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1
المؤلفون: Drago Sliskovic, Essenburg Ad, Joseph Armand Picard, J. F. Reindel, L. L. Minton, B.R. Krause, R. L. Stanfield, W. H. Roark
المصدر: Bioorganic & Medicinal Chemistry Letters. 6:713-718
مصطلحات موضوعية: chemistry.chemical_classification, Cholesterol, Organic Chemistry, Clinical Biochemistry, Pharmaceutical Science, Biological activity, Pharmacology, Biochemistry, Acyl transferase, chemistry.chemical_compound, Acyl-CoA, Enzyme, chemistry, Amide, Drug Discovery, Molecular Medicine, Bioassay, Molecular Biology, Ex vivo
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2
المؤلفون: T. L. Stoeber, R. L. Stanfield, W. H. Roark, Brian R. Krause, C. J. Blankley, Bharat K. Trivedi, J. A. Picard, Ann Holmes, Essenburg Ad, M. K. Shaw
المصدر: Journal of Medicinal Chemistry. 36:3300-3307
مصطلحات موضوعية: chemistry.chemical_classification, biology, Cholesterol, Anticholesteremic Agents, Sterol O-acyltransferase, In vitro, Structure-Activity Relationship, chemistry.chemical_compound, Enzyme, Biochemistry, chemistry, In vivo, Enzyme inhibitor, Drug Discovery, biology.protein, Urea, Molecular Medicine, Structure–activity relationship, Moiety, Carbanilides, Sterol O-Acyltransferase
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3
المؤلفون: Brian R. Krause, K. L. Hamelehle, T. L. Stoeber, Essenburg Ad, Bharat K. Trivedi, R. L. Stanfield
المصدر: Bioorganic & Medicinal Chemistry Letters. 3:259-262
مصطلحات موضوعية: Chemistry, Organic Chemistry, Clinical Biochemistry, Sterol O-acyltransferase, Pharmaceutical Science, Biochemistry, In vitro, Plasma cholesterol, In vivo, Drug Discovery, Molecular Medicine, lipids (amino acids, peptides, and proteins), Molecular Biology
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4
المؤلفون: Ann Holmes, Bruce D. Roth, C. J. Blankley, Essenburg Ad, K.A. Kieft, W. H. Roark, R. L. Stanfield, Bharat K. Trivedi, Brian R. Krause, Milton L. Hoefle
المصدر: Journal of Medicinal Chemistry. 35:1609-1617
مصطلحات موضوعية: Male, medicine.drug_class, Sterol O-acyltransferase, Alpha (ethology), Carboxamide, Cholesterol, Dietary, Structure-Activity Relationship, In vivo, Drug Discovery, medicine, Animals, Potency, IC50, Hypolipidemic Agents, chemistry.chemical_classification, Fatty acid, Rats, Inbred Strains, Rats, Cholesterol, Enzyme, chemistry, Biochemistry, Molecular Medicine, lipids (amino acids, peptides, and proteins), Rabbits, Sterol O-Acyltransferase
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5
المؤلفون: C.E. Augelli-Szafran, Essenburg Ad, B.R. Krause, R. L. Stanfield, Bharat K. Trivedi, R. F. Bousley, C. J. Blankley, K. L. Hamelehle, Bruce David Roth
المصدر: Journal of medicinal chemistry. 36(20)
مصطلحات موضوعية: Male, Stereochemistry, Sterol O-acyltransferase, Rats, Sprague-Dawley, chemistry.chemical_compound, Structure-Activity Relationship, Amide, Microsomes, Drug Discovery, Potency, Animals, Anilides, IC50, biology, Anticholesteremic Agents, Biological activity, Ketones, Oxime, Rats, Intestines, Cholesterol, chemistry, Enzyme inhibitor, Lactam, biology.protein, Molecular Medicine, Rabbits, Sterol O-Acyltransferase
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6دورية أكاديمية
لا يتم عرض هذه النتيجة على الضيوف.
تسجيل الدخول للوصول الكامل. -
7
المؤلفون: M. L. Hoefle, Holmes A, I. Nordin, J. M. Hinkley, R. W. Fleming, A. E. Werner, Cohen Dm, Essenburg Ad, Klutchko S, Blankley Cj
المصدر: Journal of Medicinal Chemistry. 29:1953-1961
مصطلحات موضوعية: Male, Stereochemistry, Molecular Conformation, Angiotensin-Converting Enzyme Inhibitors, Structure-Activity Relationship, In vivo, Tetrahydroisoquinolines, Drug Discovery, medicine, Animals, Potency, Sulfhydryl Compounds, Proline, Enalapril, biology, Chemistry, Quinapril, Rats, Inbred Strains, Angiotensin-converting enzyme, Isoquinolines, Small molecule, Rats, Biochemistry, Enzyme inhibitor, biology.protein, Molecular Medicine, medicine.drug
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8
المؤلفون: R. D. Smith, H. R. Kaplan, Robert F. Meyer, Essenburg Ad
المصدر: Journal of Medicinal Chemistry. 25:996-999
مصطلحات موضوعية: chemistry.chemical_classification, Oligopeptide, Hypertension, Renal, Chemical Phenomena, biology, Stereochemistry, Angiotensin-Converting Enzyme Inhibitors, Angiotensin-converting enzyme, Captopril, Tripeptide, Rats, Chemistry, Enzyme, chemistry, In vivo, Drug Discovery, biology.protein, medicine, Animals, Molecular Medicine, Binding site, Oligopeptides, IC50, medicine.drug
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9
المؤلفون: Francis G. Tinney, Elizabeth A. Lunney, Ronald G. Almquist, Milton L. Hoefle, Essenburg Ad, Robert F. Meyer, Ann Holmes, Ernest. Nicolaides, R. D. Smith, H. R. Kaplan
المصدر: Journal of medicinal chemistry. 24(8)
مصطلحات موضوعية: Male, Recrystallization (geology), Stereochemistry, Blood Pressure, Acylation, Structure-Activity Relationship, In vivo, Drug Discovery, Renin–angiotensin system, medicine, Animals, Teprotide, IC50, biology, Dose-Response Relationship, Drug, Chemistry, Angiotensin II, Diastereomer, Captopril, Angiotensin-converting enzyme, Dipeptides, Rats, biology.protein, Molecular Medicine, Oligopeptides, medicine.drug
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10دورية أكاديمية
لا يتم عرض هذه النتيجة على الضيوف.
تسجيل الدخول للوصول الكامل.