-
1
المؤلفون: Jay A. Markwalder, Aaron J. Balog, David K. Williams, Susheel J. Nara, Ratnakar Reddy, Saumya Roy, Yadagiri Kanyaboina, Xin Li, Kathy Johnston, Yi Fan, Hal Lewis, Frank Marsilio, Chunhong Yan, David Critton, John A. Newitt, Sarah C. Traeger, Dauh-Rurng Wu, Maria N. Jure-Kunkel, Lata Jayaraman, Tai-An Lin, Michael W. Sinz, John T. Hunt, Steven P. Seitz
مصطلحات موضوعية: Organic Chemistry, Clinical Biochemistry, Drug Discovery, Pharmaceutical Science, Molecular Medicine, Molecular Biology, Biochemistry
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::64f0da67b51d6c7282c418d8dbb98887
https://doi.org/10.2139/ssrn.4348735 -
2
المؤلفون: Ching Kim Tye, Chunhong Yan, Sarah C. Traeger, Wayne Vaccaro, Yingru Zhang, Gerry Everlof, Jianqing Li, Henry Yip, Peng Li, John T. Hunt, Michael A. Poss, Gregory D. Vite, Mussari Christopher P, Steven Sheriff, Asoka Ranasinghe, Haiying Zhang, Richard A. Westhouse, Dharmpal S. Dodd, Richard Rampulla, Zheng Yang, Frank Marsilio, Derek J. Norris, Wen-Ching Han, Tram N. Huynh, Yufen Zhao, Patrice Gill, Nirmala Raghavan, Lalgudi S. Harikrishnan, Ashvinikumar V. Gavai, Susan Wee, John S. Tokarski, Dauh-Rurng Wu, Arvind Mathur, Mei-Li Wen, Huiping Zhang, David R. Tortolani, George V. Delucca, Krista Menard, Francis Y. Lee, Claude A. Quesnelle, Dawn Sun, Vijay T. Ahuja, Daniel O'malley, Christine Huang, Muthoni G. Kamau
المصدر: Journal of Medicinal Chemistry. 64:14247-14265
مصطلحات موضوعية: Drug, Proline, Phenylalanine, media_common.quotation_subject, Carbazoles, Administration, Oral, Antineoplastic Agents, Cell Cycle Proteins, Computational biology, BET inhibitor, Structure-Activity Relationship, Pharmacokinetics, In vivo, Drug Discovery, Transcriptional regulation, Humans, Potency, media_common, Dose-Response Relationship, Drug, Molecular Structure, Chemistry, Tryptophan, Signal transducing adaptor protein, Bromodomain, Molecular Medicine, Transcription Factors
-
3
المؤلفون: Andrew P. Degnan, Haiquan Fang, Tatyana Zvyaga, Zuzana Haarhoff, Claude A. Quesnelle, Melissa Kramer, Frank Marsilio, Richard A. Westhouse, John S. Tokarski, Shilpa Madari, Jiuqiao Zhao, Amy Wiebesiek, Chunhong Yan, Francis Y. Lee, Michael Sinz, John Morrison, Jean Simmermacher-Mayer, Carolynn Fanslau, Steven Sheriff, Lisa Huang, Ashvinikumar V. Gavai, Chunshan Xie, Matthew D. Hill, Gerry Everlof
المصدر: Bioorganicmedicinal chemistry letters. 51
مصطلحات موضوعية: Stereochemistry, Cell Survival, Clinical Biochemistry, Pharmaceutical Science, Structural diversity, Administration, Oral, Antineoplastic Agents, Triple Negative Breast Neoplasms, Biochemistry, Polar surface area, BET inhibitor, Mice, Structure-Activity Relationship, Drug Development, Drug Discovery, medicine, Animals, Humans, Molecular Biology, Chemotype, Dose-Response Relationship, Drug, Molecular Structure, Chemistry, Organic Chemistry, Cancer, Mammary Neoplasms, Experimental, Proteins, medicine.disease, In vitro, Bromodomain, Molecular Medicine, Drug Screening Assays, Antitumor, Carbolines
-
4
المؤلفون: Frank Marsilio, Chiehying Chang, Steven Sheriff, Bradley C. Pearce, Iyoncy Rodrigo, Max Ruzanov, Dasa Lipovsek, Jodi K. Muckelbauer, Mian Gao, Heather Malakian, Dianlin Xie, John A. Newitt, Wai L. Lau
المصدر: Acta Crystallogr F Struct Biol Commun
مصطلحات موضوعية: Models, Molecular, Biophysics, Saccharomyces cerevisiae, Protein Serine-Threonine Kinases, Crystallography, X-Ray, Protein Engineering, Biochemistry, Method Communications, law.invention, 03 medical and health sciences, 0302 clinical medicine, Immune system, Protein Domains, Structural Biology, law, Genetics, Humans, Homology modeling, Protein Kinase Inhibitors, 030304 developmental biology, 0303 health sciences, Kinase, Chemistry, Drug discovery, Condensed Matter Physics, Yeast, Recombinant Proteins, Cell biology, Protein kinase domain, Mutagenesis, 030220 oncology & carcinogenesis, Mutation, Recombinant DNA, Cell Surface Display Techniques, Crystallization, Intracellular
-
5
المؤلفون: Juhi Juneja, Zhou Dai, Daniel Cohen, Lumelle A. Schneeweis, Ruchira Dasgupta, Frank Marsilio, Paul E. Morin
المصدر: BioTechniques. 69(3)
مصطلحات موضوعية: 0303 health sciences, medicine.diagnostic_test, Chemistry, Microfluidics, Protein engineering, Ligands, General Biochemistry, Genetics and Molecular Biology, B7-H1 Antigen, 03 medical and health sciences, 0302 clinical medicine, Positron emission tomography, 030220 oncology & carcinogenesis, Positron-Emission Tomography, medicine, Radioligand, Biophysics, Humans, 030304 developmental biology, Biotechnology, Protein Binding
-
6
المؤلفون: Chunhong Yan, Francis Y. Lee, Ashvinikumar V. Gavai, Melissa Kramer, Frank Marsilio, Eric Shields, Laura Monereau, Zuzana Haarhoff, Richard A. Westhouse, Lisa Zhang, Gerry Everlof, John S. Tokarski, Matthew D. Hill, Tatyana Zvyaga, Asoka Ranasinghe, Carolynn Fanslau, Ching Kim Tye, Steven Sheriff, Christine Huang, Andrew P. Degnan, Krista Menard, John Morrison, Haiquan Fang
المصدر: Bioorganic & Medicinal Chemistry Letters. 44:128108
مصطلحات موضوعية: Clinical Biochemistry, Pharmaceutical Science, Structural diversity, Antineoplastic Agents, Biochemistry, BET inhibitor, Mice, Structure-Activity Relationship, Drug Development, Drug Discovery, medicine, Animals, Humans, Moiety, Potency, Mouse tumor, Molecular Biology, Dose-Response Relationship, Drug, Molecular Structure, Chemistry, Organic Chemistry, Proteins, Cancer, Triazoles, medicine.disease, Combinatorial chemistry, Bromodomain, Molecular Medicine, Multiple Myeloma, Carbolines
-
7
المؤلفون: William J. Metzler, Luciano Mueller, Yaqun Zhang, Mian Gao, Nicolas Szapiel, Mark R. Witmer, David Hedin, Deepa Calambur, Dianlin Xie, Hui Wei, Frank Marsilio, Andrew E Douglas, Ping Zhang
المصدر: Journal of Biomolecular NMR. 68:237-247
مصطلحات موضوعية: 0301 basic medicine, Spodoptera, Biochemistry, 03 medical and health sciences, chemistry.chemical_compound, Stable isotope labeling by amino acids in cell culture, Sf9 Cells, Animals, Amino Acids, Nuclear Magnetic Resonance, Biomolecular, Spectroscopy, chemistry.chemical_classification, Carbon Isotopes, Growth medium, Chromatography, Nitrogen Isotopes, 030102 biochemistry & molecular biology, Insect cell culture, Yeast, Culture Media, Amino acid, 030104 developmental biology, chemistry, Focal Adhesion Kinase 1, Isotope Labeling, Protein Biosynthesis, Reagent, Yield (chemistry), CD4 Antigens, Fermentation, Baculoviridae
-
8
المؤلفون: Frank Marsilio, Ernst Schönbrunn, Stephane Betzi, Huijong Han, Jin-Yi Zhu, S.H. Olesen, Yan Yang
المصدر: Journal of Biological Chemistry. 287:12657-12667
مصطلحات موضوعية: Stereochemistry, Crystallography, X-Ray, Biochemistry, Substrate Specificity, Adduct, Phosphoenolpyruvate, DNA Adducts, Structure-Activity Relationship, Residue (chemistry), Protein structure, Mura, Enterobacter cloacae, Escherichia coli, Transferase, Molecular Biology, Alkyl and Aryl Transferases, biology, Chemistry, Active site, Cell Biology, Recombinant Proteins, Protein Structure, Tertiary, Enzyme Activation, Covalent bond, Muramic Acids, Enzymology, biology.protein, Phosphoenolpyruvate carboxykinase
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::80e5bb39139217545749e42ace0eddc4
https://doi.org/10.1074/jbc.m112.342725 -
9
المؤلفون: Wayne C. Guida, Yiyu Ge, Harshani R. Lawrence, Sanjula Jain, Yunting Luo, Said M. Sebti, Wesley H. Brooks, Kenyon G. Daniel, Frank Marsilio, Aslamuzzaman Kazi
المصدر: Journal of Medicinal Chemistry. 55:1978-1998
مصطلحات موضوعية: Stereochemistry, Carboxylic acid, Triazole, Tetrazoles, Antineoplastic Agents, Thiophenes, Article, Small Molecule Libraries, Structure-Activity Relationship, chemistry.chemical_compound, Drug Stability, Cell Line, Tumor, Drug Discovery, Side chain, Animals, Chymotrypsin, Humans, Structure–activity relationship, Tetrazole, Thioglycolic acid, chemistry.chemical_classification, Sulfonamides, Triazoles, Sulfonamide, chemistry, Thioglycolates, Molecular Medicine, Rabbits, Pharmacophore, Proteasome Inhibitors, Naphthoquinones
-
10
المؤلفون: Ann E. Weber, Reshma A. Patel, Joseph K. Wu, Aleksandr Petrov, Frank Marsilio, Jennifer E. Kowalchick, KellyAnn D. Pryor, Nancy A. Thornberry, Barbara Leiting, Kathryn A. Lyons, Giovanna Scapin, Huaibing He, George J. Eiermann, Dooseop Kim
المصدر: Bioorganic & Medicinal Chemistry Letters. 17:5934-5939
مصطلحات موضوعية: Models, Molecular, Clinical Biochemistry, Drug Evaluation, Preclinical, Pharmaceutical Science, Crystallography, X-Ray, Biochemistry, Piperazines, Dipeptidyl peptidase, Pharmacokinetics, In vivo, Drug Discovery, Animals, Protease Inhibitors, Beta (finance), Molecular Biology, Dipeptidyl-Peptidase IV Inhibitors, Chemistry, DPP-4 Inhibitors, Organic Chemistry, Amides, Rats, Bioavailability, Orally active, Design synthesis, Drug Design, Molecular Medicine