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المؤلفون: Gary J. Hom, William A. Schutt, Gabor M. Rubanyi
مصطلحات موضوعية: medicine.medical_specialty, Blood pressure, Chemistry, Internal medicine, medicine, Cardiology, Transient (oscillation), Endothelin receptor
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_________::27d35150d204cf66f8a5f49d5ec9df69
https://doi.org/10.1159/000418350 -
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المؤلفون: Doreen E. Cashen, Erin McGowan, Jennifer E. Drisko, Ravi P. Nargund, William J. Martin, D. Euan MacIntyre, Gary J Hom, Iyassu K. Sebhat, Lex H.T. Van der Ploeg, Liza Gantert, Andrew D. Howard
المصدر: European Journal of Pharmacology. 454:71-79
مصطلحات موضوعية: Male, Agonist, medicine.medical_specialty, medicine.drug_class, Binding, Competitive, Peptides, Cyclic, Piperazines, Rats, Sprague-Dawley, Tetrahydroisoquinolines, Internal medicine, medicine, Animals, Agouti-Related Protein, ACTH receptor, Receptor, Pharmacology, Camphanes, Dose-Response Relationship, Drug, Chemistry, Penile Erection, digestive, oral, and skin physiology, Antagonist, Triazoles, Isoquinolines, Receptor antagonist, Peptide Fragments, Rats, Apomorphine, Endocrinology, Receptors, Corticotropin, THIQ, Receptor, Melanocortin, Type 4, Melanocortin, hormones, hormone substitutes, and hormone antagonists, medicine.drug
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المؤلفون: Ralph A. Stearns, Randy R. Miller, William J. Martin, Ravi P. Nargund, Erin McGowan, Lex H.T. Van der Ploeg, and Arthur A. Patchett, Andrew D. Howard, David B. R. Johnston, D. Euan MacIntyre, Rubana N. Kalyani, Khaled Barakat, Raman K. Bakshi, Ralph T. Mosley, Jennifer E. Drisko, Constantin Tamvakopoulos, Rui Tang, Alison M. Strack, Zhixiong Ye, Doreen E. Cashen, Tanya MacNeil, David H. Weinberg, Palucki Brenda, Gary J Hom, Iyassu K. Sebhat
المصدر: Journal of Medicinal Chemistry. 45:4589-4593
مصطلحات موضوعية: Agonist, Chemistry, medicine.drug_class, Biological activity, Pharmacology, Melanocortin receptor, THIQ, Drug Discovery, medicine, Anorectic, Molecular Medicine, Structure–activity relationship, Melanocortin, Receptor, medicine.drug
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المؤلفون: Lawrence F. Colwell, William P. Feeney, Liping Deng, Michael J. Forrest, Randy R. Miller, Ralph A. Stearns, Ann E. Weber, Mari R. Candelore, Gary J Hom, D. E. Macintyre, Mathew J. Wyvratt, Dawn Chitty, Robert J. Mathvink, Tolman Js, Laurie Tota, Margaret A. Cascieri, M. H. Fisher
المصدر: Journal of Medicinal Chemistry. 43:3832-3836
مصطلحات موضوعية: Glycerol, Male, Agonist, Beta-3 adrenergic receptor, Stereochemistry, medicine.drug_class, Administration, Oral, Biological Availability, Adrenergic beta-3 Receptor Agonists, CHO Cells, Chemical synthesis, Radioligand Assay, Structure-Activity Relationship, chemistry.chemical_compound, Dogs, Cricetinae, Drug Discovery, medicine, Animals, Humans, Cloning, Molecular, Thiazole, Beta (finance), Sulfonamides, Trifluoromethyl, Adrenergic beta-Agonists, Macaca mulatta, Rats, Thiazoles, chemistry, Receptors, Adrenergic, beta-3, Molecular Medicine, Receptors, Adrenergic, beta-2, Receptors, Adrenergic, beta-1, Pharmacophore
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المؤلفون: Ann E. Weber, Michael J. Forrest, Matthew J. Wyvratt, D. Euan MacIntyre, Mari R. Candelore, Linda Brockunier, Gary J Hom, Emma R. Parmee, Lawrence F. Colwell, Hyun O. Ok, Margaret A. Cascieri, Michael H. Fisher, Liping Deng, William P. Feeney, Laurie Tota
المصدر: Bioorganic & Medicinal Chemistry Letters. 10:2111-2114
مصطلحات موضوعية: Agonist, 1,2,3-Triazole, Stereochemistry, medicine.drug_class, Lipolysis, Clinical Biochemistry, Administration, Oral, Biological Availability, Pharmaceutical Science, Adrenergic beta-3 Receptor Agonists, CHO Cells, Biochemistry, Chemical synthesis, Structure-Activity Relationship, chemistry.chemical_compound, Dogs, In vivo, Cricetinae, Tachycardia, Drug Discovery, Cyclic AMP, medicine, Animals, Humans, Structure–activity relationship, Infusions, Parenteral, Receptor, Molecular Biology, Sulfonamides, Dose-Response Relationship, Drug, Organic Chemistry, Isoproterenol, Triazoles, Macaca mulatta, chemistry, Receptors, Adrenergic, beta-3, Molecular Medicine, Protein Binding
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المؤلفون: Ann E. Weber, Thomas L. Shih, Michael J. Forrest, Randall R. Miller, Michael H. Fisher, Matthew J. Wyvratt, Catherine D. Strader, Margaret A. Cascieri, Liping Deng, Ralph A. Stearns, D. Euan MacIntyre, William P. Feeney, Mari R. Candelore, Gary J Hom, Lawrence F. Colwell, Laurie Tota, Shuet-Hing Lee Chiu
المصدر: Bioorganic & Medicinal Chemistry Letters. 9:1251-1254
مصطلحات موضوعية: Agonist, medicine.drug_class, Clinical Biochemistry, Administration, Oral, Biological Availability, Tetrazoles, Pharmaceutical Science, Pharmacology, Biochemistry, Inhibitory Concentration 50, Dogs, Pharmacokinetics, In vivo, Oral administration, Drug Discovery, medicine, Animals, Humans, Molecular Biology, ED50, Sulfonamides, Chemistry, Organic Chemistry, Biological activity, Adrenergic beta-Agonists, In vitro, Rats, Bioavailability, Kinetics, Molecular Medicine
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المؤلفون: Matthew J. Wyvratt, Leroy Perkins, Randall R. Miller, Ann E. Weber, William P. Feeney, Vincent J. Colandrea, Michael J. Forrest, Emma R. Parmee, Laurie Tota, Michael H. Fisher, Mari R. Candelore, Gary J Hom, Hyun O. Ok, Elizabeth M. Naylor, Catherine D. Strader, Margaret A. Cascieri, Ralph A. Stearns, Liping Deng, D. Euan MacIntyre
المصدر: Bioorganic & Medicinal Chemistry Letters. 9:749-754
مصطلحات موضوعية: Agonist, Beta-3 adrenergic receptor, medicine.medical_specialty, medicine.drug_class, Clinical Biochemistry, Administration, Oral, Pharmaceutical Science, Adrenergic, Biochemistry, Partial agonist, Structure-Activity Relationship, Dogs, Heart Rate, In vivo, Internal medicine, Receptors, Adrenergic, beta, Drug Discovery, medicine, Animals, Humans, Urea, Lipolysis, Receptor, Adrenergic beta-2 Receptor Agonists, Molecular Biology, ED50, Sulfonamides, Chemistry, Organic Chemistry, Adrenergic beta-Agonists, Macaca mulatta, Endocrinology, Adrenergic beta-1 Receptor Agonists, Receptors, Adrenergic, beta-3, Molecular Medicine
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المؤلفون: Michael J. Forrest, Catherine D. Strader, Ann E. Weber, Matthew J. Wyvratt, Margaret A. Cascieri, Lawrence F. Colwell, Liping Deng, Mari R. Candelore, Gary J Hom, Elizabeth M. Naylor, Laurie Tota, D. Euan MacIntyre, William P. Feeney, Vincent J. Colandrea, Michael H. Fisher, Pei-Ran Wang
المصدر: Bioorganic & Medicinal Chemistry Letters. 8:3087-3092
مصطلحات موضوعية: Male, Agonist, medicine.drug_class, Clinical Biochemistry, Pharmaceutical Science, Pharmacology, Biochemistry, Chemical synthesis, Structure-Activity Relationship, Dogs, Pharmacokinetics, Oral administration, Receptors, Adrenergic, beta, Drug Discovery, medicine, Carnivora, Animals, Humans, Lipolysis, Molecular Biology, Sulfonamides, biology, Chemistry, Organic Chemistry, Fissipedia, Adrenergic beta-Agonists, biology.organism_classification, Macaca mulatta, Receptors, Adrenergic, beta-3, Molecular Medicine, Selectivity
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المؤلفون: Myrna E. Trumbauer, Daniel S. Fletcher, Karen Sokol, Qiao-wen Xie, Gary J Hom, Carl Nathan, Karla Stevens, John D. MacMicking, Nicole A. Chartrain, John S. Mudget, Nancy I. Hutchinson, Howard Y. Chen
المصدر: Cell. 81(4):641-650
مصطلحات موضوعية: Lipopolysaccharide, Molecular Sequence Data, medicine.disease_cause, General Biochemistry, Genetics and Molecular Biology, Microbiology, Mice, chemistry.chemical_compound, Listeria monocytogenes, In vivo, medicine, Animals, Base Sequence, biology, Biochemistry, Genetics and Molecular Biology(all), Wild type, Bacterial Infections, medicine.disease, Shock, Septic, Mice, Mutant Strains, In vitro, Lymphoma, Nitric oxide synthase, chemistry, Shock (circulatory), Immunology, biology.protein, Amino Acid Oxidoreductases, Nitric Oxide Synthase, medicine.symptom