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1
المؤلفون: Graeme Irvine Stevenson, Juliette E Neve, Vicky M. Avery, Sarah Yong, Aaron Lock, Gregory Allen Fechner
المصدر: Bioorganicmedicinal chemistry letters. 28(14)
مصطلحات موضوعية: Stereochemistry, Organic Chemistry, Clinical Biochemistry, Pharmaceutical Science, Substrate (chemistry), Ring (chemistry), Biochemistry, chemistry.chemical_compound, Solid-phase synthesis, Biotin, chemistry, Drug Discovery, Isoprenylcysteine carboxylmethyltransferase, Molecular Medicine, Molecular Biology, Cysteine
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2
المؤلفون: Paul W. Smith, Ian Thomson Forbes, Andrea M. Bradford, Graham Walker, Graham Murkitt, Wyman Paul Adrian, Graeme Irvine Stevenson, Dale James Johnson, Jeannette M. Watson, Steve P. Watson, Adam J. Lucas, Claudette Mookherjee, Fiona Brown, Vincenzo Garzya, Sean Thomas Flynn, Jane Gartlon, Harminder Mudhar
المصدر: Bioorganic & Medicinal Chemistry Letters. 20:5434-5438
مصطلحات موضوعية: Agonist, Indoles, medicine.drug_class, Stereochemistry, education, Clinical Biochemistry, Allosteric regulation, Pharmaceutical Science, Muscarinic Agonists, Biochemistry, Chemical synthesis, chemistry.chemical_compound, Drug Discovery, Muscarinic acetylcholine receptor, medicine, Animals, Molecular Biology, Nootropic Agents, Benzoxazoles, Memory Disorders, Bicyclic molecule, Receptor, Muscarinic M1, Organic Chemistry, Brain, Oxindoles, Rats, chemistry, Lipophilicity, Lactam, Molecular Medicine, Penetrant (biochemical)
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3
المؤلفون: Victoria J. Barrett, Feng Wang, Christopher Browning, Matthew J Lindon, Henry M. Sarau, James A. Fornwald, Andy J. Harker, Guido Hartmann, Jeffery K. Kerns, David P. Andrew, Graeme Irvine Stevenson, Ashley Paul Hancock, Victoria Vinader, Michael L. Moore, James J. Foley, Jian Jin, Parvathi Rao, Anthony J. Jurewicz, Helen E. Connor, Dwight M. Morrow, Kristen E. Belmonte, Yonghui Wang, Ralph A. Rivero, Cuc Nguyen
المصدر: Bioorganic & Medicinal Chemistry Letters. 17:1722-1725
مصطلحات موضوعية: ERG1 Potassium Channel, Stereochemistry, High-throughput screening, Clinical Biochemistry, Drug Evaluation, Preclinical, Human immunodeficiency virus (HIV), Pharmaceutical Science, CHO Cells, Computational biology, Protein Serine-Threonine Kinases, medicine.disease_cause, Biochemistry, Chemical synthesis, Myotonin-Protein Kinase, Receptors, CCR8, Structure-Activity Relationship, Cricetulus, Th2 Cells, Cricetinae, Drug Discovery, medicine, Animals, Humans, Structure–activity relationship, Computer Simulation, Molecular Biology, Oxazolidinones, Chemistry, Organic Chemistry, Ether-A-Go-Go Potassium Channels, Chemotaxis, Leukocyte, Lung disease, Molecular Medicine, Indicators and Reagents, Receptors, Chemokine
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4
المصدر: Bioorganic & Medicinal Chemistry Letters. 10:2693-2696
مصطلحات موضوعية: Carbamate, Indoles, Stereochemistry, medicine.medical_treatment, Clinical Biochemistry, Pharmaceutical Science, Binding, Competitive, Biochemistry, Chemical synthesis, Solid-phase synthesis, Drug Discovery, medicine, Combinatorial Chemistry Techniques, Humans, Molecular Biology, Indole test, Bicyclic molecule, Receptors, Dopamine D2, Chemistry, Organic Chemistry, Antagonist, Biological activity, Tryptamines, Receptors, Serotonin, Molecular Medicine, Serotonin Antagonists, Linker
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5
المصدر: Tetrahedron Letters. 39:8317-8320
مصطلحات موضوعية: Annulation, Solid-phase synthesis, Stereochemistry, Chemistry, Organic Chemistry, Drug Discovery, Biochemistry, Linker, Combinatorial chemistry
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6
المؤلفون: Myra B. Kurtz, Gary G. Chicchi, Sharon Sadowski, Graeme Irvine Stevenson, Margaret A. Cascieri, Angus Murray Macleod, Jason Matthew Elliott, Ian Thomas Huscroft, Howard B. Broughton
المصدر: Bioorganic & Medicinal Chemistry Letters. 8:1851-1856
مصطلحات موضوعية: chemistry.chemical_classification, Sulfonamides, Chemistry, Stereochemistry, Aryl, Organic Chemistry, Clinical Biochemistry, Pharmaceutical Science, Receptors, Neurokinin-1, Biochemistry, Sulfonamide, Serine, Structure-Activity Relationship, chemistry.chemical_compound, Models, Chemical, Neurokinin-1 Receptor Antagonists, Piperidines, Drug Discovery, Molecular Medicine, Pharmacophore, Molecular Biology
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7
المؤلفون: Aaron Lock, Juliette E Neve, Gregory Allen Fechner, Sarah Yong, Graeme Irvine Stevenson, Vicky M. Avery
المصدر: Bioorganicmedicinal chemistry letters. 23(20)
مصطلحات موضوعية: High-throughput screening, Clinical Biochemistry, Pharmaceutical Science, Biotin, Biochemistry, Substrate Specificity, chemistry.chemical_compound, Solid-phase synthesis, Drug Discovery, Isoprenylcysteine carboxylmethyltransferase, Organic chemistry, Cysteine, Protein Methyltransferases, Molecular Biology, Solid-Phase Synthesis Techniques, Organic Chemistry, Substrate (chemistry), Trityl Compounds, Combinatorial chemistry, High-Throughput Screening Assays, Kinetics, Scintillation proximity assay, chemistry, Molecular Medicine
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8
المؤلفون: M A Casiceri, Fintan Kelleher, Andrew Pate Owens, F Brookfield, Christopher J. Swain, Angus Murray Macleod, Graeme Irvine Stevenson, E. Ber, Kevin John Merchant, Sharon Sadowski
المصدر: Journal of Medicinal Chemistry. 37:1269-1274
مصطلحات موضوعية: Male, Models, Molecular, Stereochemistry, Acylation, Guinea Pigs, Molecular Sequence Data, Molecular Conformation, CHO Cells, Substance P, Dermatitis, Contact, Substance-P Receptor, Structure-Activity Relationship, Neurokinin-1 Receptor Antagonists, Cricetinae, Drug Discovery, Animals, Humans, Structure–activity relationship, Computer Simulation, Amino Acid Sequence, Indole test, Molecular Structure, Chemistry, Tryptophan, Antagonist, Biological activity, Receptors, Neurokinin-1, Recombinant Proteins, Molecular Medicine, Sample collection
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::7720024e0e72b49653cd4233e3c73152
https://doi.org/10.1021/jm00035a006 -
9
المؤلفون: I. Sanderson, George R. Marshall, Ian Stansfield, R. Baker, John A. Kemp, Graeme Irvine Stevenson, L. Robinson, Paul D. Leeson, A M Moseley, Michael Rowley
المصدر: Journal of Medicinal Chemistry. 36:3386-3396
مصطلحات موضوعية: Receptor complex, Ketone, Lactams, Stereochemistry, Acylation, Carboxylic acid, Glycine, Receptors, N-Methyl-D-Aspartate, Structure-Activity Relationship, Drug Discovery, Animals, Binding site, Cerebral Cortex, chemistry.chemical_classification, Binding Sites, Rats, Inbred Strains, Biological activity, Ketones, Rats, Kinetics, chemistry, Hydroxyquinolines, Molecular Medicine, NMDA receptor, Anticonvulsants, Pharmacophore
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::39a295f38f0e3b0034c1f7bb82fcf2e9
https://doi.org/10.1021/jm00074a020 -
10
المؤلفون: Robert W. Carling, Ian M. Mawer, Mark Peter Ridgill, John A. Kemp, Graeme Irvine Stevenson, Raymond Baker, Alan C. Foster, Michael Rowley, Paul D. Leeson, Janusz Jozef Kulagowski, Ian Stansfield, Julian D. Smith
المصدر: Bioorganic & Medicinal Chemistry Letters. 3:299-304
مصطلحات موضوعية: chemistry.chemical_classification, Stereochemistry, Organic Chemistry, Clinical Biochemistry, Pharmaceutical Science, N-methyl-D-aspartate Receptor Antagonists, Biochemistry, Amino acid, chemistry.chemical_compound, 2-quinolone, chemistry, Drug Discovery, Glycine, Lactam, Molecular Medicine, Bioisostere, Receptor, Molecular Biology