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المؤلفون: Elisabetta Armani, Andrea Rizzi, Nicolò Iotti, Francesca Saccani, Maria Rosaria Di Lascia, Laura Tigli, Alice Pappani, Gessica Marchini, Annalisa Murgo, Anna Maria Capelli, Maurizio Delcanale, Paola Puccini, Gino Villetti, Maurizio Civelli, Claudia Beato, Marta Giuliani, Claudia Mundi, Francesca Murarolli, Mafalda Pagano, Luca F. Raveglia, Rosaria Remelli, Gabriele Amari
المصدر: Journal of Medicinal Chemistry. 66:5622-5656
مصطلحات موضوعية: Drug Discovery, Molecular Medicine
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2
المؤلفون: Maurizio Civelli, Anna Rita Pisano, Gino Villetti, Hervé Van de Poël, Francesco Amadei, Vanessa Pitozzi, Carmelida Capaldi, Gabriele Amari, Alice Pappani, Michela Salvadori, Fanti Renato De, Paola Puccini, Valentina Cenacchi, Wesley Blackaby, Maurizio Delcanale, Riccardo Patacchini, Kevin Nash, Andrea Rizzi, Gessica Marchini, Maria Pittelli, Marcello Trevisani, Elisabetta Armani, Charles Baker-Glenn
المصدر: Journal of Medicinal Chemistry. 64:9100-9119
مصطلحات موضوعية: chemistry.chemical_classification, 0303 health sciences, Antagonist, Muscarinic acetylcholine receptor M3, Pharmacology, 01 natural sciences, In vitro, 0104 chemical sciences, 010404 medicinal & biomolecular chemistry, 03 medical and health sciences, Enzyme, chemistry, In vivo, Drug Discovery, Muscarinic acetylcholine receptor, Molecular Medicine, Intracellular, Ex vivo, 030304 developmental biology
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3
المؤلفون: Elisabetta, Armani, Andrea, Rizzi, Carmelida, Capaldi, Renato, De Fanti, Maurizio, Delcanale, Gino, Villetti, Gessica, Marchini, Anna Rita, Pisano, Vanessa, Pitozzi, Maria Gloria, Pittelli, Marcello, Trevisani, Michela, Salvadori, Valentina, Cenacchi, Paola, Puccini, Francesco, Amadei, Alice, Pappani, Maurizio, Civelli, Riccardo, Patacchini, Charles A G, Baker-Glenn, Hervé, Van de Poël, Wesley P, Blackaby, Kevin, Nash, Gabriele, Amari
المصدر: Journal of medicinal chemistry. 64(13)
مصطلحات موضوعية: Male, Receptor, Muscarinic M3, Dose-Response Relationship, Drug, Molecular Structure, Guinea Pigs, Cyclic Nucleotide Phosphodiesterases, Type 4, Rats, Rats, Sprague-Dawley, Pulmonary Disease, Chronic Obstructive, Structure-Activity Relationship, Rats, Inbred BN, Drug Discovery, Animals, Phosphodiesterase 4 Inhibitors
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4
المؤلفون: Maurizio Civelli, Alice Pappani, Paola Puccini, Elisabetta Armani, Laura Carzaniga, Silvia Catinella, Roberta Volta, Riccardo Patacchini, Gabriele Amari, Valentina Cenacchi, Maurizio Delcanale, Fabrizio Facchinetti, Chiara Carnini, Carmelida Capaldi, Silvia Capacchi, Andrea Rizzi, Gessica Marchini, Valentina Bagnacani, Gino Villetti, Nadia Moretto, Loredana Battipaglia, Paola Caruso, Francesco Amadei, Eleonora Ghidini, Fanti Renato De
المصدر: Journal of Medicinal Chemistry. 60:10026-10046
مصطلحات موضوعية: Male, 0301 basic medicine, Drug, Pyrrolidines, media_common.quotation_subject, Respiratory Tract Diseases, Drug Evaluation, Preclinical, Pharmacology, Pathogenesis, Structure-Activity Relationship, 03 medical and health sciences, 0302 clinical medicine, Drug Stability, Pharmacokinetics, Rats, Inbred BN, Administration, Inhalation, Drug Discovery, Animals, Humans, Structure–activity relationship, Pulmonary Eosinophilia, ADME, media_common, chemistry.chemical_classification, Binding Sites, Dose-Response Relationship, Drug, Chemistry, Drug discovery, In vitro, Cyclic Nucleotide Phosphodiesterases, Type 4, Thiazoles, 030104 developmental biology, Enzyme, 030220 oncology & carcinogenesis, Molecular Medicine, Phosphodiesterase 4 Inhibitors
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المؤلفون: Fabrizio Facchinetti, Gessica Marchini, Silvia Carnevali
المصدر: European journal of pharmacology. 850
مصطلحات موضوعية: 0301 basic medicine, Agonist, Transcriptional Activation, Leucine zipper, medicine.drug_class, Myocytes, Smooth Muscle, Active Transport, Cell Nucleus, Bronchi, Pharmacology, Cigarette Smoking, 03 medical and health sciences, chemistry.chemical_compound, Transactivation, 0302 clinical medicine, Receptors, Glucocorticoid, Formoterol Fumarate, medicine, Humans, Phosphorylation, Receptor, Cell Nucleus, Forskolin, Chemistry, Beclomethasone, respiratory tract diseases, 030104 developmental biology, Salmeterol, Formoterol, hormones, hormone substitutes, and hormone antagonists, 030217 neurology & neurosurgery, medicine.drug, Transcription Factors
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المؤلفون: Alessandro Fioni, Anna Maria Capelli, Chiara Carnini, Gessica Marchini, Fabio Rancati, Valentina Cenacchi, Eleonora Ghidini, Fabrizio Facchinetti
المصدر: Journal of medicinal chemistry. 61(11)
مصطلحات موضوعية: Agonist, Budesonide, medicine.drug_class, Protein Conformation, Drug design, CHO Cells, Pharmacology, 01 natural sciences, 03 medical and health sciences, Mice, 0302 clinical medicine, Cricetulus, Receptors, Glucocorticoid, In vivo, Adrenal Cortex Hormones, Drug Discovery, Administration, Inhalation, medicine, Animals, Humans, Tissue Distribution, Receptor, Asthma, Lung, Inhalation, 010405 organic chemistry, Chemistry, Pneumonia, medicine.disease, 0104 chemical sciences, Molecular Docking Simulation, medicine.anatomical_structure, RAW 264.7 Cells, 030220 oncology & carcinogenesis, Drug Design, Molecular Medicine, medicine.drug
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7
المؤلفون: Stefano Cavalli, Fabrizio Facchinetti, Alessandro Accetta, Silvia Cantoni, Gino Villetti, Fiorella Pastore, Gessica Marchini, Serena Bertolini
المصدر: Pulmonary Circulation and Pulmonary Vascular Disease.
مصطلحات موضوعية: Kinase, business.industry, Endothelin receptor antagonist, Pharmacology, medicine.disease, Pulmonary hypertension, chemistry.chemical_compound, chemistry, Rho kinase inhibitor, medicine.artery, Pulmonary artery, Medicine, ROCK1, business, Rho-associated protein kinase, Macitentan
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_________::0da2e2cefd6ed26a9572e30afad9ad64
https://doi.org/10.1183/1393003.congress-2017.pa2379 -
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المؤلفون: Fabrizio Facchinetti, Silvia Cantoni, Alessandro Accetta, Gessica Marchini, Stefano Cavalli, Gino Villetti, Maurizio Civelli, Fiorella Pastore, Serena Bertolini
المصدر: European Heart Journal. 38
مصطلحات موضوعية: business.industry, Rho kinase inhibitor, Medicine, Pharmacology, Cardiology and Cardiovascular Medicine, business, medicine.disease, Pulmonary hypertension
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_________::6eba69cc2df93bb686d3a3cea554e15f
https://doi.org/10.1093/eurheartj/ehx501.p726 -
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المؤلفون: Fabrizio Facchinetti, Eleonora Ghidini, Valentina Cenacchi, Anna Maria Capelli, A. Virdis, A. Italia, Chiara Carnini, Gessica Marchini
المصدر: Steroids. 95:88-95
مصطلحات موضوعية: Lipopolysaccharides, Male, Transcriptional Activation, Ovalbumin, medicine.drug_class, Administration, Topical, Prednisolone, Myocytes, Smooth Muscle, Clinical Biochemistry, Active Transport, Cell Nucleus, Anti-Inflammatory Agents, Pharmacology, Nitric Oxide, Biochemistry, Anti-inflammatory, Cell Line, Mice, Receptors, Glucocorticoid, Endocrinology, Glucocorticoid receptor, Pharmacokinetics, Drug Discovery, Eosinophilia, medicine, Animals, Humans, Potency, Lung, Molecular Biology, Dexamethasone, Cell Nucleus, Dose-Response Relationship, Drug, Tumor Necrosis Factor-alpha, Chemistry, Macrophages, Interleukin-8, Organic Chemistry, Isoxazoles, Protein Structure, Tertiary, Rats, Molecular Docking Simulation, Receptors, Mineralocorticoid, medicine.anatomical_structure, Corticosteroid, Transcription Factors, medicine.drug
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10
المؤلفون: Maurizio Civelli, Carola Buccellati, Angelo Sala, Fabrizio Facchinetti, Laura Carzaniga, Eleonora Ghidini, Gabriele Amari, Fanti Renato De, Fiorella Pastore, Chiara Carnini, Paola Caruso, Maurizio Delcanale, Elisabetta Armani, Gino Villetti, Carmelida Capaldi, Riccardo Patacchini, Gessica Marchini, Andrea Rizzi, Emilio Hirsch, Raffaella Bosco, Nadia Moretto
المصدر: Journal of Pharmacology and Experimental Therapeutics. 352:559-567
مصطلحات موضوعية: Male, Administration, Topical, Anti-Inflammatory Agents, Pharmacology, Peripheral blood mononuclear cell, Rats, Sprague-Dawley, chemistry.chemical_compound, Rats, Inbred BN, Administration, Inhalation, medicine, Animals, Rolipram, Roflumilast, Nicotinamide, Cilomilast, Ferrets, Phosphodiesterase, Neutrophilia, Cyclic Nucleotide Phosphodiesterases, Type 4, Rats, Mice, Inbred C57BL, chemistry, Molecular Medicine, Tumor necrosis factor alpha, Phosphodiesterase 4 Inhibitors, medicine.symptom, medicine.drug
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::a255b5f8419c48e073070d82ed43f5c9
https://doi.org/10.1124/jpet.114.220541