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المؤلفون: Georg Rueedi, Cornelia Zumbrunn, Daniel Ritz, Patrick Caspers, Christina Stamm, Daniela Krüsi
المصدر: ChemMedChem. 16:891-897
مصطلحات موضوعية: Models, Molecular, Ribosomal Proteins, Microbial Sensitivity Tests, Crystallography, X-Ray, 01 natural sciences, Biochemistry, Ribosome, Structure-Activity Relationship, chemistry.chemical_compound, Ribosomal protein, Drug Discovery, Escherichia coli, Structure–activity relationship, Benzopyrans, General Pharmacology, Toxicology and Pharmaceutics, Pharmacology, Natural product, Dose-Response Relationship, Drug, Molecular Structure, biology, 010405 organic chemistry, Organic Chemistry, Total synthesis, biology.organism_classification, 16S ribosomal RNA, Anti-Bacterial Agents, 0104 chemical sciences, 010404 medicinal & biomolecular chemistry, chemistry, Molecular Medicine, Efflux, Bacteria
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2
المؤلفون: Peter Seiler, L. Jacob, Swen Seeland, S. Diethelm, N. Tidten-Luksch, Jean-Philippe Surivet, M. Wicki, Georg Rueedi, Jean-Luc Specklin, Michel Enderlin-Paput, Christian Hubschwerlen, Azely Mirre, R. Lange, G. Mathieu, Christine Schmitt, C. Herrmann, Philippe Panchaud, A.-C. Blumstein, A. Mac Sweeney, F. Masse, Daniel Ritz, Jean-Christophe Gauvin, Carmela Gnerre
المصدر: Journal of Medicinal Chemistry. 63:66-87
مصطلحات موضوعية: Gram-negative bacteria, Microbial Sensitivity Tests, Hydroxamic Acids, medicine.disease_cause, Amidohydrolases, In vivo, Gram-Negative Bacteria, Drug Discovery, Hydrolase, Escherichia coli, medicine, Animals, Pyrroles, Enzyme Inhibitors, Escherichia coli Infections, Mice, Inbred ICR, biology, Chemistry, Pseudomonas aeruginosa, biology.organism_classification, Enterobacteriaceae, In vitro, Anti-Bacterial Agents, Multiple drug resistance, Klebsiella pneumoniae, Biochemistry, Molecular Medicine, Female, Bacteria
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3
المؤلفون: Michel Enderlin-Paput, Swen Seeland, A.-C. Blumstein, Daniel Ritz, Peter Seiler, R. Lange, Jean-Philippe Surivet, Christine Schmitt, F. Masse, Jean-Christophe Gauvin, S. Diethelm, L. Jacob, Charlyse Herrmann, Carmela Gnerre, Hans H. Locher, G. Mathieu, Azely Mirre, Georg Rueedi, Philippe Panchaud
المصدر: Journal of medicinal chemistry. 63(1)
مصطلحات موضوعية: Drug, media_common.quotation_subject, Microbial Sensitivity Tests, Pharmacology, Hydroxamic Acids, 01 natural sciences, Amidohydrolases, 03 medical and health sciences, Mice, In vivo, Drug Discovery, Gram-Negative Bacteria, Animals, Solubility, Enzyme Inhibitors, Lead (electronics), Escherichia coli Infections, 030304 developmental biology, media_common, 0303 health sciences, Molecular Structure, Chemistry, 0104 chemical sciences, Anti-Bacterial Agents, Rats, 010404 medicinal & biomolecular chemistry, Hepatocytes, Molecular Medicine, Administration, Intravenous
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4
المؤلفون: Joel Roesslein, Daniel Ritz, Katja Zerbe, Georg Rueedi, Karl Gademann, Patrick Caspers, Hideki Miyatake-Ondozabal, Hiromu Hattori
المصدر: Angewandte Chemie. 130:11186-11190
مصطلحات موضوعية: Glycosylation, Macrocyclic Compounds, medicine.drug_class, Stereochemistry, Antibiotics, Disaccharide, Microbial Sensitivity Tests, Gram-Positive Bacteria, 010402 general chemistry, 01 natural sciences, Catalysis, chemistry.chemical_compound, Drug Resistance, Bacterial, Gram-Negative Bacteria, medicine, Moiety, Biological evaluation, 010405 organic chemistry, Enantioselective synthesis, Total synthesis, Stereoisomerism, General Chemistry, General Medicine, Anti-Bacterial Agents, 0104 chemical sciences, chemistry, Carbohydrate Sequence, Stereoselectivity
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5
المصدر: ChemCatChem. 10:3786-3794
مصطلحات موضوعية: photochemistry, 010405 organic chemistry, Organic Chemistry, Substrate (chemistry), chemistry.chemical_element, Photoredox catalysis, Homogeneous catalysis, solar-driven transformations, iridium, 010402 general chemistry, homogeneous catalysis, 01 natural sciences, Combinatorial chemistry, Catalysis, 0104 chemical sciences, arylations, Inorganic Chemistry, chemistry, Electrophile, Iridium, Physical and Theoretical Chemistry, Visible spectrum
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المؤلفون: Markus Gude, Georg Rueedi, Thomas Pfeifer, Christian Hubschwerlen, Daniel Ritz, Thierry Kimmerlin, L. Jacob, A.-C. Blumstein, Daniel Bur, Alain Chambovey, Lars Prade, Peter Seiler, Philippe Panchaud, Eric A. Ertel, Thierry Bruyère
المصدر: Journal of Medicinal Chemistry. 60:3755-3775
مصطلحات موضوعية: Potassium Channels, Topoisomerase IV, Stereochemistry, Microbial Sensitivity Tests, 010402 general chemistry, 01 natural sciences, DNA gyrase, chemistry.chemical_compound, Gram-Negative Bacteria, Drug Discovery, Animals, Urea, Isoquinoline, Respiratory Tract Infections, Urea binding, biology, 010405 organic chemistry, Drug discovery, Hydrogen Bonding, Prodrug, Isoquinolines, Anti-Bacterial Agents, Rats, 0104 chemical sciences, Solubility, chemistry, Area Under Curve, biology.protein, Molecular Medicine, Antibacterial activity, Lead compound, Half-Life
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المؤلفون: Thierry Bruyère, Eric A. Ertel, Stephanie Enderlin-Paput, Hans H. Locher, Michel Enderlin-Paput, Daniel Ritz, Christopher Kohl, Jean-Christophe Gauvin, Patrick Hess, Jean-Philippe Surivet, Azely Mirre, Daniel Bur, Cornelia Zumbrunn, Georg Rueedi, Christian Hubschwerlen, Peter Seiler
المصدر: Journal of Medicinal Chemistry. 60:3776-3794
مصطلحات موضوعية: 0301 basic medicine, Gram-negative bacteria, Topoisomerase Inhibitors, medicine.drug_class, Topoisomerase IV, Guinea Pigs, 030106 microbiology, Microbial Sensitivity Tests, 01 natural sciences, DNA gyrase, Microbiology, 03 medical and health sciences, Gram-Negative Bacteria, Drug Discovery, medicine, Animals, Humans, Myocytes, Cardiac, Pyrans, biology, 010405 organic chemistry, Chemistry, Topoisomerase, biology.organism_classification, Anti-Bacterial Agents, 0104 chemical sciences, Acinetobacter baumannii, Multiple drug resistance, Biochemistry, biology.protein, Molecular Medicine, Antibacterial activity, Topoisomerase inhibitor
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8
المؤلفون: Daniel Ritz, Daniel Boehringer, Georg Rueedi, Marc Leibundgut, Patrick Caspers, Daniel Bur, Alain Scaiola, Hans H. Locher
المصدر: Scientific Reports
Scientific Reports, 9
Scientific Reports, Vol 9, Iss 1, Pp 1-9 (2019)مصطلحات موضوعية: 0301 basic medicine, Staphylococcus aureus, RNA, Transfer, Met, Peptidyl transferase, medicine.drug_class, Antibiotics, lcsh:Medicine, Microbial Sensitivity Tests, medicine.disease_cause, Ribosome, Article, Microbiology, 03 medical and health sciences, chemistry.chemical_compound, 0302 clinical medicine, Acetamides, Escherichia coli, medicine, Humans, lcsh:Science, Oxazolidinones, Protein Synthesis Inhibitors, Multidisciplinary, biology, lcsh:R, Cryoelectron Microscopy, Translation (biology), Anti-Bacterial Agents, 030104 developmental biology, chemistry, Peptidyl Transferases, Linezolid, Transfer RNA, Clostridium Infections, biology.protein, lcsh:Q, Ribosomes, 030217 neurology & neurosurgery, Cadazolid, Fluoroquinolones
وصف الملف: application/application/pdf
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9
المؤلفون: Philippe Pfaff, Sarah Diggelmann, Hans H. Locher, Daniel Ritz, Daniel Bur, Georg Rueedi, Patrick Caspers
المصدر: Antimicrobial Agents and Chemotherapy. 61
مصطلحات موضوعية: Ribosomal Proteins, 0301 basic medicine, medicine.drug_class, Ribosomal Protein L3, 030106 microbiology, Antibiotics, Microbial Sensitivity Tests, Biology, Microbiology, 03 medical and health sciences, chemistry.chemical_compound, Mechanisms of Resistance, Ribosomal protein, 23S ribosomal RNA, Drug Resistance, Bacterial, medicine, Humans, Pharmacology (medical), Amino Acid Sequence, Gene, Oxazolidinones, Protein Synthesis Inhibitors, Pharmacology, Clostridioides difficile, Linezolid, Sequence Analysis, DNA, Ribosomal RNA, Clostridium difficile, Virology, Anti-Bacterial Agents, RNA, Ribosomal, 23S, Infectious Diseases, chemistry, Genome, Bacterial, Cadazolid
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::2972c0889973ad604ad75534d0b8e1e6
https://doi.org/10.1128/aac.00384-17 -
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المؤلفون: Daniel Bur, Azely Mirre, Michel Enderlin-Paput, Georg Rueedi, Christian Hubschwerlen, Hans H. Locher, Daniel Ritz, Cornelia Zumbrunn, Wolfgang Keck, Maria Boehme, Marina Dos Santos, Jean-Christophe Gauvin, Peter Seiler, Jean-Philippe Surivet, Verena Kaegi, Jonathan Delers, Christopher Kohl, Thierry Bruyère, Mika Gaertner
المصدر: Journal of Medicinal Chemistry. 56:7396-7415
مصطلحات موضوعية: DNA Topoisomerase IV, Protein Conformation, Topoisomerase Inhibitors, Topoisomerase IV, medicine.drug_class, hERG, Chemistry Techniques, Synthetic, Pharmacology, Gram-Positive Bacteria, DNA gyrase, Inhibitory Concentration 50, Mice, Structure-Activity Relationship, chemistry.chemical_compound, Drug Discovery, medicine, Animals, Humans, Topoisomerase II Inhibitors, Pyrans, biology, Topoisomerase, Tetrahydropyran, Anti-Bacterial Agents, Rats, Molecular Docking Simulation, chemistry, Biochemistry, DNA Gyrase, Drug Design, biology.protein, Molecular Medicine, Female, Antibacterial activity, DNA Topoisomerases, Topoisomerase inhibitor, DNA