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المؤلفون: Nicola Elaine Press, Clive Mccarthy, Ian N. Bruce, Lewis Whitehead, Lilya Sviridenko, Mrinalini Sachin Oza, Gaynor Elizabeth Pilgrim, Darren Le Grand, Charles Owen, Louise Kirman, Graham Charles Bloomfield, Thomas H. Keller, Peter Finan, Judy Hayler, Mohammed Akhlaq, Denise Head, Emma Budd, Julia Hatto, Bernard Cuenoud, Peter Gedeck, Desmond O'Connor, Brian Cox, Catherine Leblanc
المصدر: Bioorganicmedicinal chemistry letters. 22(17)
مصطلحات موضوعية: Gene isoform, Models, Molecular, Cellular activity, Clinical Biochemistry, Pharmaceutical Science, Alpha (ethology), Bioinformatics, Biochemistry, Mice, Phosphatidylinositol 3-Kinases, Catalytic Domain, Drug Discovery, Animals, Humans, Protein Isoforms, PI3-Kinase Inhibitors, Molecular Biology, Protein Kinase Inhibitors, PI3K/AKT/mTOR pathway, Phosphoinositide-3 Kinase Inhibitors, Kinase, Chemistry, Organic Chemistry, SUPERFAMILY, Rats, Thiazoles, Molecular Medicine, Female, Signal Transduction
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المؤلفون: Deborah Hynx, Claire Ffoulkes-Jones, Gaynor Elizabeth Pilgrim, Sarah Jeffers, Sandra Haberthuer, Elisabeth Schaebulin, John R. Fozard, Thomas H. Keller, Bernard Cuenoud, David Bentley, Katharine L. Turner, Andrew Nicholls, David Beattie, Morris Tweed, Lucy Barker, Sarah Craig, David Beer, Christoph Walker, Paul Kirkham, Rowan Stringer, David Farr, David Andrew Sandham, K D Butler, Colin Howes, Simon J. Watson, Lazzaro Mazzoni, Gillian Spooner, Louise Bidlake, Pamela Tranter, Janet Maas
المصدر: Bioorganicmedicinal chemistry. 12(19)
مصطلحات موضوعية: Stereochemistry, medicine.medical_treatment, Clinical Biochemistry, Pharmaceutical Science, Biological Availability, Thymus Gland, Pharmacology, Biochemistry, Chemical synthesis, Steroid, Cell Line, Structure-Activity Relationship, Glucocorticoid receptor, Receptors, Glucocorticoid, In vivo, Oral administration, Drug Discovery, Eosinophilia, medicine, Structure–activity relationship, Animals, Humans, Molecular Biology, Glucocorticoids, Chemistry, Tumor Necrosis Factor-alpha, Macrophages, Organic Chemistry, Esters, Organ Size, In vitro, Rats, Molecular Medicine, Androstenes, Glucocorticoid, medicine.drug, Protein Binding