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1دورية أكاديمية
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2
المؤلفون: Cecilia Pozzi, Alessandro Pratesi, Stefano Mangani, Paola Turano, Silvia Ciambellotti, G. Tassone
المصدر: Chemistry – A European Journal. 27:14690-14701
مصطلحات موضوعية: Iron, Oxide, Ferroxidase activity, Ferric Compounds, Redox, Catalysis, chemistry.chemical_compound, ferroxidase sites, medicine, Animals, Humans, Binding site, Binding Sites, accessory transient sites, biology, Chemistry, Organic Chemistry, ferroxidase reactions, human mitochondrial ferritin, MITOCHONDRIAL FERRITIN, Ceruloplasmin, General Chemistry, Ferritin, Apoferritins, Ferritins, biology.protein, Biophysics, Ferric, Oxidation-Reduction, medicine.drug
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3دورية أكاديمية
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4Xanthopsin-Like Systems via Site-Specific Click-Functionalization of a Retinoic Acid Binding Protein
المؤلفون: Cecilia Pozzi, Maurizio Orlandini, Benedetta Carlotti, Fausto Ortica, Massimo Olivucci, Loredana Latterini, Annalisa Reale, Laura Salvini, Gianluca Giorgi, Stefano Mangani, Marco Paolino, Xuchun Yang, Andrea Cappelli, G. Tassone, Federico Galvagni
المصدر: Chembiochem
مصطلحات موضوعية: Models, Molecular, Morita-Baylis-Hillman adducts, Rhodopsin, site-specific reactions, Receptors, Retinoic Acid, Retinoic acid, Optogenetics, Crystallography, X-Ray, Biochemistry, PYP-like chromophores, Article, light-sensitive proteins, chemistry.chemical_compound, Synthetic biology, Retinoic acid binding, Molecular Biology, Molecular Structure, biology, synthetic xanthopsin-like proteins, Organic Chemistry, Stereoisomerism, Transporter, Chromophore, Combinatorial chemistry, In vitro, chemistry, biology.protein, Molecular Medicine, Click Chemistry
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::c495be6a4930178e4530bc4fa123347b
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المؤلفون: Pasquale Linciano, Cecilia Pozzi, G. Tassone, Stefano Mangani, G. Landi, Maria Paola Costi
المصدر: Acta Crystallographica Section D Structural Biology. 76:558-564
مصطلحات موضوعية: Models, Molecular, Indoles, Stereochemistry, human African trypanosomiasis, Trypanosoma brucei brucei, Protozoan Proteins, Trypanosoma brucei, Cofactor, Antiparasitic drugs, High-resolution crystal structure, Human African trypanosomiasis, Pteridine reductase 1, Tricyclic compound, Structure-Activity Relationship, pteridine reductase 1, 03 medical and health sciences, tricyclic compound, 0302 clinical medicine, Structural Biology, Dihydrofolate reductase, medicine, African trypanosomiasis, Enzyme Inhibitors, Ternary complex, 030304 developmental biology, chemistry.chemical_classification, 0303 health sciences, Molecular Structure, biology, Bicyclic molecule, Chemistry, biology.organism_classification, medicine.disease, Trypanocidal Agents, antiparasitic drugs, high-resolution crystal structure, 3. Good health, Drug Design, 030220 oncology & carcinogenesis, biology.protein, Trypanosoma, Oxidoreductases, Tricyclic
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6دورية أكاديمية
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المؤلفون: Pasquale Linciano, Michele Tonelli, Cecilia Pozzi, Valeria Francesconi, Stefano Mangani, G. Landi, Lorenzo Tagliazucchi, G. Tassone, Maria Paola Costi
المصدر: Pharmaceuticals
Volume 14
Issue 7
Pharmaceuticals, Vol 14, Iss 636, p 636 (2021)مصطلحات موضوعية: Chagas disease, Cycloguanil, dual inhibitor, Trypanosoma brucei, structure–activity relationship, pteridine reductase, antifolate drug, Pharmaceutical Science, Pharmacology, cycloguanil, Article, 03 medical and health sciences, chemistry.chemical_compound, Pharmacy and materia medica, dihydrofolate reductase, Drug Discovery, Dihydrofolate reductase, parasitic diseases, medicine, 030304 developmental biology, X-ray crystallography, 0303 health sciences, biology, 030306 microbiology, Chemistry, biology.organism_classification, medicine.disease, 3. Good health, Pteridine reductase, Antifolate drug, Derivatives, Dual inhibitor, Pyrimethamine, Structure–activity relationship, RS1-441, pyrimethamine, derivatives, Trypanosoma, biology.protein, Molecular Medicine, Medicine, medicine.drug, Fexinidazole
وصف الملف: application/pdf
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المؤلفون: Massimo Olivucci, Maurizio Orlandini, G. Tassone, Cecilia Pozzi
المصدر: Biomolecules
Volume 11
Issue 5
Biomolecules, Vol 11, Iss 645, p 645 (2021)مصطلحات موضوعية: Models, Molecular, Bile acids, Chicken liver bile acid‐binding protein, Cholic acid, Fatty acid‐binding protein, High‐resolution crystal structure, X‐ray crystallography, Amino Acid Sequence, Animals, Bile Acids and Salts, Binding Sites, Carrier Proteins, Chickens, Cholic Acid, Crystallography, X-Ray, Drug Delivery Systems, Liver, Membrane Glycoproteins, Protein Binding, Recombinant Proteins, Bile acid binding, Biochemistry, law.invention, chemistry.chemical_compound, Models, law, fatty acid-binding protein, 0303 health sciences, Crystallography, Photoswitch, Chemistry, 030302 biochemistry & molecular biology, QR1-502, cholic acid, Recombinant DNA, chicken liver bile acid-binding protein, Drug carrier, Cell signaling, Microbiology, Fatty acid-binding protein, Article, 03 medical and health sciences, Affinity chromatography, Molecular Biology, 030304 developmental biology, X-ray crystallography, bile acids, Molecular, X-Ray, high-resolution crystal structure
وصف الملف: application/pdf
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المؤلفون: Cecilia Pozzi, Stefano Mangani, Maurizio Botta, G. Tassone
المصدر: Biochimica et Biophysica Acta (BBA) - Proteins and Proteomics. 1866:1190-1198
مصطلحات موضوعية: 0301 basic medicine, Protein Conformation, ATPase, Protozoan Proteins, Biophysics, Biochemistry, Leishmania braziliensis, Analytical Chemistry, 03 medical and health sciences, Adenosine Triphosphate, 0302 clinical medicine, ATP hydrolysis, Heat shock protein, Humans, Selectivity, HSP90 Heat-Shock Proteins, Heat shock protein 90, Cloning, Molecular, Nucleotides, Protozoan parasites, X-ray crystallography, Molecular Biology, Site-directed mutagenesis, chemistry.chemical_classification, Binding Sites, biology, Chemistry, Hydrolysis, biology.organism_classification, Hsp90, 030104 developmental biology, Enzyme, 030220 oncology & carcinogenesis, Chaperone (protein), Mutagenesis, Site-Directed, biology.protein, Brazil, Molecular Chaperones, Protein Binding
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المؤلفون: G. Tassone, Andrei Leitão, Carlos A. Montanari, Mattia Mori, Júlio César Borges, Maurizio Botta, Sérgio L. Ramos, Fernanda Aparecida Heleno Batista
المصدر: Journal of Enzyme Inhibition and Medicinal Chemistry, Vol 35, Iss 1, Pp 639-649 (2020)
مصطلحات موضوعية: Hsp90, RM1-950, 01 natural sciences, Microbiology, inhibitors, parasitic diseases, Drug Discovery, medicine, leishmaniasis, Pharmacology, biology, 010405 organic chemistry, Neglected Disease, food and beverages, Leishmaniasis, General Medicine, biology.organism_classification, medicine.disease, Leishmania braziliensis, Small molecule, molecular modelling, 0104 chemical sciences, 010404 medicinal & biomolecular chemistry, Chaperone (protein), biology.protein, Protozoa, Therapeutics. Pharmacology, fluorescence
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::e3285e7e93987640c3a9c8111b42723c