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1دورية أكاديمية
المؤلفون: David Adams, Sven Taylor, Stephan Röver, Hans Richter, Jean-Marc Plancher, Jacques Mizrahi, Craig S. Malcolm, Antony R. Knight, Guy A. Kennett, Paul Hebeisen, Ian A. Cliffe, Anne Bourson, Caterina Bissantz, Jon M. Bentley, Mike J. Bickerdike, Agnès Bénardeau, Steven P. Vickers
المصدر: CHIMIA, Vol 58, Iss 9 (2004)
مصطلحات موضوعية: Obesity, Pyrroloindole, 5-ht2c receptor agonist, Sulfamidate, Chemistry, QD1-999
وصف الملف: electronic resource
Relation: https://chimia.ch/chimia/article/view/3877; https://doaj.org/toc/0009-4293; https://doaj.org/toc/2673-2424
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2
المؤلفون: Sarah Dugdale, Ian Yule, Anthony R Knight, Chen I-Jen, Tim Haymes, Sean Lightowler, Heather Simmonite, Mike Comer, Anthony Padfield, Teresa Brooks, Allan M. Jordan, A Misra, Guy A. Kennett, Angela Merrett, Simon Bedford, K Benwell, Melanie Wong, Karine G. Poullennec, Loic LeStrat, Mark Reece, Burkhard Klenke
المصدر: Bioorganic & Medicinal Chemistry Letters. 19:5945-5949
مصطلحات موضوعية: Receptor, Adenosine A2A, Clinical Biochemistry, Pharmaceutical Science, Pharmacology, Receptor, Adenosine A2B, Biochemistry, Receptor subtype, Pulmonary Disease, Chronic Obstructive, Administration, Inhalation, Drug Discovery, Animals, Humans, Receptor, Molecular Biology, Chemistry, Organic Chemistry, Antagonist, Adenosine receptor, Asthma, In vitro, Adenosine A2 Receptor Antagonists, Rats, Pharmacokinetic analysis, Pyrimidines, Nociception, Drug Design, Molecular Medicine, Adenosine A2B receptor
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المؤلفون: Nathaniel J. T. Monck, A Misra, K Benwell, Teresa Brooks, Antony R. Knight, Nicolas Foloppe, Guy A. Kennett
المصدر: Bioorganic & Medicinal Chemistry Letters. 19:4183-4190
مصطلحات موضوعية: Cannabinoid receptor, Molecular model, Chemistry, Pharmaceutical, medicine.medical_treatment, Clinical Biochemistry, Drug Evaluation, Preclinical, Pharmaceutical Science, Ligands, Biochemistry, Receptor, Cannabinoid, CB2, Mice, Piperidines, Receptor, Cannabinoid, CB1, Rimonabant, Drug Discovery, medicine, Animals, Humans, Obesity, Receptor, Molecular Biology, Binding selectivity, Cannabis, Virtual screening, Dose-Response Relationship, Drug, Molecular Structure, Cannabinoids, Chemistry, Organic Chemistry, Models, Chemical, Drug Design, Pyrazoles, Molecular Medicine, Cannabinoid, Pharmacophore, medicine.drug
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4
المصدر: European Journal of Neuroscience. 25:3115-3124
مصطلحات موضوعية: Agonist, medicine.medical_specialty, medicine.drug_class, Chemistry, General Neuroscience, Receptor antagonist, Serotonergic, 5-HT2C receptor, medicine.anatomical_structure, Endocrinology, Internal medicine, medicine, Serotonin 5-HT2 Receptor Antagonists, Serotonin, Receptor, Basolateral amygdala
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5
المؤلفون: Peter G. Clifton, Guy A. Kennett
المصدر: CNS & Neurological Disorders - Drug Targets. 5:293-312
مصطلحات موضوعية: Pharmacology, Chemistry, General Neuroscience, media_common.quotation_subject, Dopaminergic, Histaminergic, Adrenergic, Appetite, Feeding Behavior, Serotonergic, Receptors, Adrenergic, Reuptake, Monoamine neurotransmitter, Receptors, Biogenic Amine, Receptors, Serotonin, Animals, Humans, Receptors, Histamine, Energy Metabolism, Receptor, media_common
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::7af00fe7dcec565f67902a09181e0989
https://doi.org/10.2174/187152706777452254 -
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المصدر: Psychopharmacology. 185:45-57
مصطلحات موضوعية: Male, Agonist, medicine.medical_specialty, Indoles, Pyridines, medicine.drug_class, Aminopyridines, Biology, Satiety Response, Piperazines, Mice, chemistry.chemical_compound, Internal medicine, Receptor, Serotonin, 5-HT2C, medicine, Animals, Receptor, Neurotransmitter, 5-HT receptor, Mice, Knockout, Pharmacology, Antagonist, Feeding Behavior, Serotonin 5-HT1 Receptor Agonists, Receptor antagonist, Serotonin Receptor Agonists, 5-HT2C receptor, Endocrinology, chemistry, Receptor, Serotonin, 5-HT1B, Serotonin 5-HT2 Receptor Antagonists, Female, Serotonin Antagonists, Serotonin, Serotonin 5-HT2 Receptor Agonists
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7
المؤلفون: Guy A. Kennett, A Misra, David R. Adams, Ashley Roger George, Howard Langham Mansell, Corinna Dagmar Bodkin, Ian Anthony Cliffe, K Quirk, K Benwell, Steven P. Vickers, Jonathan Mark Bentley, M J Bickerdike, Colin T. Dourish, C.S. Malcolm, Roffey Jonathan Richard Anthon, Antony R. Knight
المصدر: Bioorganic & Medicinal Chemistry Letters. 16:677-680
مصطلحات موضوعية: Agonist, Stereochemistry, medicine.drug_class, Clinical Biochemistry, Pharmaceutical Science, Biochemistry, Chemical synthesis, Eating, Radioligand Assay, chemistry.chemical_compound, In vivo, Drug Discovery, medicine, Animals, Pyrroles, Receptor, Molecular Biology, 5-HT receptor, Chemistry, Organic Chemistry, Quinoline, Isoquinolines, In vitro, Rats, Serotonin Receptor Agonists, 5-HT2C receptor, Disease Models, Animal, Quinolines, Molecular Medicine, Anti-Obesity Agents, Serotonin 5-HT2 Receptor Agonists
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8
المؤلفون: A Misra, Porter Richard Hugh Phillip, Anne Bourson, M. Muller, P Coassolo, Jacques Mizrahi, Hans Richter, Ian Anthony Cliffe, M J Bickerdike, Steven P. Vickers, David R. Adams, C.S. Malcolm, Patrizio Mattei, Jonathan Mark Bentley, Guy A. Kennett, Colin T. Dourish, Stephan Röver, Sven Taylor, James Edward Paul Davidson, Paul Hebeisen, Antony R. Knight, Agnès Bénardeau
المصدر: Bioorganic & Medicinal Chemistry Letters. 15:3604-3608
مصطلحات موضوعية: Agonist, Indoles, Pyridines, medicine.drug_class, Stereochemistry, Injections, Subcutaneous, Clinical Biochemistry, Pharmaceutical Science, Biochemistry, Chemical synthesis, Eating, Structure-Activity Relationship, In vivo, Drug Discovery, medicine, Animals, Rats, Wistar, Receptor, Molecular Biology, 5-HT receptor, Chemistry, Organic Chemistry, Rats, Serotonin Receptor Agonists, 5-HT2C receptor, Pyrazines, Molecular Medicine, 5-HT2C receptor agonist, Selectivity, Serotonin 5-HT2 Receptor Agonists
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9
المؤلفون: A. Wyatt, L. J. Webster, Steven P. Vickers, Colin T. Dourish, Guy A. Kennett
المصدر: Europe PubMed Central
مصطلحات موضوعية: Male, medicine.medical_specialty, Time Factors, Cannabinoid receptor, Receptors, Drug, medicine.medical_treatment, Motor Activity, Weight Gain, Eating, Piperidines, Rimonabant, Internal medicine, Appetite Depressants, medicine, Animals, Receptors, Cannabinoid, Pharmacology, Dose-Response Relationship, Drug, Cannabinoids, Chemistry, Antagonist, Rats, Rats, Zucker, Endocrinology, nervous system, Anorectic, Lean body mass, Pyrazoles, lipids (amino acids, peptides, and proteins), Cannabinoid, medicine.symptom, Energy Metabolism, Weight gain, Cyclobutanes, medicine.drug, Sibutramine
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10
المصدر: European Journal of Neuroscience. 17:185-190
مصطلحات موضوعية: medicine.medical_specialty, medicine.drug_class, General Neuroscience, Wild type, Biology, Receptor antagonist, Locomotor activity, 5-HT2C receptor, Endocrinology, Internal medicine, Knockout mouse, medicine, Psychopharmacology, Receptor, Function (biology)