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1دورية أكاديمية
المؤلفون: Laurent Besret, Sébastien d’Heilly, Cathy Aubert, Guillaume Bluet, Florence Gruss-Leleu, Françoise Le-Gall, Anne Caron, Laurent Andrieu, Sylvie Vincent, Maysoun Shomali, Monsif Bouaboula, Carole Voland, Jeffrey Ming, Sébastien Roy, Srinivas Rao, Chantal Carrez, Erwan Jouannot
المصدر: EJNMMI Research, Vol 10, Iss 1, Pp 1-13 (2020)
مصطلحات موضوعية: SAR439859, Estrogen-positive breast cancer, SERD, Target engagement, Combination therapy, Palbociclib, Medical physics. Medical radiology. Nuclear medicine, R895-920
وصف الملف: electronic resource
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المؤلفون: Chrystelle Girardet, Magali Mathieu, François Vallée, Jacques Le-Roux, Fangxian Sun, Laurence Fabien, Corinne Terrier, Celine Ginesty, Bruno Filoche-Romme, Florence Gruss-Leleu, Maysoun Shomali, Monsif Bouaboula, Sylvie Beccari, Pascal Desmazeau, Gilles Lebourg, Tsiala Benard, Victor Certal, Pascale Vicat, Andrew Hebert, Carlos Garcia-Echeverria, Laurent Schio, Youssef El-Ahmad, Gary Mccort, Claire Muller, Maurice Brollo, Mikhail Levit, Luc Bertin, Hong Cheng, Véronique Loyau, Valerie Steier, Fabienne Thompson, Audrey Louboutin, Fabienne Pilorge, Alexey Rak, Frank Halley, Patrick Richepin, Christelle Perrault, Pierre-Yves Abecassis, Michel Tabart, Albane Courjaud
المصدر: Journal of Medicinal Chemistry. 63:512-528
مصطلحات موضوعية: 0303 health sciences, biology, Fulvestrant, Chemistry, Estrogen receptor, medicine.disease, 01 natural sciences, 0104 chemical sciences, 010404 medicinal & biomolecular chemistry, 03 medical and health sciences, Breast cancer, Hormone receptor, Drug Discovery, biology.protein, medicine, Cancer research, Molecular Medicine, Aromatase, Receptor, Estrogen receptor alpha, Tamoxifen, 030304 developmental biology, medicine.drug
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المؤلفون: Guillaume Bluet, Srinivas Rao, Jeffrey Ming, Maysoun Shomali, Laurent Besret, Carole Voland, Monsif Bouaboula, Chantal Carrez, Florence Gruss-Leleu, Erwan Jouannot, Sylvie Vincent, Sébastien d’Heilly, Cathy Aubert, Sébastien Roy, Anne Caron, Laurent Andrieu, Françoise Le-Gall
المصدر: EJNMMI Research
EJNMMI Research, Vol 10, Iss 1, Pp 1-13 (2020)مصطلحات موضوعية: lcsh:Medical physics. Medical radiology. Nuclear medicine, 0301 basic medicine, Target engagement, Estrogen-positive breast cancer, Positron emission tomography, Imaging biomarker, Combination therapy, Proliferation index, lcsh:R895-920, Estrogen receptor, [18F]-FDG, Palbociclib, 03 medical and health sciences, 0302 clinical medicine, In vivo, [18F]-FLT, medicine, Radiology, Nuclear Medicine and imaging, Original Research, Fluorodeoxyglucose, medicine.diagnostic_test, business.industry, SAR439859, 030104 developmental biology, [18F]-FES, 030220 oncology & carcinogenesis, SERD, Cancer research, business, medicine.drug
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المؤلفون: Mathilde, Pauton, Raphaël, Gillet, Catherine, Aubert, Guillaume, Bluet, Florence, Gruss-Leleu, Sébastien, Roy, Cécile, Perrio
المصدر: Organicbiomolecular chemistry. 17(26)
URL الوصول: https://explore.openaire.eu/search/publication?articleId=pmid________::b5e7cce94fc687af97d21c2a91a4e526
https://pubmed.ncbi.nlm.nih.gov/31218326 -
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المؤلفون: Jean Pierre Marquette, Andreas Karlsson, Sylvie Monget, Thomas Bertrand, Jean Christophe Carry, Frank Halley, Marc Antoine Perrin, Jean Paul Nicolas, Tsiala Benard, Angela Virone-Oddos, Luc Bertin, Céline Amara, Hélène Bonnevaux, Laurence Delbarre, Gilles Doerflinger, Pierre Yves Abecassis, Youssef El-Ahmad, Véronique Charrier, Victor Certal, Bruno Filoche-Romme, Florence Gruss-Leleu, Sébastien Perron, Alexey Rak, Patrick Richepin, Stephane Guerif, Carlos Garcia-Echeverria, Loic Vincent, Nadine Michot, Magali Mathieu, Véronique Loyau, Olivier Lemaitre, Maurice Brollo, Christoph Lengauer, Houlfa Guizani, Laurent Schio, Fabienne Thompson, Cécile Delorme
المصدر: Journal of Medicinal Chemistry. 57:903-920
مصطلحات موضوعية: Male, Cell Membrane Permeability, Indoles, Phosphatase, Molecular Conformation, Biological Availability, Antineoplastic Agents, Mice, SCID, Pyrimidinones, Crystallography, X-Ray, Mice, Rats, Nude, Structure-Activity Relationship, chemistry.chemical_compound, Dogs, In vivo, Cell Line, Tumor, Neoplasms, Drug Discovery, Animals, Humans, PTEN, Tensin, Pyrimidone, Phosphoinositide-3 Kinase Inhibitors, Mice, Inbred BALB C, biology, PTEN Phosphohydrolase, Stereoisomerism, In vitro, Rats, Molecular Docking Simulation, Solubility, chemistry, Structural biology, Biochemistry, Indoline, Microsomes, Liver, biology.protein, Cancer research, Heterografts, Molecular Medicine, Female, Drug Screening Assays, Antitumor, Neoplasm Transplantation, Protein Binding
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المؤلفون: Christoph Lengauer, Pierre Yves Abecassis, Luc Bertin, Véronique Charrier, Laurent Schio, Jean Christophe Carry, Patrick Richepin, Loic Vincent, Bruno Filoche-Romme, Florence Gruss-Leleu, Houlfa Guizani, Carlos Garcia-Echeverria, Angela Virone-Oddos, Andreas Karlsson, Jean Paul Nicolas, Victor Certal, Fabienne Pilorge, Frank Halley
المصدر: Bioorganicmedicinal chemistry letters. 24(6)
مصطلحات موضوعية: Male, Indoles, Stereochemistry, Carboxylic acid, Clinical Biochemistry, Carboxylic Acids, Pharmaceutical Science, Biochemistry, Permeability, Rats, Sprague-Dawley, chemistry.chemical_compound, Phosphatidylinositol 3-Kinases, Amide, Drug Discovery, Animals, Humans, Protein Isoforms, Thiazole, Molecular Biology, Protein Kinase Inhibitors, Phosphoinositide-3 Kinase Inhibitors, chemistry.chemical_classification, Binding Sites, Organic Chemistry, Combinatorial chemistry, Amides, Protein Structure, Tertiary, Rats, Molecular Docking Simulation, Thiazoles, chemistry, Molecular Medicine, Caco-2 Cells, Proto-Oncogene Proteins c-akt