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1
المؤلفون: Liping Wang, Shihyun You, Ninad V. Prabhu, Hongfeng Deng, Danielle G. Smith, Jing Chai, Ginger H Tomberlin, Robert T. Nolte, James H. Nichols, G. Bruce Wisely, Edgar R. Wood, Cecil E Rise, Hamilton D. Dickson, J. David Taylor, Luz Helena Kryn, Randy K. Bledsoe, Timothy P. Sheahan, Yun Ding, Sarah Harris-Gurley, Eldridge N. Nartey, J. Brad Shotwell, Bing Xia, Philias Daka, Vince Tai
المصدر: Journal of Biological Chemistry
مصطلحات موضوعية: Models, Molecular, Rhinovirus, Biology, Crystallography, X-Ray, Biochemistry, Antiviral Agents, Virus, Small Molecule Libraries, Gene Knockout Techniques, Structure-Activity Relationship, Interferon, Transcription (biology), Endoribonucleases, medicine, 2',5'-Oligoadenylate Synthetase, Escherichia coli, Humans, Encephalomyocarditis virus, Molecular Biology, Regulation of gene expression, Innate immune system, Oligoribonucleotides, Effector, Adenine Nucleotides, Phosphodiesterase, Interferon-alpha, Molecular Bases of Disease, Cell Biology, Virology, Immunity, Innate, Recombinant Proteins, Respiratory Syncytial Viruses, Poly I-C, Gene Expression Regulation, Cell culture, Exoribonucleases, medicine.drug, HeLa Cells, Signal Transduction
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::aef2ae03677c0520338a9d289226a214
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2
المؤلفون: Harry B. Marr, Kevin P. Madauss, Jonathan Y. Bass, Shawn P. Williams, Dan Todd, Paul Kenneth Spearing, Adwoa Akwabi-Ameyaw, Lihong Chen, Robert B. McFadyen, Justin A. Caravella, Derek J. Parks, Frank Navas, David N. Deaton, Katrina L. Creech, G. Bruce Wisely, Richard Dana Caldwell, Aaron B. Miller
المصدر: Bioorganic & Medicinal Chemistry Letters. 19:4733-4739
مصطلحات موضوعية: Agonist, Stereochemistry, medicine.drug_class, Clinical Biochemistry, Receptors, Cytoplasmic and Nuclear, Pharmaceutical Science, Thiophenes, Naphthalenes, Crystallography, X-Ray, Biochemistry, Chemical synthesis, Structure-Activity Relationship, chemistry.chemical_compound, Drug Discovery, medicine, Animals, Humans, Computer Simulation, Molecular Biology, Binding Sites, Organic Chemistry, Benzothiophene, Isoxazoles, Rats, Nuclear receptor, chemistry, Molecular Medicine, Farnesoid X receptor
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المؤلفون: Justin A. Caravella, David N. Deaton, Katrina L. Creech, G. Bruce Wisely, Jonathan Y. Bass, Lihong Chen, Harry B. Marr, Robert B. McFadyen, Shawn P. Williams, Richard Dana Caldwell, Kevin P. Madauss, Aaron B. Miller, Derek J. Parks, Dan Todd
المصدر: Bioorganic & Medicinal Chemistry Letters. 19:2969-2973
مصطلحات موضوعية: Agonist, medicine.drug_class, Stereochemistry, Clinical Biochemistry, Receptors, Cytoplasmic and Nuclear, Pharmaceutical Science, Crystallography, X-Ray, Biochemistry, Chemical synthesis, Structure-Activity Relationship, chemistry.chemical_compound, Drug Discovery, Fluorescence Resonance Energy Transfer, medicine, Animals, Structure–activity relationship, Isoxazole, Molecular Biology, Aryl, Organic Chemistry, Isoxazoles, G protein-coupled bile acid receptor, Rats, Nuclear receptor, chemistry, Molecular Medicine, Farnesoid X receptor
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المؤلفون: Lihong Chen, Jonathan Y. Bass, David N. Deaton, Aaron B. Miller, Justin A. Caravella, Istvan Kaldor, Robert B. McFadyen, Stacey A. Jones, Dan Todd, Paul Kenneth Spearing, Kevin P. Madauss, Adwoa Akwabi-Ameyaw, Derek J. Parks, Richard Dana Caldwell, Frank Navas, Yaping Liu, Katrina L. Creech, G. Bruce Wisely, Harry B. Marr, Shawn P. Williams
المصدر: Bioorganic & Medicinal Chemistry Letters. 18:4339-4343
مصطلحات موضوعية: Agonist, Molecular model, medicine.drug_class, Stereochemistry, Clinical Biochemistry, Carboxylic Acids, Molecular Conformation, Administration, Oral, Receptors, Cytoplasmic and Nuclear, Pharmaceutical Science, Naphthalenes, Crystallography, X-Ray, Biochemistry, Chemical synthesis, Mice, Structure-Activity Relationship, Dogs, Drug Discovery, medicine, Animals, Structure–activity relationship, Receptor, Molecular Biology, Cholestasis, Molecular Structure, Chemistry, Stomach, Organic Chemistry, Haplorhini, Isoxazoles, G protein-coupled bile acid receptor, Rats, DNA-Binding Proteins, Disease Models, Animal, Nuclear receptor, Gastric Mucosa, Molecular Medicine, Farnesoid X receptor, Transcription Factors
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5
المؤلفون: Kenneth H. Pearce, Robert A. Reid, Nan Wu, Lei Yin, G. Bruce Wisely, Mohammed Qatanani, Derek J. Parks, Nava R. Szwergold, Mitchell A. Lazar, Joshua C. Curtin, Gregory M. Waitt
المصدر: Science. 318:1786-1789
مصطلحات موضوعية: Male, Circadian clock, Receptors, Cytoplasmic and Nuclear, Heme, Histone Deacetylases, Article, Cofactor, Cell Line, Mice, chemistry.chemical_compound, Biological Clocks, Cell Line, Tumor, Animals, Homeostasis, Humans, Nuclear Receptor Co-Repressor 1, Glucose homeostasis, Circadian rhythm, Transcription factor, Multidisciplinary, biology, Gluconeogenesis, Nuclear Proteins, Circadian Rhythm, Cell biology, DNA-Binding Proteins, Repressor Proteins, Glucose, Gene Expression Regulation, Biochemistry, Nuclear receptor, chemistry, Nuclear Receptor Subfamily 1, Group D, Member 1, Glucose-6-Phosphatase, biology.protein, Hemin, Energy Metabolism, Corepressor, Metabolic Networks and Pathways
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::1de58dda8076924425e0ce4e76ac79c4
https://doi.org/10.1126/science.1150179 -
6
المؤلفون: Olivia R. R. Ittoop, Hongbing Wang, G. Bruce Wisely, Virginia E. Carnahan, Tom Luntz, Julie B. Stimmel, Linda B. Moore, Schroeder M. Noble, Paula R. Davis-Searles, Edward L. LeCluyse, Ashutosh Tripathy, Donald P. McDonnell, Ryan E. Watkins, Matthew R. Redinbo
المصدر: Biochemistry. 45:8579-8589
مصطلحات موضوعية: Receptors, Steroid, Receptors, Cytoplasmic and Nuclear, Biology, Ligands, Biochemistry, Article, Nuclear Receptor Coactivator 1, Constitutive androstane receptor, Humans, Nuclear receptor co-repressor 1, Histone Acetyltransferases, Pregnane X receptor, Retinoid X Receptor alpha, Retinoid X receptor alpha, Pregnane X Receptor, Tryptophan, DNA, Protein Structure, Tertiary, Nuclear receptor coactivator 1, Nuclear receptor, Nuclear receptor coactivator 3, Nuclear receptor coactivator 2, Biophysics, Dimerization, Ultracentrifugation, Transcription Factors
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المؤلفون: Dana R Hohman, Lisa A. Orband-Miller, Susan L. Weaver, Eugene L. Stewart, Shawn P. Williams, John T. Moore, Thomas G. Consler, Paul Kenneth Spearing, Ning Go, Philip Stewart Turnbull, Millard H. Lambert, Ron L. Hale, Linda B. Moore, Stacey A. Jones, Amy T. Lu, Brad R. Henke, G. Bruce Wisely, Jean Shearin, R. Graham Robinett
المصدر: Journal of Medicinal Chemistry. 45:5492-5505
مصطلحات موضوعية: Models, Molecular, endocrine system, Transcription, Genetic, Estrogen receptor, Crystallography, X-Ray, Ligands, Partial agonist, Radioligand Assay, Structure-Activity Relationship, Genes, Reporter, Drug Discovery, Tumor Cells, Cultured, polycyclic compounds, Estrogen Receptor beta, Humans, Structure–activity relationship, Receptor, reproductive and urinary physiology, Estrogen receptor beta, Triazines, Chemistry, Ligand binding assay, Estrogen Receptor alpha, Stereoisomerism, Antiestrogen, Receptors, Estrogen, Biochemistry, Molecular Medicine, Estrogen receptor alpha, hormones, hormone substitutes, and hormone antagonists
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المؤلفون: Timothy M. Willson, John T. Moore, Robert L. Johnson, Roderick G. Davis, Andrea M. Sefler, Barry G. Shearer, Alan D. Thornquest, Ann B. Miller, Tim Spitzer, Aaron B. Miller, G. Bruce Wisely, Shawn P. Williams
المصدر: Structure. 10(9):1225-1234
مصطلحات موضوعية: Models, Molecular, Magnetic Resonance Spectroscopy, Transcription, Genetic, Protein Conformation, Molecular Sequence Data, Plasma protein binding, Biology, Crystallography, X-Ray, HNF4, Gas Chromatography-Mass Spectrometry, Cell Line, Palmitic acid, Structure-Activity Relationship, chemistry.chemical_compound, Protein structure, Structural Biology, Fatty acid binding, Humans, Protein Isoforms, nuclear receptor, Amino Acid Sequence, Transcription factor, Molecular Biology, transcription factor, chemistry.chemical_classification, diabetes, Sequence Homology, Amino Acid, Basic Helix-Loop-Helix Leucine Zipper Transcription Factors, Fatty Acids, Fatty acid, Phosphoproteins, Molecular biology, DNA-Binding Proteins, Hepatocyte Nuclear Factor 4, chemistry, Biochemistry, Hepatocyte nuclear factor 4, MODY, Free fatty acid receptor, Protein Binding, Transcription Factors
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المؤلفون: Jürgen M. Lehmann, Millard H. Lambert, Daniel D. Sternbach, Valerie G. Montana, Timothy M. Willson, H. Eric Xu, Derek J. Parks, G. Bruce Wisely, Peter Brown, Steven G. Blanchard, Michael V. Milburn, Steven A. Kliewer
المصدر: Molecular Cell. 3:397-403
مصطلحات موضوعية: Models, Molecular, Protein Conformation, medicine.drug_class, Molecular Conformation, Receptors, Cytoplasmic and Nuclear, Fibrate, Plasma protein binding, Biology, Crystallography, X-Ray, Ligands, Protein Structure, Secondary, Inhibitory Concentration 50, Protein structure, medicine, Animals, Humans, Receptor, Molecular Biology, Binding Sites, Phenylurea Compounds, Fatty Acids, Hydrogen Bonding, Cell Biology, Peroxisome, Eicosapentaenoic acid, Butyrates, Eicosapentaenoic Acid, Biochemistry, Nuclear receptor, lipids (amino acids, peptides, and proteins), Peroxisome proliferator-activated receptor delta, Crystallization, Protein Binding, Transcription Factors
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10دورية أكاديمية
المؤلفون: Stefan Westin, Riki Kurokawa, Robert T. Nolte, G. Bruce Wisely, Eileen M. McInerney, David W. Rose, Michael V. Milburn, Michael G. Rosenfeld, Christopher K. Glass
المصدر: Nature, Nature. 395(6698):199-202