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المؤلفون: Richard M. Angell, John Ludes-Meyers, Simon E. Ward, Michael Paradowski, Irina Chuckowree, Alexandre Bedernjak, James Lumley, Carol Villalonga Barber, Kenneth Powell, Edward Littler, Daniel Watterson, Geraldine Taylor, Elaine Thomas, Jose Gascon-Simorte, Mark E. Peeples, Michelle Thom, Jason S. McLellan, Dereck Tait, Neil Mathews, Paul R. Young, Ian M. Fraser, Morgan S.A. Gilman, James A. D. Good, G. Stuart Cockerill, Rachel Harland, Sara M. Johnson, Graham Lunn, Claire Scott, Gareth Williams
مصطلحات موضوعية: Biological Availability, Microbial Sensitivity Tests, Placebo, Antiviral Agents, 01 natural sciences, Virus, 03 medical and health sciences, Cell Line, Tumor, Drug Discovery, Animals, Humans, Respiratory system, IC50, 030304 developmental biology, Clinical Trials as Topic, 0303 health sciences, Drug discovery, Chemistry, Virus Internalization, Virology, 3. Good health, 0104 chemical sciences, Bioavailability, 010404 medicinal & biomolecular chemistry, Cell culture, Respiratory Syncytial Virus, Human, Molecular Medicine, Benzimidazoles, Viral Fusion Proteins, Viral load, Protein Binding
وصف الملف: application/pdf
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2
المؤلفون: Andrews Mark David, Robert M. Owen, Mathilde Grenie, Kevin Beaumont, David C. Pryde, Sebastien Galan, Dannielle Frances Roberts, Tram T. Tran, Paul Alan Glossop, Amy S. Kenyon, Graham Lunn, Alan S. Jessiman, Maw Graham Nigel, Kerry af Forselles
المصدر: ACS Medicinal Chemistry Letters. 6:419-424
مصطلحات موضوعية: Chemistry, Organic Chemistry, Antagonist, Hypothermia, Thermoregulation, Pharmacology, Biochemistry, Transient receptor potential channel, Allodynia, Drug Discovery, Hyperalgesia, medicine, TRPM8, medicine.symptom, Ion channel
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3
المؤلفون: Graham Lunn, David Winpenny, M. J. Gardner, M. Abid Masood, Dack Kevin Neil
المصدر: Bioorganic & Medicinal Chemistry Letters. 22:3682-3687
مصطلحات موضوعية: Chemistry, Stereochemistry, Receptors, Prostaglandin, Organic Chemistry, Clinical Biochemistry, Carboxylic Acids, Pharmaceutical Science, Ligands, Biochemistry, Combinatorial chemistry, Chemical space, Small Molecule Libraries, Th2 Cells, Drug Discovery, Humans, Molecular Medicine, Receptors, Immunologic, Molecular Biology, Protein Binding
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المؤلفون: Graham Lunn, Lee R. Roberts, Stephane Content, Douglas J. Critcher, Sara Douglas, Ashley E. Fenwick, David M. Gethin, Graham Goodwin, David Greenway, Sean Greenwood, Kim Hall, Martin Thomas, Stephen Thompson, David Williams, Gavin Wood, Andrew Wylie
المصدر: Bioorganic & Medicinal Chemistry Letters. 22:2200-2203
مصطلحات موضوعية: μ receptor, Stereochemistry, medicine.drug_class, Guinea Pigs, Clinical Biochemistry, Receptors, Opioid, mu, Pharmaceutical Science, In Vitro Techniques, Ligands, Biochemistry, Structure-Activity Relationship, chemistry.chemical_compound, Dogs, Opioid receptor, Receptors, Opioid, delta, Drug Discovery, medicine, Animals, Hexanes, Humans, skin and connective tissue diseases, Molecular Biology, Biological evaluation, Chemistry, Pruritus, Receptors, Opioid, kappa, Organic Chemistry, Antipruritics, Bridged Bicyclo Compounds, Heterocyclic, Ligand (biochemistry), Hexane, Kinetics, Opioid, Lead structure, Molecular Medicine, Functional activity, medicine.drug
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المؤلفون: Michael Yeadon, Tanya Hay, Wai L. S. Liu, Charles E. Mowbray, Valerie M. Joynson, Graham Lunn
المصدر: Med. Chem. Commun.. 3:339-343
مصطلحات موضوعية: Pharmacology, integumentary system, Chemistry, Drug Discovery, Organic Chemistry, Antagonist, Low permeability, Pharmaceutical Science, Molecular Medicine, Histamine H3 receptor, Biochemistry, Efflux transporters
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_________::686aec730e5fd6b030bae89265f437a6
https://doi.org/10.1039/c2md00276k -
6
المؤلفون: Yogesh A. Sabnis, Alan John Pettman, Bernard Joseph Banks, Neil Feeder, Robert Crook, Graham Lunn
المصدر: Bioorganic & Medicinal Chemistry Letters. 21:4608-4611
مصطلحات موضوعية: Stereochemistry, medicine.drug_class, Clinical Biochemistry, Drug Evaluation, Preclinical, Receptors, Opioid, mu, Administration, Oral, Pharmaceutical Science, CHO Cells, Ligands, Biochemistry, chemistry.chemical_compound, Cricetulus, Dogs, In vivo, Opioid receptor, Cricetinae, Drug Discovery, medicine, Animals, Hexanes, Humans, Molecular Biology, Sulfonamides, Chemistry, Pruritus, Organic Chemistry, Antagonist, Rats, Hexane, Opioid, Molecular Medicine, Azabicyclo Compounds, Protein Binding, medicine.drug
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المؤلفون: Graham Lunn, Iain Kilty, David J. Lamb, Mark O Reilly, Cheryl Butler
المصدر: Journal of Pulmonary & Respiratory Medicine.
مصطلحات موضوعية: chemistry.chemical_classification, business.industry, Insulin, medicine.medical_treatment, Pharmacology, In vitro, Enzyme, Therapeutic index, chemistry, In vivo, Medicine, Binding site, business, Homeostasis, PI3K/AKT/mTOR pathway
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_________::60d51fa78a6fc686da4d79ce9e30a5f5
https://doi.org/10.4172/2161-105x.1000157 -
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المؤلفون: Yogesh A. Sabnis, Alan John Pettman, Neil Feeder, Bernard Joseph Banks, Robert Crook, Graham Lunn
المصدر: ChemInform. 42
مصطلحات موضوعية: Hexane, chemistry.chemical_compound, Opioid, Chemistry, Stereochemistry, medicine, General Medicine, medicine.drug
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المؤلفون: Paul Driscoll, Miller Duncan Charles, Nichola L. Davies, Peter Jones, Graham Lunn, Yogesh A. Sabnis
المصدر: MedChemComm. 3:449
مصطلحات موضوعية: Pharmacology, Stereochemistry, Chemistry, Biological target, Ligand, Computational chemistry, Drug Discovery, Organic Chemistry, Pharmaceutical Science, Molecular Medicine, Dissociation kinetics, Biochemistry, Receptor–ligand kinetics
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_________::77b0f03c9a0f9217ba086206d1295f70
https://doi.org/10.1039/c2md00270a -
10Optimized glucuronidation of dual pharmacology β-2 agonists/M3 antagonists for the treatment of COPD
المؤلفون: Rachel Osborne, David A. Entwistle, Michael Yeadon, Graham Lunn, Karen N. Wright, Jane L. Burrows, Emilio F. Stuart, Lyn H. Jones, Sandra D. Newman, Kim James, Amy S. Kenyon, Fiona J. Spence, Susan Summerhill, Matthew D. Selby, Nick Clarke, David Price, Stuart Marshall, Laura Hilton, Helen Baldock, Rhys M. Jones, Neil Feeder, Michael A. Trevethick, Sheena Patel, Nadia Laouar, Michele Coghlan, Mark E. Bunnage, David Fairman
المصدر: MedChemComm. 2:870
مصطلحات موضوعية: Pharmacology, COPD, Inhalation, Chemistry, Organic Chemistry, Glucuronidation, Pharmaceutical Science, medicine.disease, Biochemistry, Drug Discovery, medicine, Molecular Medicine, Potency
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_________::e8e88fd334de3783a85ab6566fddbc69
https://doi.org/10.1039/c1md00140j