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المؤلفون: David M. Glover, Frederic Scaerou, Emma Easthope, David O. Jones, David A. Sorrell, Amy Emery, Daniella Zheleva, Stacy Lawrence, Mark W. Stockdale
المصدر: SLAS Discovery. 16:925-931
مصطلحات موضوعية: Mitotic index, Cell, Aurora inhibitor, Regulator, Aurora A kinase, Mitosis, Uterine Cervical Neoplasms, Antineoplastic Agents, macromolecular substances, Protein Serine-Threonine Kinases, Biology, Biochemistry, Piperazines, Analytical Chemistry, Small Molecule Libraries, Aurora Kinases, medicine, Humans, Phosphorylation, Protein Kinase Inhibitors, Automation, Laboratory, Centrosome, Tumor Suppressor Proteins, Organophosphates, High-Throughput Screening Assays, Molecular Imaging, Cell biology, enzymes and coenzymes (carbohydrates), medicine.anatomical_structure, embryonic structures, Quinazolines, Molecular Medicine, Female, biological phenomena, cell phenomena, and immunity, Antibodies, Phospho-Specific, Microtubule-Associated Proteins, HeLa Cells, Biotechnology
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::1544d1b347478bdde0bac8b9e63930fd
https://doi.org/10.1177/1087057111413923 -
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المؤلفون: Peter Fischer, Christopher Meades, Iain Stuart, Mokdad Mezna, Carol Midgley, Joanna B. Grabarek, Campbell McInnes, Mark P. Thomas, George Kontopidis, Frederic Scaerou, David M. Glover, Gavin Wood, Wayne Jackson, Andy Plater, Rosemary G. Clarke, David Blake, Gary Griffiths, Steven J. McClue, Robert C. Jackson, Shudong Wang, David P. Lane, Daniella Zheleva
المساهمون: Wang, Shudong, Midgley, Carol A, Scaerou, Frederic, Grabarek, Joanna, Fischer, Peter M
المصدر: Journal of medicinal chemistry. 53(11)
مصطلحات موضوعية: Models, Molecular, Protein Conformation, Aurora inhibitor, Mitosis, Protein Serine-Threonine Kinases, Binding, Competitive, Substrate Specificity, Histone H3, Inhibitory Concentration 50, Mice, Aurora kinase, Adenosine Triphosphate, Aurora Kinases, Cell Line, Tumor, Drug Discovery, Animals, Humans, Cytotoxicity, Protein Kinase Inhibitors, Aurora Kinase A, Cell Proliferation, Kinase, Chemistry, Xenograft Model Antitumor Assays, Thiazoles, Pyrimidines, Biochemistry, Molecular Medicine, Phosphorylation
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المؤلفون: Amy Emery, Nicola L. Rogers, Michael G. Thomas, David Blake, Graeme Thomson, Stuart Jones, Simon Green, Abhijeet Choudhary, David M. Glover, Frederic Scaerou, Claire June Flynn, Jonathan Hollick, Janice Mclachlan
المصدر: Cancer Research. 70:4435-4435
مصطلحات موضوعية: Cancer Research, Kinase, Cell, Polo-like kinase, Biology, medicine.disease_cause, PLK1, medicine.anatomical_structure, Oncology, Immunology, Cancer research, medicine, Protein kinase A, Carcinogenesis, Mitosis, Cytokinesis
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_________::cf88c64f7cfba9166c2c19d15758b182
https://doi.org/10.1158/1538-7445.am10-4435