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1
المؤلفون: Yoshitaka Satoh, Gilles Carmel, Frans Baculi, Peter H. Schafer, Laurie LeBrun, Matt Hickman, Thomas O. Daniel, Brian E. Cathers, James Carmichael, Godrej Khambatta, Hon-Wah Man, Mary E Matyskiela, Philip P Chamberlain, Weihong Zhang, Mariko Riley, George W. Muller, Barbra Pagarigan, Gang Lu, Chin-Chun Lu
المصدر: Journal of Medicinal Chemistry. 61:535-542
مصطلحات موضوعية: 0301 basic medicine, Morpholines, Ubiquitin-Protein Ligases, Phthalimides, Crystallography, X-Ray, Heterocyclic Compounds, 4 or More Rings, Ikaros Transcription Factor, 03 medical and health sciences, DDB1, 0302 clinical medicine, Cell Line, Tumor, Drug Discovery, Fluorescence Resonance Energy Transfer, medicine, Humans, Binding site, Lenalidomide, Transcription factor, Piperidones, Adaptor Proteins, Signal Transducing, chemistry.chemical_classification, DNA ligase, biology, Cereblon, Protein Cereblon, Pomalidomide, Molecular biology, Ubiquitin ligase, Cell biology, DNA-Binding Proteins, 030104 developmental biology, chemistry, 030220 oncology & carcinogenesis, Proteolysis, biology.protein, Molecular Medicine, Multiple Myeloma, Peptide Hydrolases, Protein Binding, medicine.drug
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2
المؤلفون: Kevin Ronald Condroski, Matt Hickman, Wei Liu, Laurie LeBrun, Gilles Carmel, Joshua Hansen, Gang Lu, Afshin Mahmoudi, Frans Baculi, Correa Matthew D, Tim Crea, Hon-Wah Man, George W. Muller, Chin-Chun Lu, Alexander L. Ruchelman, Fan Vocanson, Weihong Zhang
المصدر: Journal of Medicinal Chemistry. 61:492-503
مصطلحات موضوعية: 0301 basic medicine, Quantitative structure–activity relationship, biology, 010405 organic chemistry, Chemistry, Stereochemistry, Cereblon, Glutarimide, Protein degradation, 01 natural sciences, Molecular Docking Simulation, 0104 chemical sciences, Ubiquitin ligase, 03 medical and health sciences, chemistry.chemical_compound, 030104 developmental biology, Biochemistry, Docking (molecular), Drug Discovery, biology.protein, Molecular Medicine, Ternary complex
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3
المؤلفون: Alexander L. Ruchelman, Jack Houston, Nai-Yu Wang, Lyn'Al Nosaka, Antonia Lopez-Girona, Takumi Ito, Gilles Carmel, Mary E Matyskiela, Wei Fang, Derek Nguyen, Philip P Chamberlain, Thomas O. Daniel, Karen Miller, Chin-Chun Lu, Barbra Pagarigan, Svetlana Gaidarova, Gang Lu, Shuichan Xu, James Carmichael, Tam Tran, Gabriel C. Lander, Mariko Riley, Brian E. Cathers, Hiroshi Handa
المصدر: Nature. 535:252-257
مصطلحات موضوعية: Models, Molecular, 0301 basic medicine, Ubiquitin-Protein Ligases, Amino Acid Motifs, Antineoplastic Agents, Plasma protein binding, Crystallography, X-Ray, 01 natural sciences, DNA-binding protein, Substrate Specificity, Ikaros Transcription Factor, 03 medical and health sciences, Ubiquitin, Humans, Adaptor Proteins, Signal Transducing, chemistry.chemical_classification, DNA ligase, Binding Sites, Multidisciplinary, biology, 010405 organic chemistry, Chemistry, Phenylurea Compounds, Cereblon, Thalidomide, 0104 chemical sciences, Ubiquitin ligase, Cell biology, DNA-Binding Proteins, 030104 developmental biology, Multiprotein Complexes, Proteolysis, biology.protein, Degron, Peptide Hydrolases, Peptide Termination Factors, Protein Binding
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4دورية أكاديمية
المؤلفون: Mary E. Matyskiela, Gang Lu, Takumi Ito, Barbra Pagarigan, Chin-Chun Lu, Karen Miller, Wei Fang, Nai-Yu Wang, Derek Nguyen, Jack Houston, Gilles Carmel, Tam Tran, Mariko Riley, Lyn'Al Nos
المصدر: Nature, Nature. 535(7611):252-257
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5
المؤلفون: Joshua D, Hansen, Kevin, Condroski, Matthew, Correa, George, Muller, Hon-Wah, Man, Alexander, Ruchelman, Weihong, Zhang, Fan, Vocanson, Tim, Crea, Wei, Liu, Gang, Lu, Frans, Baculi, Laurie, LeBrun, Afshin, Mahmoudi, Gilles, Carmel, Matt, Hickman, Chin-Chun, Lu
المصدر: Journal of medicinal chemistry. 61(2)
مصطلحات موضوعية: Ubiquitin-Protein Ligases, Drug Evaluation, Preclinical, Quantitative Structure-Activity Relationship, Antineoplastic Agents, Phthalimides, Chemistry Techniques, Synthetic, Molecular Docking Simulation, Ikaros Transcription Factor, Proteolysis, Humans, Multiple Myeloma, Piperidones, Adaptor Proteins, Signal Transducing, Peptide Hydrolases, Peptide Termination Factors
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6
المؤلفون: Philip P Chamberlain, Maria Wang, Yoshinori Hirano, Brian E. Cathers, Gilles Carmel, Toshio Hakoshima, Hiroshi Handa, Barbra Pagarigan, Emily Rychak, Yan J Ren, Barbara Chie-Leon, Silvia L. Delker, Laura G. Corral, Tomoyuki Mori, Takumi Ito, Thomas O. Daniel, Antonia Lopez-Girona, Karen Miller, Hideki Ando, Mariko Riley
المصدر: Nature Structural & Molecular Biology. 21:803-809
مصطلحات موضوعية: Protein Conformation, Ubiquitin-Protein Ligases, Molecular Sequence Data, Angiogenesis Inhibitors, Crystallography, X-Ray, Mice, DDB1, Ubiquitin, Structural Biology, medicine, Animals, Humans, Amino Acid Sequence, Lenalidomide, Molecular Biology, Adaptor Proteins, Signal Transducing, biology, Cereblon, Protein Cereblon, IKZF3, Protein Structure, Tertiary, Thalidomide, Ubiquitin ligase, DNA-Binding Proteins, Molecular Docking Simulation, Biochemistry, biology.protein, Cancer research, Sequence Alignment, Peptide Hydrolases, Protein Binding, medicine.drug
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7
المؤلفون: Gengxin Chen, Yan Ren, Anita Gandhi, Peter H. Schafer, Michelle Waldman, Emily Rychak, Antonia Lopez-Girona, Mahan Abbasian, Derek Mendy, Rajesh Chopra, Thomas O. Daniel, Pilgrim Jackson, Anjan Thakurta, Michael Breider, Gilles Carmel, Afshin Mahmoudi, Svetlana Gaidarova, Maria Wang, Brian E. Cathers, Karen Miller
المصدر: British Journal of Haematology
مصطلحات موضوعية: medicine.drug_class, Ubiquitin-Protein Ligases, Biology, Monoclonal antibody, immunomodulatory drugs, Antibody Specificity, Cell Line, Tumor, Gene expression, medicine, Biomarkers, Tumor, RNA Isoforms, Humans, Multiple myeloma, Lenalidomide, cullin 4 ring ligase complex, DNA damage binding protein 1, Adaptor Proteins, Signal Transducing, Haematological Malignancy, Cereblon, cereblon, Antibodies, Monoclonal, Hematology, medicine.disease, Pomalidomide, Molecular biology, Thalidomide, Reverse transcription polymerase chain reaction, Alternative Splicing, myeloma, Drug Resistance, Neoplasm, Cancer research, Biomarker (medicine), Multiple Myeloma, medicine.drug, Peptide Hydrolases
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8
المؤلفون: Peter H. Schafer, Anita Gandhi, Emily Rychak, Svetlana Gaidarova, Brian E. Cathers, Hiroshi Handa, Takumi Ito, Afshin Mahmoudi, Thomas O. Daniel, Antonia Lopez-Girona, Roger Shen-Chu Chen, Jilly F. Evans, Pilgrim Jackson, Mahan Abbasian, Rajesh Chopra, Derek Mendy, Gilles Carmel, Karen Miller, Jian Kang, Satoki Karasawa
المصدر: Leukemia
مصطلحات موضوعية: Cancer Research, Ubiquitin-Protein Ligases, lenalidomide, pomalidomide, Antineoplastic Agents, Pharmacology, DDB1, Adjuvants, Immunologic, antiproliferative, medicine, Humans, immunomodulatory, Lenalidomide, Adaptor Proteins, Signal Transducing, business.industry, Cereblon, cereblon, Ubiquitination, Hematology, Protein Cereblon, Pomalidomide, IKZF3, Thalidomide, myeloma, HEK293 Cells, Oncology, Original Article, Corrigendum, business, medicine.drug, IRF4, Peptide Hydrolases
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::c03579afee9c0c69c2956c87ab3cdc19
http://t2r2.star.titech.ac.jp/cgi-bin/publicationinfo.cgi?q_publication_content_number=CTT100691788 -
9
المؤلفون: Richard A. Alm, Mikael Berg, Bo Xu, Wei Yang, Peter J. Tummino, Daniel J Krosky, Gilles Carmel
المصدر: Biochimica et Biophysica Acta (BBA) - Protein Structure and Molecular Enzymology. 1594:297-306
مصطلحات موضوعية: Stereochemistry, Biophysics, chemistry.chemical_element, Zinc, medicine.disease_cause, Biochemistry, Cofactor, Structural Biology, Escherichia coli, medicine, Cloning, Molecular, Enzyme Inhibitors, Picolinic Acids, Molecular Biology, Edetic Acid, Aldehyde-Lyases, Chelating Agents, chemistry.chemical_classification, Aquifex aeolicus, Helicobacter pylori, ATP synthase, biology, Chemistry, Circular Dichroism, Cobalt, biology.organism_classification, Recombinant Proteins, carbohydrates (lipids), Kinetics, Dicarboxylic acid, Enzyme, Spectrophotometry, biology.protein, lipids (amino acids, peptides, and proteins), Phosphoenolpyruvate carboxykinase, Cadmium
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10
المؤلفون: Tam Tran, Gabriel C. Lander, James Carmichale, Thomas O. Daniel, Svetlana Gaidarova, Mary E Matyskiela, Lyn'Al Nosaka, Antonia Lopez-Girona, Takumi Ito, Alexander L. Ruchelman, Gilles Carmel, Jack Houston, Brian E. Cathers, Philip P Chamberlain, Wei Fang, Hiroshi Handa, Derek Nguyen, Mariko Riley, Karen Miller, Shuichan Xu, Barbra Pagarigan, Gang Lu, Chin-Chu Lu, Nai-Yu Wang
المصدر: Cancer Research. 77:SY37-02
مصطلحات موضوعية: chemistry.chemical_classification, Cancer Research, DNA ligase, biology, Chemistry, Cereblon, Protein Cereblon, Protein degradation, Ubiquitin ligase, Cell biology, DDB1, Oncology, Proteasome, biology.protein, Degron
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_________::2acec69e19aebcc0985034bd9ab2603b
https://doi.org/10.1158/1538-7445.am2017-sy37-02