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1
المؤلفون: Jia Lei, Joon Jung, Sylvie G. Bernier, Joel D. Moore, Glen Rennie, Mermerian Ara, Nicholas Robert Perl, Thomas Wai-Ho Lee, Andrew Carvalho, Barden Timothy Claude, Peter Germano, Jenny Tobin, Colleen Hudson, Renee Deming, Rajesh R. Iyengar, Takashi Nakai, G-Yoon Jamie Im, Paul A. Renhowe, Daniel P. Zimmer, Elise Kim
المصدر: Bioorganicmedicinal chemistry letters. 40
مصطلحات موضوعية: Male, Models, Molecular, Carboxylic acid, Hypertension, Pulmonary, Vasodilator Agents, Clinical Biochemistry, Carboxylic Acids, Drug Evaluation, Preclinical, Pharmaceutical Science, Administration, Oral, Pharmacology, Nitric Oxide, Biochemistry, Nitric oxide, Rats, Sprague-Dawley, chemistry.chemical_compound, Structure-Activity Relationship, Glucuronides, Soluble Guanylyl Cyclase, Drug Discovery, medicine, Animals, Humans, Molecular Biology, chemistry.chemical_classification, Dose-Response Relationship, Drug, Organic Chemistry, Soluble Guanylate Cyclase Stimulator, medicine.disease, Pulmonary hypertension, Bioavailability, Oxidative Stress, chemistry, Metabolome, Molecular Medicine, Signal transduction, Metabolic profile, Guanylate cyclase, Protein Binding, Signal Transduction
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2
المؤلفون: Theresa L. Johnson, Steven Kazmirski, Simon Low, Cyrille Kuhn, Robert V. Stanton, Yuan-Hua Ding, Gayatri D. Deshmukh, Jessie M. English, Haile Tecle, Glen Rennie, Ping Ye, Hu Liu, Joseph Wu, Alan C. Cheng, Suzanne L. Jacques, Rocco Coli, Frederic Feru
المصدر: Bioorganic & Medicinal Chemistry Letters. 20:4885-4891
مصطلحات موضوعية: medicine.drug_class, Stereochemistry, Amino Acid Motifs, Clinical Biochemistry, Pharmaceutical Science, Carboxamide, Pyrazole, Biochemistry, Chemical synthesis, Mitogen-Activated Protein Kinase 14, Structure-Activity Relationship, chemistry.chemical_compound, Microsomes, Drug Discovery, medicine, Humans, Structure–activity relationship, Amino Acid Sequence, Binding site, Protein Kinase Inhibitors, Molecular Biology, Binding Sites, Adenine binding, biology, Chemistry, Adenine, Phenylurea Compounds, Organic Chemistry, Enzyme inhibitor, biology.protein, Pyrazoles, Molecular Medicine, Selectivity
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3
المؤلفون: Darcy Kohls, Simon Low, Glen Rennie, Yuan-Hua Ding, Cyrille Kuhn, Frederic Feru, Michael Kothe, Rocco Coli
المصدر: Chemical Biology & Drug Design. 70:540-546
مصطلحات موضوعية: Pharmacology, Gene isoform, Kinase, Chemistry, Organic Chemistry, Regulator, Polo-like kinase, medicine.disease_cause, Biochemistry, PLK1, enzymes and coenzymes (carbohydrates), Drug Discovery, medicine, Molecular Medicine, Transferase, biological phenomena, cell phenomena, and immunity, Carcinogenesis, Selectivity
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4
المؤلفون: Karen Stapleton, Messersmith David, Paul Hawkins, Jimmy Dumornay, Mark L. Nelson, Peter Viski, Beena Bhatia, Glen Rennie, David Andorsky, Paul Sheahan, and Tadeusz Warchol, Mohamed Y. Ismail, Stuart B. Levy, Laura Mcintyre, Atul K. Verma
المصدر: The Journal of Organic Chemistry. 68:5838-5851
مصطلحات موضوعية: chemistry.chemical_classification, Doxycycline, Methacycline, Magnetic Resonance Spectroscopy, Ketone, Diazonium Compounds, Tetracycline, Organic Chemistry, Molecular Conformation, Minocycline, Chemical synthesis, Catalysis, chemistry, Tetracyclines, medicine, Organic chemistry, Indicators and Reagents, Amine gas treating, Palladium, medicine.drug
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5
المؤلفون: Cyrille Kuhn, James R. Kiefer, Christine M. Kornmeier, Joseph B. Moon, John I. Trujillo, Wei Huang, Christine P. Bono, Melanie L. Williams, Gina M. Jerome, Christopher P. Carron, Atli Thorarensen, Jacqueline E. Day, Glen Rennie, Thomas A. Wynn
المصدر: Bioorganicmedicinal chemistry letters. 22(11)
مصطلحات موضوعية: Clinical Biochemistry, Binding pocket, Anti-Inflammatory Agents, Pharmaceutical Science, Prostaglandin, Naphthalenes, Crystallography, X-Ray, Biochemistry, chemistry.chemical_compound, Protein structure, Drug Discovery, Anti-Allergic Agents, Humans, Computer Simulation, Binding site, Enzyme Inhibitors, Molecular Biology, chemistry.chemical_classification, Binding Sites, ATP synthase, biology, Organic Chemistry, Prostaglandin D2 synthase, Water, Isoquinolines, Lipocalins, Protein Structure, Tertiary, Intramolecular Oxidoreductases, Haematopoiesis, Enzyme, chemistry, biology.protein, Molecular Medicine