-
1
المؤلفون: Laurence B. Peterson, Gregory J. Wiederrecht, William H. Parsons, John G. Cryan, Mark A. Holmes, Peter J. Sinclair, Mary-Jo Staruch, Matthew J. Wyvratt, Ray Rosa, Mary Beth Wilusz, Frederick Wong, Mark T. Goulet, Helen M. Armstrong, Francis J. Dumont, Samuel Koprak
المصدر: Bioorganic & Medicinal Chemistry Letters. 9:2089-2094
مصطلحات موضوعية: Male, Stereochemistry, T-Lymphocytes, Calcineurin Inhibitors, Clinical Biochemistry, Drug Evaluation, Preclinical, Administration, Oral, Pharmaceutical Science, Ether, Hypothermia, Alkylation, Biochemistry, Chemical synthesis, Tacrolimus, Rats, Sprague-Dawley, Tacrolimus Binding Proteins, Inhibitory Concentration 50, Mice, Structure-Activity Relationship, chemistry.chemical_compound, In vivo, Toxicity Tests, parasitic diseases, Drug Discovery, medicine, Animals, Ascomycin, Immunophilins, Molecular Biology, Mice, Inbred BALB C, Bicyclic molecule, Organic Chemistry, Combinatorial chemistry, Rats, chemistry, Injections, Intravenous, Toxicity, Molecular Medicine, Hemiacetal, Kidney Diseases, Macrolides, Immunosuppressive Agents, medicine.drug
-
2A TACROLIMUS-RELATED IMMUNOSUPPRESSANT WITH BIOCHEMICAL PROPERTIES DISTINCT FROM THOSE OF TACROLIMUS
المؤلفون: Mary M. Martin, Laurence B. Peterson, Gregory J. Wiederrecht, Janey N. Parsons, William H. Parsons, Peter J. Sinclair, Mary Beth Wilusz, Frederick Wong, John G. Cryan, Stephen J. O'Keefe, Matthew J. Wyvratt, Ray Rosa, Nolan H. Sigal, Alan R. Williamson
المصدر: Transplantation. 65:10-18
مصطلحات موضوعية: Macromolecular Substances, Recombinant Fusion Proteins, medicine.medical_treatment, Calcineurin Inhibitors, Molecular Sequence Data, chemical and pharmacologic phenomena, Pharmacology, Biology, Tacrolimus, Tacrolimus Binding Proteins, Jurkat Cells, Therapeutic index, medicine, Humans, Lymphocytes, Ascomycin, Promoter Regions, Genetic, Heat-Shock Proteins, Transplantation, Base Sequence, Immunosuppression, Oligonucleotides, Antisense, DNA-Binding Proteins, Calcineurin, surgical procedures, operative, FKBP, Immunosuppressive drug, Models, Chemical, Immunology, Toxicity, Interleukin-2, Carrier Proteins, Cell Division, Immunosuppressive Agents, medicine.drug
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::4d629f9f28c4924d99389136bd19b5cd
https://doi.org/10.1097/00007890-199801150-00004 -
3
المصدر: Biochemical and Biophysical Research Communications. 232:437-443
مصطلحات موضوعية: DNA, Complementary, Leukemia, T-Cell, T-Lymphocytes, T cell, Molecular Sequence Data, Biophysics, Thymus Gland, Biology, Biochemistry, Tacrolimus Binding Proteins, Phosphoprotein Phosphatases, Tumor Cells, Cultured, medicine, Humans, Distribution (pharmacology), Tissue Distribution, Amino Acid Sequence, Cloning, Molecular, Molecular Biology, Gene, Heat-Shock Proteins, Messenger RNA, Base Sequence, cDNA library, Calcineurin, Cell Biology, Molecular biology, In vitro, DNA-Binding Proteins, FKBP, medicine.anatomical_structure, Calmodulin-Binding Proteins, Carrier Proteins
-
4
المؤلفون: Gregory J. Wiederrecht, Gregory J. Brunn, John C. Lawrence, Robert T. Abraham, Candace J. Sabers, Josie M. Williams
المصدر: The EMBO Journal. 15:5256-5267
مصطلحات موضوعية: Phosphoinositide 3-kinase, General Immunology and Microbiology, General Neuroscience, RPTOR, Lipid kinase activity, Biology, mTORC2, General Biochemistry, Genetics and Molecular Biology, Cell biology, Wortmannin, chemistry.chemical_compound, chemistry, Biochemistry, biology.protein, TOR Serine-Threonine Kinases, LY294002, Molecular Biology, PI3K/AKT/mTOR pathway
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_________::a5635f26fb0081e81185d4b9c143d57b
https://doi.org/10.1002/j .1460-2075.1996.tb00911.x -
5
المؤلفون: Robert T. Abraham, Gregory J. Brunn, Gregory J. Wiederrecht, Josie M. Williams, Mary M. Martin, Francis J. Dumont, Candace J. Sabers
المصدر: Journal of Biological Chemistry. 270:815-822
مصطلحات موضوعية: DNA, Complementary, Saccharomyces cerevisiae Proteins, Molecular Sequence Data, Cell Cycle Proteins, Polyenes, Biology, Lymphoma, T-Cell, Biochemistry, mTORC2, Fungal Proteins, Rats, Sprague-Dawley, Tacrolimus Binding Proteins, Phosphatidylinositol 3-Kinases, Tumor Cells, Cultured, medicine, Animals, Humans, Amino Acid Sequence, Molecular Biology, MLST8, Heat-Shock Proteins, PI3K/AKT/mTOR pathway, DNA Primers, Sirolimus, Base Sequence, Sequence Homology, Amino Acid, Cell growth, TOR Serine-Threonine Kinases, RPTOR, Cell Biology, Rats, Cell biology, DNA-Binding Proteins, Phosphotransferases (Alcohol Group Acceptor), FKBP, Carrier Proteins, Protein Kinases, medicine.drug
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::a9540cf342215e63cd2761a93445d8c9
https://doi.org/10.1074/jbc.270.2.815 -
6
المؤلفون: L L Rokosz, J J Burbaum, Janey N. Parsons, Scott P. Salowe, Gregory J. Wiederrecht, Stephen J. O'Keefe, R L Kincaid
المصدر: Journal of Biological Chemistry. 269:19610-19616
مصطلحات موضوعية: Dephosphorylation, Calcineurin, FKBP, Biochemistry, Protein subunit, Binding protein, Phosphatase, Wild type, Cell Biology, Biology, Signal transduction, Molecular Biology
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_________::ea498aaa8cfdff1e2b5e2bf50f949cba
https://doi.org/10.1016/s0021-9258(17)32213-5 -
7
المصدر: Cell Calcium. 15:99-108
مصطلحات موضوعية: Physiology, Ryanodine receptor, Muscles, T-type calcium channel, chemistry.chemical_element, Cell Biology, Calcium, N-type calcium channel, Ryanodine receptor 2, Tacrolimus, R-type calcium channel, Sarcoplasmic Reticulum, chemistry, Biochemistry, Caffeine, Calcium flux, Biophysics, Animals, Calcium Channels, Rabbits, Terminal cisternae, Molecular Biology, Immunosuppressive Agents
-
8
المؤلفون: Thottala Jayaraman, Andrew Marks, Gregory J. Wiederrecht, Hitoshi Onoue, Sidney Fleischer, A.P. Timerman
المصدر: Biochemical and Biophysical Research Communications. 198:701-706
مصطلحات موضوعية: Biophysics, Muscle Proteins, chemistry.chemical_element, Calcium, Biology, Biochemistry, Ryanodine receptor 2, law.invention, Tacrolimus Binding Proteins, Cytosol, Dogs, Western blot, law, medicine, Animals, Molecular Biology, Heat-Shock Proteins, medicine.diagnostic_test, Ryanodine receptor, Muscles, Myocardium, Endoplasmic reticulum, Binding protein, Skeletal muscle, Ryanodine Receptor Calcium Release Channel, Cell Biology, Molecular biology, Sarcoplasmic Reticulum, medicine.anatomical_structure, chemistry, Recombinant DNA, Calcium Channels, Rabbits, Carrier Proteins, Protein Binding
-
9
المصدر: Journal of Biological Chemistry. 268:22737-22745
مصطلحات موضوعية: Cyclin E, Cyclin D, Cyclin A, Cyclin B, Cell Biology, Biology, Biochemistry, Cell biology, Cyclin-dependent kinase, Cyclin-dependent kinase complex, biology.protein, Molecular Biology, Cyclin A2, CDC2 Protein Kinase
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_________::884d6360d1271314cc8bb47a39af0dda
https://doi.org/10.1016/s0021-9258(18)41589-x -
10
المؤلفون: Gregory J. Wiederrecht, James P. Springer, Jeffrey D. Hermes, Jennifer Rotonda, Joseph W. Becker, Brian M. McKeever, H K Chan, Alice I. Marcy
المصدر: Journal of Biological Chemistry. 268:11335-11339
مصطلحات موضوعية: medicine.medical_treatment, Binding protein, Cell Biology, Biology, Ligand (biochemistry), Biochemistry, Calcineurin, Immunosuppressive drug, FKBP, Intracellular receptor, medicine, Receptor, Molecular Biology, Intracellular
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_________::9243f0f0ce375443ec4cee7341349bbb
https://doi.org/10.1016/s0021-9258(18)82129-9