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1دورية أكاديمية
المؤلفون: Talakad G. Lohith, Charalambos Kaittanis, Anthony P. Belanger, Shin Hye Ahn, Phil Sandoval, Lawrence Cohen, Girija Rajarshi, Wanida Ruangsiriluk, Rizwana Islam, Christopher T. Winkelmann, Paul McQuade
المصدر: Molecules, Vol 28, Iss 20, p 7144 (2023)
مصطلحات موضوعية: Fabry disease, alpha-galactosidase A, positron emission tomography, fluorine-18, radiolabeling, AGAL, Organic chemistry, QD241-441
وصف الملف: electronic resource
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2
المؤلفون: Shakiru O. Alapafuja, Jodi Anne T. Wood, Dimitrios N. Pelekoudas, Christina Miyabe Shields, Alexandros Makriyannis, Girija Rajarshi, Nicholas Thomas Perry, Spiro Pavlopoulos, Honrao Chandrashekhar, Michael S. Malamas, Khadijah A. Mohammad, Alexander Zvonok, Jay A. A. West, Shrouq I. Farah
المصدر: Journal of Medicinal Chemistry. 64:5956-5972
مصطلحات موضوعية: 0303 health sciences, Palmitoylethanolamide, 01 natural sciences, 0104 chemical sciences, Amidase, Serine, 010404 medicinal & biomolecular chemistry, 03 medical and health sciences, chemistry.chemical_compound, Biochemistry, chemistry, N-Acylethanolamine, Drug Discovery, Isothiocyanate, Molecular Medicine, Structure–activity relationship, Pharmacophore, 030304 developmental biology, Cysteine
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3
المؤلفون: Michael S, Malamas, Spiro, Pavlopoulos, Shakiru O, Alapafuja, Shrouq I, Farah, Alexander, Zvonok, Khadijah A, Mohammad, Jay, West, Nicholas Thomas, Perry, Dimitrios N, Pelekoudas, Girija, Rajarshi, Christina, Shields, Honrao, Chandrashekhar, Jodi, Wood, Alexandros, Makriyannis
المصدر: Journal of medicinal chemistry. 64(9)
مصطلحات موضوعية: Structure-Activity Relationship, Drug Stability, Isothiocyanates, Drug Design, Hydrolysis, Humans, Enzyme Inhibitors, Amidohydrolases
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4
المؤلفون: David R. Janero, Spiro Pavlopoulos, Alexandros Makriyannis, Nikolai Zvonok, Sergiy Tyukhtenko, Girija Rajarshi, Ioannis Karageorgos
المصدر: Journal of Biological Chemistry. 291:2556-2565
مصطلحات موضوعية: 0301 basic medicine, chemistry.chemical_classification, Serine protease, Conformational change, 030102 biochemistry & molecular biology, biology, Active site, Serine hydrolase, Cell Biology, Biochemistry, Monoacylglycerol lipase, 03 medical and health sciences, 030104 developmental biology, Enzyme, chemistry, biology.protein, Structure–activity relationship, Lipase, Molecular Biology
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_________::3c046094bf6cb7222edd15f6a105e830
https://doi.org/10.1074/jbc.m115.670257 -
5
المؤلفون: Christina Yume Miyabe, Jay A. A. West, Michael S. Malamas, Girija Rajarshi, Dimitrios N. Pelekoudas, Nicholas Thomas Perry, Honrao Chandrashekhar, Manjunath Lamani, Spiro Pavlopoulos, Alexandros Makriyannis, Shrouq I. Farah
المصدر: Bioorganic & Medicinal Chemistry. 28:115195
مصطلحات موضوعية: Models, Molecular, Cannabinoid receptor, Clinical Biochemistry, Pharmaceutical Science, 01 natural sciences, Biochemistry, Amidohydrolases, Amidase, Mice, Structure-Activity Relationship, chemistry.chemical_compound, Oleoylethanolamide, Drug Discovery, Animals, Enzyme Inhibitors, Molecular Biology, Palmitoylethanolamide, Dose-Response Relationship, Drug, Molecular Structure, 010405 organic chemistry, Organic Chemistry, ABHD6, Cysteine protease, Rats, 0104 chemical sciences, 010404 medicinal & biomolecular chemistry, chemistry, Cyanamide, Drug Design, Molecular Medicine, Pharmacophore, Endogenous agonist
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6
المؤلفون: Alex Straiker, Girija Rajarshi, Christina Yume Miyabe, Shakiru O. Alapafuja, Sally Miller, Vidyanand G. Shukla, Michael S. Malamas, Alexandros Makriyannis, JodiAnne T. Wood, Laura Daily, Honrao Chandrashekhar, Alexander Zvonok, Sergiy Tyukhtenko
المصدر: Bioorg Med Chem
مصطلحات موضوعية: Male, Cannabinoid receptor, genetic structures, Clinical Biochemistry, Pharmaceutical Science, Glaucoma, Pharmacology, 01 natural sciences, Biochemistry, Piperazines, Article, law.invention, Serine, Structure-Activity Relationship, Piperidines, law, Catalytic Domain, Drug Discovery, medicine, Animals, Humans, Enzyme Inhibitors, Receptor, Molecular Biology, Molecular Structure, 010405 organic chemistry, Chemistry, Organic Chemistry, Ligand (biochemistry), ABHD6, medicine.disease, eye diseases, Monoacylglycerol Lipases, 0104 chemical sciences, Rats, Monoacylglycerol lipase, Mice, Inbred C57BL, Molecular Docking Simulation, 010404 medicinal & biomolecular chemistry, Recombinant DNA, Microsomes, Liver, Molecular Medicine, Carbamates
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7
المؤلفون: Mahmoud L. Nasr, Nikolai Zvonok, Xiaoyu Ma, Kiran Vemuri, Hongwei Huang, Spiro Pavlopoulos, Sergiy Tyukhtenko, Jeffrey W. Hudgens, Elyssia S. Gallagher, Alexandros Makriyannis, Ioannis Karageorgos, Girija Rajarshi
المصدر: Scientific Reports
Scientific Reports, Vol 8, Iss 1, Pp 1-17 (2018)مصطلحات موضوعية: 0301 basic medicine, Models, Molecular, Protein Conformation, Allosteric regulation, DNA Mutational Analysis, Mutation, Missense, lcsh:Medicine, medicine.disease_cause, Article, 03 medical and health sciences, Protein structure, Allosteric Regulation, Catalytic triad, medicine, Humans, Lipase, lcsh:Science, Mutation, Multidisciplinary, biology, Chemistry, lcsh:R, Active site, Monoacylglycerol Lipases, Monoacylglycerol lipase, 030104 developmental biology, Amino Acid Substitution, biology.protein, Biophysics, lcsh:Q, Mutant Proteins, Function (biology)
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8
المؤلفون: Roger S. Gifford, Alexandros Makriyannis, Jack Bergman, Girija Rajarshi, Dow P. Hurst, Ganesh A. Thakur, Jimit Girish Raghav, Shashank Kulkarni, Jason J. Guo, Carol A. Paronis, Patricia H. Reggio, Spyros P. Nikas, Rishi Sharma, JodiAnne T. Wood, Torbjörn U. C. Järbe, Yingpeng Liu
المصدر: Journal of Medicinal Chemistry
مصطلحات موضوعية: Stereochemistry, Metabolite, Druggability, In vitro, Article, chemistry.chemical_compound, Structure-Activity Relationship, HEK293 Cells, chemistry, Receptor, Cannabinoid, CB1, In vivo, Drug Design, Drug Discovery, Side chain, Molecular Medicine, Structure–activity relationship, Potency, Humans, Dronabinol, Receptor
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9
المؤلفون: Alexandros Makriyannis, Jordan Ward, Greig Turvey, Shakiru O. Alapafuja, Othman Benchama, Cheryl L. Limebeer, Linda A. Parker, Martin A. Sticht, Erin M. Rock, JodiAnne T. Wood, Girija Rajarshi
المصدر: Psychopharmacology. 233(12)
مصطلحات موضوعية: 0301 basic medicine, Male, Nausea, Pharmacology, Article, Amidohydrolases, Rats, Sprague-Dawley, 03 medical and health sciences, chemistry.chemical_compound, 0302 clinical medicine, In vivo, Fatty acid amide hydrolase, medicine, Animals, Enzyme Inhibitors, IC50, Cerebral Cortex, Anandamide, Endocannabinoid system, In vitro, Monoacylglycerol Lipases, 3. Good health, Rats, Monoacylglycerol lipase, Disease Models, Animal, 030104 developmental biology, nervous system, chemistry, Acute Disease, lipids (amino acids, peptides, and proteins), Vomiting, Anticipatory, medicine.symptom, psychological phenomena and processes, 030217 neurology & neurosurgery, Endocannabinoids
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المؤلفون: Sergiy, Tyukhtenko, Ioannis, Karageorgos, Girija, Rajarshi, Nikolai, Zvonok, Spiro, Pavlopoulos, David R, Janero, Alexandros, Makriyannis
المصدر: The Journal of biological chemistry. 291(6)
مصطلحات موضوعية: Kinetics, Structure-Activity Relationship, Humans, Hydrogen-Ion Concentration, Nuclear Magnetic Resonance, Biomolecular, Monoacylglycerol Lipases, Molecular Biophysics, Protein Structure, Tertiary
URL الوصول: https://explore.openaire.eu/search/publication?articleId=pmid________::9dd139b47b37a500b119d73f209352c6
https://pubmed.ncbi.nlm.nih.gov/26555264