-
1
المؤلفون: Yao Cheng, Shao Ru Chen, Wing Lam, Xiaoming Yang, Ginger E. Dutschman, Yung-Chi Cheng, Elizabeth A. Gullen, Ya Ha, Alois Fürstner, Samson Francis, David C. Baker, Sangwon Lee, Ying Wang, Susan P. Grill, Kuo Hsiung Lee
المصدر: Scientific Reports, Vol 7, Iss 1, Pp 1-11 (2017)
Scientific Reportsمصطلحات موضوعية: 0301 basic medicine, animal structures, Hepatitis C virus, Allosteric regulation, lcsh:Medicine, Arthritis, Inflammation, Hepacivirus, macromolecular substances, Plasma protein binding, Biology, Virus Replication, medicine.disease_cause, Article, 03 medical and health sciences, Alkaloids, 0302 clinical medicine, Allosteric Regulation, In vivo, ATP hydrolysis, medicine, Humans, Nucleotide Motifs, lcsh:Science, Multidisciplinary, lcsh:R, HSC70 Heat-Shock Proteins, Indolizines, virus diseases, RNA, Phenanthrenes, medicine.disease, Molecular biology, digestive system diseases, 3. Good health, 030104 developmental biology, 030220 oncology & carcinogenesis, embryonic structures, RNA, Viral, lcsh:Q, medicine.symptom, Allosteric Site, Protein Binding
-
2
المصدر: Bioorganic & Medicinal Chemistry Letters. 22:3358-3361
مصطلحات موضوعية: Anti-HIV Agents, Clinical Biochemistry, Human immunodeficiency virus (HIV), Surface binding, Pharmaceutical Science, Plasma protein binding, HIV Envelope Protein gp120, Virus Replication, medicine.disease_cause, Binding, Competitive, Biochemistry, Article, Viral entry, Drug Discovery, medicine, Humans, Potency, Molecular Biology, Blocking (linguistics), biology, Chemistry, Organic Chemistry, virus diseases, Virus Internalization, Virology, Cell biology, Viral replication, HIV-1, biology.protein, Molecular Medicine, Antibody, Protein Binding
-
3
المؤلفون: Kazuhiro Haraguchi, Masanori Baba, Yung-Chi Cheng, Jan Balzarini, Hiromichi Tanaka, Hiroshi Abe, Keiogo Kimura, Elizabeth A. Gullen, Takayuki Hamasaki, Ginger E. Dutschman, Genta Akutsu, Hisashi Shimada
المصدر: ACS Medicinal Chemistry Letters
مصطلحات موضوعية: chemistry.chemical_classification, Glycal, Chemistry, Stereochemistry, Organic Chemistry, glycal, electrophilic glycosidation, anti-hiv-1 activity, Biochemistry, Combinatorial chemistry, stereoselective-synthesis, Nucleoside Reverse Transcriptase Inhibitor, Nucleobase, nucleoside reverse transcriptase inhibitors, chemistry.chemical_compound, Drug Discovery, Electrophile, analogs, lipids (amino acids, peptides, and proteins), 4 '-thionucleosides, Glycosyl donor, Selectivity, Cytosine, nucleosides
وصف الملف: Print
-
4
المؤلفون: Wei, Zhang, Ginger E, Dutschman, Xin, Li, Yung-Chi, Cheng
المصدر: Journal of Chromatography B. 879:2018-2022
مصطلحات موضوعية: Analysis of Variance, Spectrometry, Mass, Electrospray Ionization, Paclitaxel, Chemical Hazard Release, Clinical Biochemistry, Reproducibility of Results, Cell Biology, General Medicine, Sensitivity and Specificity, Biochemistry, Analytical Chemistry, Drug Stability, Tandem Mass Spectrometry, Linear Models, Humans, Taxoids, Chromatography, Liquid
-
5
المؤلفون: Tatyana Kharlamova, Angela Corona, Francesca Esposito, Giovanni Floris, Simona Distinto, Luca Zinzula, Yung-Chi Cheng, Ginger E. Dutschman, Enzo Tramontano, Patrick Markt
المصدر: FEBS Journal. 278:1444-1457
مصطلحات موضوعية: biology, DNA polymerase, Active site, Cell Biology, Biochemistry, Molecular biology, Reverse transcriptase, chemistry.chemical_compound, chemistry, Docking (molecular), biology.protein, Binding site, RNase H, Molecular Biology, DNA, Polymerase
-
6
المؤلفون: Rong Ju, John Hines, Yung-Chi Cheng, Craig M. Crews, Ginger E. Dutschman
المصدر: Journal of Pharmacology and Experimental Therapeutics. 334:729-738
مصطلحات موضوعية: Cellular and Molecular, Guanine, GTP', Blotting, Western, Fluorescent Antibody Technique, Guanosine, Biology, Mice, chemistry.chemical_compound, Adenosine Triphosphate, Cyclohexanes, medicine, Animals, Nucleotide, p21-activated kinases, Inosine, Chromatography, High Pressure Liquid, Cell Proliferation, Pharmacology, chemistry.chemical_classification, O-(Chloroacetylcarbamoyl)fumagillol, Antibiotics, Antineoplastic, Cell Cycle, Endothelial Cells, Mycophenolic Acid, Flow Cytometry, Molecular biology, Guanine Nucleotides, Endothelial stem cell, p21-Activated Kinases, chemistry, Enzyme Induction, Molecular Medicine, Cattle, Tumor Suppressor Protein p53, Sesquiterpenes, Thymidine, Guanine salvage, medicine.drug
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::8cc974d335502ea777ed6f37655da042
https://doi.org/10.1124/jpet.110.169110 -
7
المؤلفون: Guangwei Yang, Elijah Paintsil, Chuan-Jen Wang, Ginger E. Dutschman, Yung-Chi Cheng, Jimin Wang, Hiromichi Tanaka, Susan P. Grill, Masanori Baba, Takayuki Hamasaki
المصدر: Antimicrobial Agents and Chemotherapy. 53:4640-4646
مصطلحات موضوعية: Anti-HIV Agents, viruses, Mutant, Microbial Sensitivity Tests, Drug resistance, Biology, medicine.disease_cause, Antiviral Agents, Virus, immune system diseases, Drug Resistance, Viral, medicine, Humans, Computer Simulation, Pharmacology (medical), Gene, Pharmacology, Mutation, virus diseases, biochemical phenomena, metabolism, and nutrition, Nucleotidyltransferase, Resistance mutation, Virology, Molecular biology, HIV Reverse Transcriptase, Reverse transcriptase, Stavudine, Infectious Diseases, HIV-1, Reverse Transcriptase Inhibitors
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::3f94f1a8a538083065688b29c7df884a
https://doi.org/10.1128/aac.00686-09 -
8
المؤلفون: Hiromichi Tanaka, Yung-Chi Cheng, Masanori Baba, Ginger E. Dutschman, Elijah Paintsil, Rong Hu, Wing Lam, Susan P. Grill
المصدر: Antimicrobial Agents and Chemotherapy. 51:3870-3879
مصطلحات موضوعية: Anti-HIV Agents, Metabolite, Biology, Virus Replication, Antiviral Agents, Thymidylate kinase, Cell Line, Zidovudine, chemistry.chemical_compound, medicine, Humans, Thymine Nucleotides, Pharmacology (medical), Phosphorylation, Pharmacology, Dose-Response Relationship, Drug, Kinase, Stavudine, HIV, virus diseases, Biological activity, Virology, Infectious Diseases, chemistry, Cell culture, Reverse Transcriptase Inhibitors, Thymidine, Dideoxynucleotides, HeLa Cells, medicine.drug
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::3f57a7a9953733a45ae598f8a275ddc9
https://doi.org/10.1128/aac.00692-07 -
9
المؤلفون: Ginger E. Dutschman, Rong Hu, Yung-Chi Cheng, Hiromichi Tanaka, Masanori Baba, Guangwei Yang, Preethi Krishnan, Chih-Hung Hsu
المصدر: Antimicrobial Agents and Chemotherapy. 51:1687-1693
مصطلحات موضوعية: Anti-HIV Agents, Biology, Antiviral Agents, Structure-Activity Relationship, chemistry.chemical_compound, Zidovudine, parasitic diseases, medicine, Humans, Pharmacology (medical), Phosphorylation, Thymidine kinase 1, Pharmacology, Nucleoside-phosphate kinase, Kinase, Molecular biology, Nucleoside-diphosphate kinase, Stavudine, Infectious Diseases, Biochemistry, chemistry, Nucleoside-Phosphate Kinase, Thymidine, Pyruvate kinase, medicine.drug
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::ff7cdfc1eff495507d58249324924aef
https://doi.org/10.1128/aac.01432-06 -
10
المؤلفون: Lei Fu, Yashang Lee, Ju-Liang Zhu, Eng-Shang Huang, Ginger E. Dutschman, Hosup Yeo, Elizabeth A. Gullen, Ying Li, Yung-Chi Cheng, Raymond T. Chung, David J. Austin
المصدر: Journal of Medicinal Chemistry. 48:534-546
مصطلحات موضوعية: Hepatitis B virus, Herpesvirus 4, Human, Stereochemistry, Herpesvirus 2, Human, Hepatitis C virus, Cytomegalovirus, Dioxoles, Hepacivirus, Herpesvirus 1, Human, Naphthalenes, Hydrazide, medicine.disease_cause, Antiviral Agents, Lignans, Virus, Methylenedioxy, Lactones, Structure-Activity Relationship, chemistry.chemical_compound, Drug Discovery, medicine, Structure–activity relationship, Benzofurans, chemistry.chemical_classification, HIV, Herpes simplex virus, chemistry, Lactam, Molecular Medicine, Lactone