Seal, Lionel Trottet, Rémi Tellier, Jean-Marie Brusq, Olivier Mirguet, Anne Marie Jeanne Bouillot, Sandrine Martin, Gael Krysa, Anne-Benedicte Boullay, Jorge Kirilovsky, Eric Boursier, Jérôme Toum, Yann Dudit, Van-Loc Nguyen, Edwige Nicodeme, Françoise Gellibert, Alizon M. Riou, Pascal Huet, Romain Luc Marie Gosmini, Yann Lamotte, Florence Blandel, Frédéric Donche
المصدر: Bioorganicmedicinal chemistry letters. 22(8)
مصطلحات موضوعية: Clinical Biochemistry, Anti-Inflammatory Agents, Pharmaceutical Science, Nerve Tissue Proteins, Biochemistry, Chemical synthesis, Heterocyclic Compounds, 4 or More Rings, Inhibitory Concentration 50, Mice, Structure-Activity Relationship, Downregulation and upregulation, Drug Discovery, Structure–activity relationship, Animals, Humans, Histone Chaperones, Molecular Biology, Biological evaluation, Histone Acetyltransferases, Mice, Inbred BALB C, Apolipoprotein A-I, Chemistry, Drug discovery, Organic Chemistry, Nuclear Proteins, Hep G2 Cells, In vitro, Bromodomain, Cell biology, Rats, Up-Regulation, Immunology, Hepatic stellate cell, Quinolines, Molecular Medicine
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8
المؤلفون: Rab K. Prinjha, Helen R. Flynn, Stephen A. Hughes, Jérôme Toum, Rachel Grimley, Chun-wa Chung, Sandrine Martin, Jean-Marie Brusq, Hervé Coste, Kevin Lee, Chris J. Delves, Alizon M. Riou, Romain Luc Marie Gosmini, Catherine A. Clément, Edwige Nicodeme, Anne Marie Jeanne Bouillot, Eric Boursier, Robert Woodward, Anne-Benedicte Boullay, Olivier Mirguet, Jorge Kirilovsky, Paul Homes, Jonathan I. Wilde, Paul Bamborough, Iain Uings, Julia H. White, Françoise Gellibert, Emma J. Jones, Florence Blandel, Sylvie M. Magny
المصدر: Journal of medicinal chemistry. 54(11)
مصطلحات موضوعية: Epigenomics, Models, Molecular, BRD4, Protein family, Phenotypic screening, Molecular Sequence Data, Protein Serine-Threonine Kinases, Crystallography, X-Ray, Histones, Benzodiazepines, Drug Discovery, Humans, Chemoproteomics, Amino Acid Sequence, Molecular Targeted Therapy, Binding Sites, biology, Apolipoprotein A-I, Molecular Structure, Chemistry, Drug discovery, Lysine, Acetylation, Stereoisomerism, Hep G2 Cells, Small molecule, Bromodomain, Up-Regulation, Histone, Biochemistry, biology.protein, Molecular Medicine, Protein Binding, Transcription Factors
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9دورية أكاديمية
المؤلفون: Sophie M. Bertrand, Nicolas Ancellin, Benjamin Beaufils, Ryan P. Bingham, Jennifer A. Borthwick, Anne-Bénédicte Boullay, Eric Boursier, Paul S. Carter, Chun-wa Chung, Ian Churcher, Nerina Dodic, Marie-Hélène Fouchet, Charlène Fournier, PeterL. Francis, Laura A. Gummer, Kenny Herry, Andrew Hobbs, Clare I. Hobbs, Paul Homes, Craig Jamieson
المصدر: Journal of Medicinal Chemistry; Sep2015, Vol. 58 Issue 18, p7140-7163, 24p