-
1
المؤلفون: Elisabetta Armani, Andrea Rizzi, Nicolò Iotti, Francesca Saccani, Maria Rosaria Di Lascia, Laura Tigli, Alice Pappani, Gessica Marchini, Annalisa Murgo, Anna Maria Capelli, Maurizio Delcanale, Paola Puccini, Gino Villetti, Maurizio Civelli, Claudia Beato, Marta Giuliani, Claudia Mundi, Francesca Murarolli, Mafalda Pagano, Luca F. Raveglia, Rosaria Remelli, Gabriele Amari
المصدر: Journal of Medicinal Chemistry. 66:5622-5656
مصطلحات موضوعية: Drug Discovery, Molecular Medicine
-
2
المؤلفون: Maurizio Civelli, Anna Rita Pisano, Gino Villetti, Hervé Van de Poël, Francesco Amadei, Vanessa Pitozzi, Carmelida Capaldi, Gabriele Amari, Alice Pappani, Michela Salvadori, Fanti Renato De, Paola Puccini, Valentina Cenacchi, Wesley Blackaby, Maurizio Delcanale, Riccardo Patacchini, Kevin Nash, Andrea Rizzi, Gessica Marchini, Maria Pittelli, Marcello Trevisani, Elisabetta Armani, Charles Baker-Glenn
المصدر: Journal of Medicinal Chemistry. 64:9100-9119
مصطلحات موضوعية: chemistry.chemical_classification, 0303 health sciences, Antagonist, Muscarinic acetylcholine receptor M3, Pharmacology, 01 natural sciences, In vitro, 0104 chemical sciences, 010404 medicinal & biomolecular chemistry, 03 medical and health sciences, Enzyme, chemistry, In vivo, Drug Discovery, Muscarinic acetylcholine receptor, Molecular Medicine, Intracellular, Ex vivo, 030304 developmental biology
-
3
المؤلفون: Elisabetta, Armani, Andrea, Rizzi, Carmelida, Capaldi, Renato, De Fanti, Maurizio, Delcanale, Gino, Villetti, Gessica, Marchini, Anna Rita, Pisano, Vanessa, Pitozzi, Maria Gloria, Pittelli, Marcello, Trevisani, Michela, Salvadori, Valentina, Cenacchi, Paola, Puccini, Francesco, Amadei, Alice, Pappani, Maurizio, Civelli, Riccardo, Patacchini, Charles A G, Baker-Glenn, Hervé, Van de Poël, Wesley P, Blackaby, Kevin, Nash, Gabriele, Amari
المصدر: Journal of medicinal chemistry. 64(13)
مصطلحات موضوعية: Male, Receptor, Muscarinic M3, Dose-Response Relationship, Drug, Molecular Structure, Guinea Pigs, Cyclic Nucleotide Phosphodiesterases, Type 4, Rats, Rats, Sprague-Dawley, Pulmonary Disease, Chronic Obstructive, Structure-Activity Relationship, Rats, Inbred BN, Drug Discovery, Animals, Phosphodiesterase 4 Inhibitors
-
4
المؤلفون: Maurizio Civelli, Alice Pappani, Paola Puccini, Elisabetta Armani, Laura Carzaniga, Silvia Catinella, Roberta Volta, Riccardo Patacchini, Gabriele Amari, Valentina Cenacchi, Maurizio Delcanale, Fabrizio Facchinetti, Chiara Carnini, Carmelida Capaldi, Silvia Capacchi, Andrea Rizzi, Gessica Marchini, Valentina Bagnacani, Gino Villetti, Nadia Moretto, Loredana Battipaglia, Paola Caruso, Francesco Amadei, Eleonora Ghidini, Fanti Renato De
المصدر: Journal of Medicinal Chemistry. 60:10026-10046
مصطلحات موضوعية: Male, 0301 basic medicine, Drug, Pyrrolidines, media_common.quotation_subject, Respiratory Tract Diseases, Drug Evaluation, Preclinical, Pharmacology, Pathogenesis, Structure-Activity Relationship, 03 medical and health sciences, 0302 clinical medicine, Drug Stability, Pharmacokinetics, Rats, Inbred BN, Administration, Inhalation, Drug Discovery, Animals, Humans, Structure–activity relationship, Pulmonary Eosinophilia, ADME, media_common, chemistry.chemical_classification, Binding Sites, Dose-Response Relationship, Drug, Chemistry, Drug discovery, In vitro, Cyclic Nucleotide Phosphodiesterases, Type 4, Thiazoles, 030104 developmental biology, Enzyme, 030220 oncology & carcinogenesis, Molecular Medicine, Phosphodiesterase 4 Inhibitors
-
5
المؤلفون: Monica Borgatti, Eugenia Prus, Ilaria Lampronti, Gabriele Amari, Nicoletta Bianchi, Eitan Fibach, Francesco Chiavilli, Cristina Zuccato, Cristiano Chiarabelli, Roberto Gambari, Maurizio Delcanale
المصدر: European Journal of Pharmacology. 752:84-91
مصطلحات موضوعية: Cellular differentiation, Cell, Biology, NO, Patents as Topic, Erythroid Cells, hemic and lymphatic diseases, Fetal hemoglobin, Gene expression, medicine, Humans, gamma-Globins, Erythroid differentiation, Fetal Hemoglobin, Erythroid Precursor Cells, Cell Proliferation, Pharmacology, Regulation of gene expression, Butyrate analogues, Foetal haemoglobin production γ-globin mRNA induction, Real-time PCR, Butyric Acid, Cell Differentiation, Gene Expression Regulation, K562 Cells, beta-Thalassemia, Medicine (all), Cell growth, Molecular biology, medicine.anatomical_structure, Biochemistry, K562 cells
-
6
المؤلفون: Maurizio Civelli, Carola Buccellati, Angelo Sala, Fabrizio Facchinetti, Laura Carzaniga, Eleonora Ghidini, Gabriele Amari, Fanti Renato De, Fiorella Pastore, Chiara Carnini, Paola Caruso, Maurizio Delcanale, Elisabetta Armani, Gino Villetti, Carmelida Capaldi, Riccardo Patacchini, Gessica Marchini, Andrea Rizzi, Emilio Hirsch, Raffaella Bosco, Nadia Moretto
المصدر: Journal of Pharmacology and Experimental Therapeutics. 352:559-567
مصطلحات موضوعية: Male, Administration, Topical, Anti-Inflammatory Agents, Pharmacology, Peripheral blood mononuclear cell, Rats, Sprague-Dawley, chemistry.chemical_compound, Rats, Inbred BN, Administration, Inhalation, medicine, Animals, Rolipram, Roflumilast, Nicotinamide, Cilomilast, Ferrets, Phosphodiesterase, Neutrophilia, Cyclic Nucleotide Phosphodiesterases, Type 4, Rats, Mice, Inbred C57BL, chemistry, Molecular Medicine, Tumor necrosis factor alpha, Phosphodiesterase 4 Inhibitors, medicine.symptom, medicine.drug
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::a255b5f8419c48e073070d82ed43f5c9
https://doi.org/10.1124/jpet.114.220541 -
7
المؤلفون: Gabriele Amari, Puccini Paola, Roberto Gambari, Eleonora Ghidini, Felicia D'Andrea, Giorgio Catelani, M. Landi, Nicoletta Bianchi
المصدر: European Journal of Medicinal Chemistry. 44:745-754
مصطلحات موضوعية: Stereochemistry, Cellular differentiation, Pentoses, Antineoplastic Agents, Structure-Activity Relationship, Erythroid Cells, Drug Discovery, medicine, Humans, Urea, Structure–activity relationship, Inducer, Erythroid differentiation, K562 cells, Pharmacology, Chemistry, Monosaccharides, Organic Chemistry, Galactose, Cell Differentiation, General Medicine, medicine.disease, Carbamides, In vitro, Cell biology, Leukemia, Glucose, Aminosugar, Cell culture, Carbamides, Monosaccharides, Erythroid differentiation, K562 cells, Leukemia, Erythroblastic, Acute, Drug Screening Assays, Antitumor
-
8
المؤلفون: Elisabetta Armani, Alessio Lodola, Marco Mor, Silvia Ghirardi, Silvia Rivara, Gabriele Amari, Paola Lorenza Caruso, Milco Lipreri, Maurizio Delcanale, Maurizio Civelli, Elisabetta Galbiati
المصدر: Bioorganic & Medicinal Chemistry. 12:3763-3782
مصطلحات موضوعية: Selective Estrogen Receptor Modulators, Spectrometry, Mass, Electrospray Ionization, Magnetic Resonance Spectroscopy, Stereochemistry, Clinical Biochemistry, Drug Evaluation, Preclinical, Substituent, Pharmaceutical Science, Biochemistry, Structure-Activity Relationship, chemistry.chemical_compound, Drug Discovery, Animals, Humans, Structure–activity relationship, Benzopyrans, Binding site, Molecular Biology, Estrogen receptor beta, Organic Chemistry, Biological activity, Rats, Benzopyran, Receptors, Estrogen, chemistry, Docking (molecular), Molecular Medicine, Female, Estrogen receptor alpha
-
9
المؤلفون: Maurizio Delcanale, Elisabetta Galbiati, Elisabetta Armani, Paola Caruso, Maurizio Civelli, Gabriele Amari, Silvia Ghirardi
المصدر: Journal of Pharmacology and Experimental Therapeutics. 303:196-203
مصطلحات موضوعية: medicine.medical_specialty, medicine.drug_class, 9,10-Dimethyl-1,2-benzanthracene, Ovariectomy, DMBA, Pharmacology, Rats, Sprague-Dawley, Piperidines, Bone Density, Oral administration, In vivo, Internal medicine, medicine, Animals, Anticarcinogenic Agents, Estrogen Receptor beta, Humans, Potency, Benzopyrans, Raloxifene, Dose-Response Relationship, Drug, Molecular Structure, Chemistry, Uterus, Estrogen Receptor alpha, Antagonist, Mammary Neoplasms, Experimental, Estrogens, Organ Size, Rats, Endocrinology, Receptors, Estrogen, Estrogen, Raloxifene Hydrochloride, Ovariectomized rat, Molecular Medicine, Female, medicine.drug
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::0956ef2fd54de7a602998324e2cc6389
https://doi.org/10.1124/jpet.102.038034 -
10
المؤلفون: Gabriele Amari, Elisabetta Galbiati, Elisabetta Armani, Maurizio Civelli, Maurizio Delcanale, Paola Caruso, Silvia Ghirardi
المصدر: Journal of Pharmacology and Experimental Therapeutics. 300:802-809
مصطلحات موضوعية: Selective Estrogen Receptor Modulators, medicine.medical_specialty, Eosinophil Peroxidase, Pyrrolidines, medicine.drug_class, Ovariectomy, Estrogen receptor, In Vitro Techniques, Pharmacology, Ethinyl Estradiol, Partial agonist, Rats, Sprague-Dawley, chemistry.chemical_compound, Estradiol Congeners, Piperidines, Bone Density, Internal medicine, medicine, Animals, Estrogen Receptor beta, Humans, Benzopyrans, Dose-Response Relationship, Drug, Cholesterol, Uterus, Estrogen Antagonists, Estrogen Receptor alpha, Antagonist, Rats, Endocrinology, Peroxidases, Receptors, Estrogen, chemistry, Estrogen, Selective estrogen receptor modulator, Ovariectomized rat, Molecular Medicine, Female, Levormeloxifene, hormones, hormone substitutes, and hormone antagonists, medicine.drug
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::cdf5a7c2786a6dfb11e34f355b47f2f0
https://doi.org/10.1124/jpet.300.3.802