-
1
المؤلفون: Matthias M. Herth, Frank Roesch, Dianne E. Lee, Ulrich Schmitt, Christoph Hiemke, Markus Piel, Hartmut Lueddens, Fabian Debus, Hans-Georg Buchholz
المصدر: Neuropsychobiology. 63:183-190
مصطلحات موضوعية: Fluorine Radioisotopes, Pharmacology, Biology, Serotonergic, Blood–brain barrier, Mice, Piperidines, Pharmacokinetics, Cerebellum, medicine, Animals, Receptor, Serotonin, 5-HT2A, ATP Binding Cassette Transporter, Subfamily B, Member 1, Receptor, Biological Psychiatry, P-glycoprotein, Mice, Knockout, Brain uptake, Biological Transport, Ligand (biochemistry), Frontal Lobe, Fluorobenzenes, Psychiatry and Mental health, Neuropsychology and Physiological Psychology, medicine.anatomical_structure, Blood-Brain Barrier, Positron-Emission Tomography, biology.protein, Neuroscience
-
2
المؤلفون: Konrad J. Werhahn, Erwan Dupont, Mathias Schreckenberger, Hans-Georg Buchholz, Andreas Fellgiebel, Christian Landvogt, Julia Tillmanns, Heiko J. Luhmann, Peter Bartenstein, Paul Cumming, Heidrun Potschka, Axel Heimann, Fabian Debus, Igor Yakushev
المصدر: Epilepsia. 51:415-422
مصطلحات موضوعية: Male, Pyrrolidines, Dopamine, Receptors, Dopamine, Temporal lobe, Epilepsy, Neuroimaging, In vivo, Animals, Humans, Medicine, Brain Mapping, Receptors, Dopamine D2, business.industry, Pilocarpine, Receptors, Dopamine D3, Brain, medicine.disease, Corpus Striatum, Rats, Disease Models, Animal, Epilepsy, Temporal Lobe, Neurology, Dopamine receptor, Positron-Emission Tomography, Benzamides, Autoradiography, Neurology (clinical), business, Neuroscience, Preclinical imaging, Ex vivo, medicine.drug
-
3
المؤلفون: Ulrich Schmitt, Matthias M. Herth, Hartmut Lüddens, Markus Piel, Fabian Debus, Frank Rösch
المصدر: Nuclear Medicine and Biology. 36:447-454
مصطلحات موضوعية: Male, Cancer Research, Biodistribution, Pharmacology, chemistry.chemical_compound, Piperidines, In vivo, Animals, Humans, Receptor, Serotonin, 5-HT2A, Tissue Distribution, Radiology, Nuclear Medicine and imaging, Receptor, 5-HT receptor, Brain, Binding potential, Ligand (biochemistry), Rats, Fluorobenzenes, Radioactivity, chemistry, Positron-Emission Tomography, Altanserin, Biophysics, Autoradiography, Molecular Medicine, Ex vivo
-
4
المؤلفون: Vasko Kramer, Fabian Debus, Hartmut Lüddens, Matthias M. Herth, Nicole Bausbacher, Hans-Georg Buchholz, Frank Rösch, Markus Piel
المصدر: Nuclear medicine and biology. 37(4)
مصطلحات موضوعية: Male, Cancer Research, Fluorine Radioisotopes, Stereochemistry, Rats, Sprague-Dawley, Piperidines, Animals, Radiology, Nuclear Medicine and imaging, Receptor, Serotonin, 5-HT2A, Radioactive Tracers, Radiochemistry, Chemistry, Synthon, Binding potential, Desmethyl, Cortex (botany), Molecular Imaging, Rats, Fluorobenzenes, Positron-Emission Tomography, Serotonin 5-HT2 Receptor Antagonists, Molecular Medicine, Autoradiography, Specific activity, Steady state (chemistry), Enantiomer, Selectivity
-
5
المؤلفون: Patrick J. Riss, Frank Roesch, Ulrich Schmidt, Hartmut Lueddens, Fabian Debus, Patrick Schloss, René Hummerich
المصدر: ChemMedChem. 4(9)
مصطلحات موضوعية: Male, Fluorine Radioisotopes, Dopamine Plasma Membrane Transport Proteins, Biochemistry, Cell Line, Rats, Sprague-Dawley, In vivo, Drug Discovery, Animals, Humans, Tissue Distribution, General Pharmacology, Toxicology and Pharmaceutics, Serotonin transporter, Dopamine transporter, Pharmacology, Serotonin Plasma Membrane Transport Proteins, Norepinephrine Plasma Membrane Transport Proteins, biology, Chemistry, Organic Chemistry, Transporter, Ligand (biochemistry), Imaging agent, Rats, Positron-Emission Tomography, biology.protein, Biophysics, Molecular Medicine, Radiopharmaceuticals, Ex vivo, Tropanes
-
6
المؤلفون: Michaela Jansen, Hartmut Lüddens, Fabian Debus, Sandra Dieler, Myles H. Akabas, Axelle Strehle, Holger Rabe, Gerd Dannhardt
المصدر: Journal of medicinal chemistry. 51(15)
مصطلحات موضوعية: Models, Molecular, Patch-Clamp Techniques, Stereochemistry, Alpha (ethology), gamma-Aminobutyric acid, Article, GABAA-rho receptor, Cell Line, chemistry.chemical_compound, Structure-Activity Relationship, Xenopus laevis, Piperidines, Drug Discovery, medicine, Animals, Humans, GABA-A Receptor Agonists, Binding site, Receptor, gamma-Aminobutyric Acid, G alpha subunit, Binding Sites, Molecular Structure, Chemistry, GABAA receptor, Muscimol, Brain, Isoxazoles, Receptors, GABA-A, Rats, Electrophysiology, Protein Subunits, Biochemistry, Mutation, Oocytes, Molecular Medicine, Female, medicine.drug
-
7
المؤلفون: Hartmut Lüddens, Frank Rösch, Gitte M. Knudsen, Markus Piel, Fabian Debus, Mikael Palner, Matthias M. Herth
المصدر: Bioorganicmedicinal chemistry letters. 18(4)
مصطلحات موضوعية: Fluorine Radioisotopes, Stereochemistry, Clinical Biochemistry, Pharmaceutical Science, Biochemistry, Binding, Competitive, Radioligand Assay, Piperidines, In vivo, Drug Discovery, Animals, Radionuclide imaging, Receptor, Serotonin, 5-HT2A, Radionuclide Imaging, Molecular Biology, Chemistry, Organic Chemistry, Synthon, Total synthesis, Brain, Biological activity, Rats, Fluorobenzenes, Kinetics, Yield (chemistry), Isotope Labeling, Serotonin 5-HT2 Receptor Antagonists, Molecular Medicine, Specific activity, Ketanserin, Serotonin Antagonists, Radiopharmaceuticals, Nuclear chemistry
-
8
المؤلفون: Esa R. Korpi, Anni-Maija Linden, Cécile Malécot, William Wisden, M. Isabel Aller, Olga Vekovischeva, Hartmut Lüddens, Elli Leppä, Ingo Böhme, Fabian Debus, Holger Rabe
المساهمون: Academy of Finland, Sigrid Juselius Foundation
المصدر: Alcohol (Fayetteville, N.Y.). 41(3)
مصطلحات موضوعية: Azides, Health (social science), Pharmacology, Toxicology, Biochemistry, Binding, Competitive, 03 medical and health sciences, Behavioral Neuroscience, chemistry.chemical_compound, Benzodiazepines, Mice, 0302 clinical medicine, In vivo, Animals, Humans, Binding site, Receptor, Gene knockout, 030304 developmental biology, 0303 health sciences, Ethanol, Chemistry, GABAA receptor, HEK 293 cells, Central Nervous System Depressants, General Medicine, Drug Tolerance, Receptors, GABA-A, Cell biology, Rats, Neurology, Knockout mouse, 030217 neurology & neurosurgery
-
9دورية أكاديمية
المؤلفون: Michaela Jansen, Holger Rabe, Axelle Strehle, Sandra Dieler, Fabian Debus, Gerd Dannhardt, Myles H. Akabas, Hartmut Lüddens
المصدر: Journal of Medicinal Chemistry; Jul2008, Vol. 51 Issue 15, p4430-4448, 19p