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1
المؤلفون: Odra Pinato, Marco Catto, Fausta Palluotto, Barbara Gatto, Angelo Carotti, Alice Sosic, Grigoris Zoidis, Claudia Sissi
المصدر: European Journal of Medicinal Chemistry. 123:704-717
مصطلحات موضوعية: DNA Topoisomerase IV, 0301 basic medicine, Stereochemistry, Antineoplastic Agents, Chemistry Techniques, Synthetic, G-quadruplex, G-quadruplex stabilizers, 01 natural sciences, Quinoline derivatives, HeLa, Structure-Activity Relationship, 03 medical and health sciences, chemistry.chemical_compound, Antigens, Neoplasm, Quinoxalines, Drug Discovery, Humans, Topoisomerase II Inhibitors, Structure–activity relationship, Cytotoxic agents, Cytotoxicity, IC50, Pharmacology, chemistry.chemical_classification, Topoisomerase IIα inhibitors, biology, 010405 organic chemistry, Drug Discovery3003 Pharmaceutical Science, Organic Chemistry, Quinoline, General Medicine, Pyridazine derivatives, biology.organism_classification, 0104 chemical sciences, DNA-Binding Proteins, G-Quadruplexes, DNA Topoisomerases, Type II, 030104 developmental biology, chemistry, Quinolines, Topoisomerase-II Inhibitor, HeLa Cells, Tricyclic
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2
المؤلفون: Fausta Palluotto, Grigoris Zoidis, Marco Catto, Claudia Sissi, Angelo Carotti, Silvia Da Ros, Alice Sosic, Barbara Gatto
المصدر: Bioorganicmedicinal chemistry. 25(9)
مصطلحات موضوعية: 0301 basic medicine, DNA Topoisomerase IV, Topoisomerase iiα, Stereochemistry, Clinical Biochemistry, Intercalation (chemistry), Pharmaceutical Science, Antineoplastic Agents, G-quadruplex, Ligands, Indenocinnoline derivatives, Biochemistry, Heterocyclic Compounds, 4 or More Rings, HeLa, 03 medical and health sciences, chemistry.chemical_compound, Topoisomerase inhibitors, Drug Discovery, Moiety, Humans, Topoisomerase II Inhibitors, Benzothiazoles, Molecular Biology, Antitumor agents, biology, Chemistry, Drug Discovery3003 Pharmaceutical Science, Organic Chemistry, G-quadruplex binders, Intercalating agents, Molecular Medicine, 3003, biology.organism_classification, Fluorescence, Intercalating Agents, G-Quadruplexes, 030104 developmental biology, DNA Topoisomerases, Type II, Nucleic acid, MCF-7 Cells, Quinolines, DNA, HeLa Cells
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3
المؤلفون: Francesco Campagna, Carla Marra, Fausta Palluotto, Elisabetta Maciocco, Maria Paola Mascia, Angelo Carotti, Antonio Carrieri
المصدر: Il Farmaco. 58:129-140
مصطلحات موضوعية: Male, Molecular model, Ligand, GABAA receptor, Stereochemistry, Chemistry, Ligand binding assay, Drug Evaluation, Preclinical, Pharmaceutical Science, Receptors, GABA-A, Chemical synthesis, In vitro, Rats, Pyridazines, Rats, Sprague-Dawley, Weak binding, Drug Discovery, Animals, Biological evaluation
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4
المؤلفون: Angelo Carotti, G. Genchi, Giovanni Casini, Fausta Palluotto, Francesco Campagna
المصدر: Bioorganic & Medicinal Chemistry. 7:1533-1538
مصطلحات موضوعية: Models, Molecular, Indoles, Magnetic Resonance Spectroscopy, medicine.drug_class, Stereochemistry, Clinical Biochemistry, Pharmaceutical Science, Biochemistry, Chemical synthesis, Structure-Activity Relationship, Drug Discovery, medicine, Structure–activity relationship, Receptor, Molecular Biology, Benzodiazepine, Chemistry, Ligand binding assay, Organic Chemistry, Hydrogen Bonding, Nuclear magnetic resonance spectroscopy, Receptors, GABA-A, Ligand (biochemistry), Pyridazines, Molecular Medicine, Pharmacophore
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5
المؤلفون: Francesco Campagna, Giovanni Casini, A. De Luca, D. Conte-Camerino, Sabata Pierno, Angelo Carotti, Fausta Palluotto, Domenico Tricarico
المصدر: ChemInform. 26
مصطلحات موضوعية: chemistry.chemical_classification, Taurine, Ionic bonding, Skeletal muscle, General Medicine, Sulfonic acid, Amidine, chemistry.chemical_compound, Membrane, medicine.anatomical_structure, chemistry, Homotaurine, medicine, Organic chemistry
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6
المصدر: ChemInform. 28
مصطلحات موضوعية: chemistry.chemical_compound, Chemistry, Quinoline, Organic chemistry, General Medicine
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7
المؤلفون: M. Ferappi, Antonio Rosato, Francesco Campagna, Angelo Carotti, Cesare Vitali, Fausta Palluotto, Giovanni Casini
المصدر: ChemInform. 30
مصطلحات موضوعية: Indole test, Antifungal, biology, medicine.drug_class, Aryl, General Medicine, biology.organism_classification, In vitro, chemistry.chemical_compound, chemistry, medicine, Organic chemistry, Antibacterial activity, Bacteria
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8
المؤلفون: Francesco Campagna, Rosa Purgatorio, Fausta Palluotto, Angelo Carotti, Angelo De Stradis, Rosaria Aliano, Marco Catto, Saverio Cellamare
المصدر: European journal of medicinal chemistry 45 (2010): 1359–1366. doi:10.1016/j.ejmech.2009.12.029
info:cnr-pdr/source/autori:Catto M.; Aliano R.; Carotti A.; Cellamare S.; Palluotto F.; Purgatorio R.; De Stradis A.; Campagna F.;/titolo:Design, synthesis and biological evaluation of indane-2-arylhydrazinylmethylene-1,3-diones and indol-2-aryldiazenylmethylene-3-ones as a b-amyloid aggregation inhibitors./doi:10.1016%2Fj.ejmech.2009.12.029/rivista:European journal of medicinal chemistry/anno:2010/pagina_da:1359/pagina_a:1366/intervallo_pagine:1359–1366/volume:45مصطلحات موضوعية: Indoles, Magnetic Resonance Spectroscopy, Stereochemistry, Indane, Chemical synthesis, s disease, chemistry.chemical_compound, Microscopy, Electron, Transmission, b-Amyloid peptide, Drug Discovery, Benzothiazoles, Amyloid aggregation inhibitors, IC50, Pharmacology, Indole test, Amyloid beta-Peptides, Bicyclic molecule, Hydrogen bond, Organic Chemistry, Hydrogen Bonding, General Medicine, In vitro, Peptide Fragments, Thiazoles, Spectrometry, Fluorescence, chemistry, Alzheimer, Thioflavin
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::fc20b5a17258446e4e92c60af62a5abd
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9
المصدر: Farmaco (Societa chimica italiana : 1989). 59(11)
مصطلحات موضوعية: Male, Stereochemistry, medicine.drug_class, Pharmaceutical Science, Pyrazole, Ligands, Rats, Sprague-Dawley, chemistry.chemical_compound, Inhibitory Concentration 50, Drug Discovery, medicine, Animals, Polycyclic Aromatic Hydrocarbons, Receptor, Binding affinities, chemistry.chemical_classification, Benzodiazepine, Ligand, GABAA receptor, Ligand binding assay, General Medicine, Highly selective, Ligand (biochemistry), Receptors, GABA-A, Rats, chemistry, Pyrazoles, Tricyclic
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10
المؤلفون: Maria Paola Mascia, Angelo Carotti, Carla Marra, Fausta Palluotto, Elisabetta Maciocco, Antonio Carrieri, Francesco Campagna
المصدر: ChemInform. 34
مصطلحات موضوعية: Weak binding, Stereochemistry, Chemistry, GABAA receptor, General Medicine, Biological evaluation, Binding affinities