-
1دورية أكاديمية
المؤلفون: Inga R. Grin, Grigory V. Mechetin, Rustem D. Kasymov, Evgeniia A. Diatlova, Anna V. Yudkina, Sergei N. Shchelkunov, Irina P. Gileva, Alexandra A. Denisova, Grigoriy A. Stepanov, Ghermes G. Chilov, Dmitry O. Zharkov
المصدر: Molecules, Vol 26, Iss 21, p 6668 (2021)
مصطلحات موضوعية: DNA repair, uracil–DNA glycosylase, inhibitors, virtual screening, pyrimidines, Organic chemistry, QD241-441
وصف الملف: electronic resource
-
2
المؤلفون: Michael G. Medvedev, Oleg V. Stroganov, Artem O. Dmitrienko, Maria V. Panova, Alexey A. Lisov, Igor V. Svitanko, Fedor N. Novikov, Ghermes G. Chilov
المصدر: Mendeleev Communications. 32:735-738
مصطلحات موضوعية: General Chemistry
-
3
المؤلفون: Rustem D. Kasymov, Evgeniia A. Diatlova, Grigoriy A. Stepanov, Grigory V. Mechetin, Ghermes G. Chilov, Anna V. Yudkina, I. P. Gileva, Dmitry O. Zharkov, Sergei N. Shchelkunov, Inga R. Grin, Alexandra A. Denisova
المصدر: Molecules
Molecules, Vol 26, Iss 6668, p 6668 (2021)
Volume 26
Issue 21مصطلحات موضوعية: pyrimidines, Deamination, Pharmaceutical Science, DNA repair, Vaccinia virus, Ligands, Article, Analytical Chemistry, chemistry.chemical_compound, QD241-441, Drug Discovery, inhibitors, Humans, uracil–DNA glycosylase, Enzyme Inhibitors, Physical and Theoretical Chemistry, Uracil-DNA Glycosidase, chemistry.chemical_classification, Molecular Structure, Organic Chemistry, Uracil, Base excision repair, virtual screening, Molecular Docking Simulation, Kinetics, Enzyme, chemistry, Biochemistry, Chemistry (miscellaneous), DNA glycosylase, Uracil-DNA glycosylase, Molecular Medicine, Cytosine, DNA
وصف الملف: application/pdf
-
4
المؤلفون: Robert Peter Gale, Oliver G. Ottmann, I.A. Mikhailov, Fedor N. Novikov, Irina Nemchenko, Andrey Zaritskey, Elza Lomaia, Michele Baccarani, Jorge E. Cortes, Ghermes G. Chilov, Nadia Siordia, Ekaterina Chelysheva, Dzhariyat Shikhbabaeva, Oleg Shukhov, Veronika Shulgina, Anna G. Turkina, Olga Vinogradova, Vasily Shuvaev, Evgeniya Shatokhina, Anastasiya Bykova, Anna Petrova
المصدر: Blood. 138:1482-1482
مصطلحات موضوعية: medicine.drug_class, business.industry, Immunology, medicine, Cancer research, breakpoint cluster region, In patient, Cell Biology, Hematology, business, Biochemistry, Tyrosine-kinase inhibitor
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_________::ab1c3da530e1a2eab8f9b71b0fb3b3d5
https://doi.org/10.1182/blood-2021-150120 -
5
المؤلفون: Michael G. Medvedev, Ivan S. Bushmarinov, Oleg V. Stroganov, Maria V. Panova, Igor V. Svitanko, Fedor N. Novikov, Ghermes G. Chilov, Alexey A. Zeifman
المصدر: Mendeleev Communications. 27:224-227
مصطلحات موضوعية: biology, 010405 organic chemistry, Chemistry, Active site, General Chemistry, 010402 general chemistry, 01 natural sciences, Transition state, 0104 chemical sciences, Maxima and minima, Transition state theory, Computational chemistry, biology.protein, Conformational isomerism, Quantum
-
6
المؤلفون: Oleg V. Stroganov, Michael G. Medvedev, Artem O. Dmitrienko, Fedor N. Novikov, Igor S. Gerasimov, Ghermes G. Chilov, Igor V. Svitanko
المصدر: Journal of computer-aided molecular design. 34(2)
مصطلحات موضوعية: Computer science, Context (language use), Ligands, 01 natural sciences, Field (computer science), Small Molecule Libraries, 0103 physical sciences, Drug Discovery, Human-in-the-loop, Aspartic Acid Endopeptidases, Humans, Physical and Theoretical Chemistry, Representation (mathematics), Structure (mathematical logic), Lead Finder, Binding Sites, 010304 chemical physics, Drug discovery, Hydrogen Bonding, Data science, Cathepsins, 0104 chemical sciences, Computer Science Applications, Molecular Docking Simulation, 010404 medicinal & biomolecular chemistry, Drug Design, Predictive power, Thermodynamics, Amyloid Precursor Protein Secretases, Protein Binding
-
7
المؤلفون: Alvina I. Khamidullina, Yulia V. Dutikova, Alexander A. Shtil, Victor V. Tatarskiy, Margarita A. Yastrebova, Fedor N. Novikov, Ekaterina S. Ivanova, Alexei V. Shunaev, Ghermes G. Chilov, Alexei A. Zeifman, Anastasia A. Kalinina
المصدر: International Journal of Oncology.
مصطلحات موضوعية: STAT3 Transcription Factor, 0301 basic medicine, Cancer Research, Cell Survival, Pyridines, Fusion Proteins, bcr-abl, HL-60 Cells, Biology, Mice, 03 medical and health sciences, chemistry.chemical_compound, 0302 clinical medicine, Cell Line, Tumor, Leukemia, Myelogenous, Chronic, BCR-ABL Positive, hemic and lymphatic diseases, medicine, Animals, Humans, Phosphorylation, Protein kinase B, Cell Proliferation, ABL, Ponatinib, breakpoint cluster region, Imatinib, Triazoles, medicine.disease, Xenograft Model Antitumor Assays, 030104 developmental biology, Oncology, chemistry, 030220 oncology & carcinogenesis, Mutation, Cancer research, K562 Cells, Tyrosine kinase, K562 cells, Chronic myelogenous leukemia, medicine.drug
-
8
المؤلفون: Ghermes G. Chilov, Alexey A. Zeifman, Konstantin A. Lyssenko, Ivan S. Bushmarinov, Michael S. Polkovnichenko, Michael G. Medvedev, Igor V. Svitanko, Oleg V. Stroganov, Fedor N. Novikov
المصدر: Mendeleev Communications. 27:500-502
مصطلحات موضوعية: 010405 organic chemistry, Chemistry, fungi, Cationic polymerization, General Chemistry, 010402 general chemistry, Photochemistry, 01 natural sciences, Cycloaddition, 0104 chemical sciences, Catalysis, Delocalized electron, Redistribution (chemistry), Diels–Alder reaction
-
9
المؤلفون: Daniil V. Katkov, Oleg V. Stroganov, Ilya Yu. Titov, Fedor N. Novikov, Igor V. Svitanko, Ghermes G. Chilov, Victor S. Stroylov
المصدر: Mendeleev Communications. 27:349-351
مصطلحات موضوعية: 0301 basic medicine, Free energy perturbation, 03 medical and health sciences, 030104 developmental biology, Molecular model, biology, Stereochemistry, Kinase, Chemistry, biology.protein, Bruton's tyrosine kinase, General Chemistry, Selectivity
-
10
المؤلفون: Ekaterina S. Ivanova, Victor S. Stroylov, Maria Pelecanou, Polyxeni Alexiou, Victor V. Tatarskiy, Marina Sagnou, Murad Vagida, Fedor N. Novikov, Alexander A. Shtil, Ilya Yu. Titov, Ghermes G. Chilov
المصدر: European Journal of Medicinal Chemistry. 198:112331
مصطلحات موضوعية: Models, Molecular, ATP Binding Cassette Transporter, Subfamily B, Curcumin, Cell Survival, Antineoplastic Agents, Apoptosis, Pharmacology, 01 natural sciences, Structure-Activity Relationship, 03 medical and health sciences, chemistry.chemical_compound, Drug Discovery, polycyclic compounds, medicine, Humans, Doxorubicin, Cytotoxicity, 030304 developmental biology, P-glycoprotein, 0303 health sciences, biology, 010405 organic chemistry, Organic Chemistry, General Medicine, Amides, Drug Resistance, Multiple, 0104 chemical sciences, carbohydrates (lipids), Multiple drug resistance, chemistry, Drug Resistance, Neoplasm, Leukemia, Myeloid, Docking (molecular), biology.protein, Efflux, Drug Screening Assays, Antitumor, K562 Cells, K562 cells, medicine.drug