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1
المصدر: Bioorganic & Medicinal Chemistry. 21:7216-7221
مصطلحات موضوعية: Ramipril, Clinical Biochemistry, Organophosphonates, Pharmaceutical Science, Angiotensin-Converting Enzyme Inhibitors, Peptidyl-Dipeptidase A, Pharmacology, Biochemistry, chemistry.chemical_compound, Catalytic Domain, Drug Discovery, Perindopril, medicine, Humans, Molecular Biology, Binding Sites, biology, Chemistry, Organic Chemistry, Stereoisomerism, Angiotensin-converting enzyme, Phosphonate, Enzyme Activation, Molecular Docking Simulation, biology.protein, Molecular Medicine, Protein Binding, circulatory and respiratory physiology, medicine.drug
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2
المؤلفون: Gilles Ferry, Philip M. Kubara, Bruno Pfeiffer, Jean-Paul Renaud, Stéphane Léonce, Celine Bossard, Patrick Casara, Michelle Prudhomme, Guillaume de Nanteuil, Roy M. Golsteyn, Alain Pierré, Jean A. Boutin, Michel Wierzbicki, Denis Zeyer, Aurélie Studeny
المصدر: Life Sciences. 89:259-268
مصطلحات موضوعية: animal structures, Cell Survival, medicine.drug_class, Carbazoles, Adenocarcinoma, Spodoptera, Topoisomerase-I Inhibitor, Biology, environment and public health, General Biochemistry, Genetics and Molecular Biology, Cell Line, Tumor, medicine, Animals, Humans, CHEK1, General Pharmacology, Toxicology and Pharmaceutics, Protein kinase A, DNA-PKcs, DNA, Neoplasm, General Medicine, G2-M DNA damage checkpoint, Cell cycle, Cell biology, enzymes and coenzymes (carbohydrates), Biochemistry, Checkpoint Kinase 1, Colonic Neoplasms, Cancer cell, Drug Screening Assays, Antitumor, Topoisomerase I Inhibitors, biological phenomena, cell phenomena, and immunity, Protein Kinases, Topoisomerase inhibitor, DNA Damage
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3
المؤلفون: Anne Bretéché, Pascal Marchand, Marie-Renée Nourrisson, Patrick Hautefaye, Guillaume De Nanteuil, Muriel Duflos
المصدر: Tetrahedron. 67:4767-4773
مصطلحات موضوعية: Organic Chemistry, Drug Discovery, Biochemistry
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4
المؤلفون: Gunnar Flik, Trynke R. de Jong, Millan Mark, Guillaume de Nanteuil, Anne Dekeyne, Clotilde Mannoury la Cour, Berend Olivier, Françoise Lejeune, Thomas I. F. H. Cremers, Mauricette Brocco, Jean-Michel Rivet, Alain Gobert, Benjamin Di Cara
المصدر: European Neuropsychopharmacology. 20:599-621
مصطلحات موضوعية: Male, Substance P, Pharmacology, Piperazines, Reuptake, Mice, Radioligand Assay, chemistry.chemical_compound, Neurokinin-1 Receptor Antagonists, Pregnancy, Pharmacology (medical), Extracellular Signal-Regulated MAP Kinases, Aprepitant, Pain Measurement, Serotonin Plasma Membrane Transport Proteins, Behavior, Animal, Brain, Receptors, Neurokinin-1, Receptor antagonist, Antidepressive Agents, Paroxetine, Psychiatry and Mental health, Neurology, Indans, Antidepressant, Female, Selective Serotonin Reuptake Inhibitors, medicine.drug, Serotonin, medicine.medical_specialty, medicine.drug_class, Morpholines, Guinea Pigs, Motor Activity, Stress, Physiological, Internal medicine, medicine, Animals, Humans, Rats, Wistar, Biological Psychiatry, Rats, Endocrinology, Anxiogenic, chemistry, Neurology (clinical), Gerbillinae, Reuptake inhibitor
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5
المؤلفون: Pascal Marchand, Marie-Renée Nourrisson, Anne Breteche, Muriel Duflos, Guillaume De Nanteuil
المصدر: Tetrahedron. 66:4490-4494
مصطلحات موضوعية: chemistry.chemical_compound, Chemistry, Group (periodic table), Stereochemistry, Organic Chemistry, Drug Discovery, Pyridine, Surface modification, Biochemistry
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6
المؤلفون: Clotilde Mannoury la Cour, Manuelle Touzard, Trynke R. deJong, Mauricette Brocco, Sylvie Girardon, Anne Dekeyne, Guillaume de Nanteuil, Millan Mark, Sylvie Veiga, Berend Olivier
المصدر: European Neuropsychopharmacology. 18:729-750
مصطلحات موضوعية: Male, Agonist, medicine.drug_class, Substance P, Motor Activity, Pharmacology, Binding, Competitive, Anxiolytic, Vestipitant, Mice, chemistry.chemical_compound, Neurokinin-1 Receptor Antagonists, Piperidines, medicine, Animals, Interpersonal Relations, Pharmacology (medical), Rats, Wistar, Extracellular Signal-Regulated MAP Kinases, Receptor, Biological Psychiatry, Behavior, Animal, Dose-Response Relationship, Drug, Chemistry, Antagonist, Fear, Receptor antagonist, Rats, Enzyme Activation, Fluorobenzenes, Psychiatry and Mental health, Nociception, Neurology, Female, Neurology (clinical), Vocalization, Animal, Gerbillinae, Locomotion, Psychomotor Performance, Protein Binding
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7
المؤلفون: Jean-Charles Quirion, Philippe Gloanec, Guillaume De Nanteuil, Nicolas Boyer, Philippe Jubault
المصدر: European Journal of Organic Chemistry. 2008:4277-4295
مصطلحات موضوعية: chemistry.chemical_compound, Amino esters, Chemistry, Stereochemistry, Organic Chemistry, Functional group, β lactams, Organic chemistry, Physical and Theoretical Chemistry, Reformatsky reaction
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8
المؤلفون: Isabelle Richard, Roger Gaertner, Guillaume De Nanteuil, Alain Benoist, Philippe Mennecier, Alain Rupin, Tony Verbeuren
المصدر: Thrombosis Research. 122:265-270
مصطلحات موضوعية: Risk, Time Factors, medicine.medical_treatment, Thiophenes, Pharmacology, Inhibitory Concentration 50, chemistry.chemical_compound, In vivo, Plasminogen Activator Inhibitor 1, Fibrinolysis, medicine, Animals, Humans, Vitronectin, Infusions, Intravenous, IC50, Urokinase, Dose-Response Relationship, Drug, Indoleacetic Acids, biology, Biphenyl Compounds, Thrombosis, Hematology, Recombinant Proteins, In vitro, Rats, Models, Chemical, chemistry, Biochemistry, Tissue Plasminogen Activator, Plasminogen activator inhibitor-1, biology.protein, Plasminogen activator, medicine.drug
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9
المؤلفون: Nicolas Boyer, Guillaume De Nanteuil, Philippe Jubault, Jean-Charles Quirion, Philippe Gloanec
المصدر: Tetrahedron. 63:12352-12366
مصطلحات موضوعية: Chiral auxiliary, chemistry.chemical_compound, chemistry, Stereochemistry, Organic Chemistry, Drug Discovery, β lactams, Amine gas treating, Stereoselectivity, Reformatsky reaction, Biochemistry
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10
المؤلفون: Pierre-Alain Boyer, Philippe Morain, Jean-Loïc Robin, Pierre Lestage, Guillaume De Nanteuil, David Guez, Roeline Jochemsen
المصدر: CNS Drug Reviews. 8:31-52
مصطلحات موضوعية: Aging, Indoles, Serine Proteinase Inhibitors, Amnesia, Substance P, Pharmacology, Neuroprotection, Article, chemistry.chemical_compound, Prolyl endopeptidase, medicine, Animals, Humans, Learning, Memory impairment, Memory Disorders, Working memory, Serine Endopeptidases, Cognition, S-17092, Thiazoles, Neuropsychology and Physiological Psychology, chemistry, Mechanism of action, Models, Animal, Thiazolidines, medicine.symptom, Cognition Disorders, Prolyl Oligopeptidases, Psychology, Neuroscience, medicine.drug