نتائج البحث - "Francesco Bavo"

المصدر: Bavo, F, Pallavicini, M, Pucci, S, Appiani, R, Giraudo, A, Eaton, B, Lucero, L, Gotti, C, Moretti, M, Whiteaker, P & Bolchi, C 2022, ' From 2-Triethylammonium Ethyl Ether of 4-Stilbenol (MG624) to Selective Small-Molecule Antagonists of Human α9α10 Nicotinic Receptor by Modifications at the Ammonium Ethyl Residue ', Journal of Medicinal Chemistry, vol. 65, no. 14, pp. 10079-10097 . https://doi.org/10.1021/acs.jmedchem.2c00746

مصطلحات موضوعية: Quaternary Ammonium Compounds, Ammonium Compounds, Stilbenes, Drug Discovery, Humans, Molecular Medicine, Nicotinic Antagonists, Receptors, Nicotinic, Ether

وصف الملف: application/pdf

URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::bfd6ad38d76bc9fea125d38149cbb80c
https://curis.ku.dk/portal/da/publications/from-2triethylammonium-ethyl-ether-of-4stilbenol-mg624-to-selective-smallmolecule-antagonists-of-human-910-nicotinic-receptor-by-modifications-at-the-ammonium-ethyl-residue(0a208a35-2a1c-4134-86c9-ece88c9bf045).html

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Develop of new fluorescent probe to target hDHODH enzyme

المؤلفون: Martino, Elena, Sainas, Stefano, Francesco, Bavo, Garino, Claudio, Pippione, Agnese Chiara, Giorgis, Marta, Boschi, Donatella, Bente, Frølund, Lolli, Marco Lucio

URL الوصول: https://explore.openaire.eu/search/publication?articleId=od_______970::e1011e7a815bcb00a660b667e65a8b49
https://hdl.handle.net/2318/1883062

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Structure–activity studies of 3,9-diazaspiro[5.5]undecane-based γ-aminobutyric acid type A receptor antagonists with immunomodulatory effect

المؤلفون: Francesco Bavo, Heleen de-Jong, Jonas Petersen, Christina Birkedahl Falk-Petersen, Rebekka Löffler, Emma Sparrow, Frederik Rostrup, Jannik Nicklas Eliasen, Kristine S. Wilhelmsen, Kasper Barslund, Christoffer Bundgaard, Birgitte Nielsen, Uffe Kristiansen, Petrine Wellendorph, Yury Bogdanov, Bente Frølund

مصطلحات موضوعية: GABA Antagonists, Structure-Activity Relationship, Adjuvants, Immunologic, T-Lymphocytes, Drug Discovery, Alkanes, Molecular Medicine, Humans, Receptors, GABA-A, Cell Proliferation

وصف الملف: text

URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::fa1b8597a5aeec1385cffce2213ce18f
https://eprints.soton.ac.uk/454543/

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Efficient One-Pot Reductive Aminations of Carbonyl Compounds with Aquivion-Fe as a Recyclable Catalyst and Sodium Borohydride

المؤلفون: Riccardo Tassini, Marco Pallavicini, Oreste Piccolo, Veronica Airoldi, Sebastiano Arnoldi, Gabriella Roda, Stefano Paganelli, Cristiano Bolchi, Francesco Bavo, Rebecca Appiani

المصدر: European Journal of Organic Chemistry. 2020:162-168

مصطلحات موضوعية: Sodium borohydride, chemistry.chemical_compound, chemistry, Organic Chemistry, Organic chemistry, Physical and Theoretical Chemistry, Recyclable catalyst

URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_________::b542c1b1600e089813e37862c1f16f01
https://doi.org/10.1002/ejoc.201901614

View record at Wiley

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Determinants for α4β2 vs. α3β4 subtype selectivity of pyrrolidine-based nachrs ligands:A computational perspective with focus on recent cryo-em receptor structures

المؤلفون: Francesco Bavo, Marco Pallavicini, Cristiano Bolchi, Rebecca Appiani

المصدر: Bavo, F, Pallavicini, M, Appiani, R & Bolchi, C 2021, ' Determinants for α4β2 vs. α3β4 subtype selectivity of pyrrolidine-based nachrs ligands : A computational perspective with focus on recent cryo-em receptor structures ', Molecules, vol. 26, no. 12, 3603 . https://doi.org/10.3390/molecules26123603
Molecules
Molecules, Vol 26, Iss 3603, p 3603 (2021)
Volume 26
Issue 12

مصطلحات موضوعية: Alpha3beta4, Pyrrolidines, Pyridines, Pharmaceutical Science, N-methyl-pyrrolidinyl, Receptors, Nicotinic, Ligands, 01 natural sciences, Synaptic Transmission, Pyrrolidine, Analytical Chemistry, Docking, chemistry.chemical_compound, QD241-441, alpha4beta2, Drug Discovery, Databases, Genetic, Alpha4beta2, Selectivity, Nicotinic Agonists, Receptor, Cryo-EM, 0303 health sciences, NAChR, Molecular Docking Simulation, Nicotinic agonist, Chemistry (miscellaneous), docking, Molecular Medicine, benzodioxane, Agonist, medicine.drug_class, Structural similarity, Stereochemistry, Benzodioxane, Ether, (S)-nicotine, nAChR, Article, 03 medical and health sciences, Structure-Activity Relationship, medicine, Animals, Humans, Physical and Theoretical Chemistry, 030304 developmental biology, Binding Sites, 010405 organic chemistry, Organic Chemistry, Cryoelectron Microscopy, selectivity, 0104 chemical sciences, Rats, chemistry, Docking (molecular), cryo-EM, alpha3beta4

وصف الملف: application/pdf

URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::512c7f5ba85f13f25e44ad6f04bd9fa1
https://curis.ku.dk/ws/files/285447571/molecules_26_03603_v2.pdf

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Modifications at C(5) of 2-(2-Pyrrolidinyl)-Substituted 1,4-Benzodioxane Elicit Potent α4β2 Nicotinic Acetylcholine Receptor Partial Agonism with High Selectivity over the α3β4 Subtype

المؤلفون: Cecilia Gotti, Susanna Pucci, Sara Francesca Colombo, Massimiliano Renzi, Rebecca Appiani, Marco Pallavicini, Roberta Budriesi, Sergio Fucile, Francesco Bavo, Milena Moretti, Cristiano Bolchi, Paola Viani

المساهمون: Bavo F., Pallavicini M., Gotti C., Appiani R., Moretti M., Colombo S.F., Pucci S., Viani P., Budriesi R., Renzi M., Fucile S., Bolchi C.

مصطلحات موضوعية: Pyrrolidines, α4β2 α3β4 NAchRs Partial Agonism Patch-Clamp Computational Modeling, Stereochemistry, Nicotinic Agonist, High selectivity, Substituent, Nicotinic Antagonists, Receptors, Nicotinic, 01 natural sciences, Pyrrolidine, Dioxanes, 03 medical and health sciences, chemistry.chemical_compound, Structure-Activity Relationship, Drug Discovery, Humans, Nicotinic Agonists, Dioxane, 030304 developmental biology, 0303 health sciences, Binding Sites, Cryoelectron Microscopy, Diastereomer, Binding Site, Hydrogen Bonding, Stereoisomerism, 0104 chemical sciences, Molecular Docking Simulation, 010404 medicinal & biomolecular chemistry, Nicotinic acetylcholine receptor, chemistry, Nicotinic Antagonist, Mutagenesis, Site-Directed, Molecular Medicine, Human