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1
المؤلفون: Halina T Serafinowska, Claire M. Scott, Jeannette M. Watson, Kathryn R. Starr, Peter J. Lovell, Giancarlo Merlo, Frank E. Blaney, Paul W. Smith
المصدر: Bioorganic & Medicinal Chemistry Letters. 18:5581-5585
مصطلحات موضوعية: Male, Stereochemistry, Chemistry, Pharmaceutical, Clinical Biochemistry, Molecular Conformation, Administration, Oral, Pharmaceutical Science, Serotonin 5-HT1 Receptor Antagonists, Biochemistry, Reuptake, chemistry.chemical_compound, Drug Discovery, Animals, Humans, Receptor, Neurotransmitter, Molecular Biology, 5-HT receptor, Serotonin transporter, Chromatography, biology, Chemistry, Organic Chemistry, Rats, Kinetics, Models, Chemical, Docking (molecular), Drug Design, biology.protein, Molecular Medicine, Serotonin, Reuptake inhibitor, Selective Serotonin Reuptake Inhibitors
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2
المؤلفون: Halina T Serafinowska, Helen Newman, Frank D. King, Douglas R Smith, Stephen E. Clarke, Graham J. Riley, Steven Mark Bromidge, Peter J. Lovell, David R. Thomas, Carol Routledge
المصدر: Bioorganic & Medicinal Chemistry Letters. 12:1357-1360
مصطلحات موضوعية: Models, Molecular, Stereochemistry, Clinical Biochemistry, Molecular Conformation, Pharmaceutical Science, Biochemistry, Chemical synthesis, Piperazines, Structure-Activity Relationship, chemistry.chemical_compound, SB-271046, Drug Discovery, Thiophene, Structure–activity relationship, Receptor, Molecular Biology, 5-HT receptor, Sulfonamides, Bicyclic molecule, Organic Chemistry, Kinetics, chemistry, Drug Design, Receptors, Serotonin, 5-HT6 receptor, Molecular Medicine, Serotonin Antagonists
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3
المؤلفون: Douglas R Smith, Warren D. Hirst, Derek C. Rogers, Neil Upton, Mark S. Duxon, Nigel Deeks, Sarah Bartlett, Graham J. Riley, Tania O. Stean, David R. Thomas, Gary W. Price, Steven Mark Bromidge, Halina T Serafinowska
المصدر: Pharmacology Biochemistry and Behavior. 71:645-654
مصطلحات موضوعية: Male, Swine, medicine.drug_class, Clinical Biochemistry, Pharmacology, Toxicology, Biochemistry, Piperazines, Rats, Sprague-Dawley, Radioligand Assay, Behavioral Neuroscience, chemistry.chemical_compound, Cognition, Seizures, Cyclic AMP, medicine, Animals, Humans, Maze Learning, Receptor, Biological Psychiatry, 5-HT receptor, Brain Chemistry, Electroshock, Sulfonamides, Membranes, Seizure threshold, Chemistry, Antagonist, Brain, SB-357134, Biological activity, Receptor antagonist, Recombinant Proteins, Rats, Receptors, Serotonin, Anesthesia, Exploratory Behavior, 5-HT6 receptor, Serotonin Antagonists, Algorithms
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4
المؤلفون: Ivan Leo Pinto, Richard L. Jarvest, Halina T. Serafinowska
المصدر: Tetrahedron Letters. 41:1597-1600
مصطلحات موضوعية: chemistry.chemical_compound, Four component, Chemistry, Organic Chemistry, Drug Discovery, Polymer chemistry, Alkoxy group, Thiophene, Condensation reaction, Biochemistry
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5
المؤلفون: Richard L. Jarvest, L.John Jennings, Susan C. Connor, Halina T. Serafinowska, Joselina G. Gorniak, Andrew West
المصدر: Bioorganic & Medicinal Chemistry Letters. 7:1733-1738
مصطلحات موضوعية: chemistry.chemical_classification, Proteases, Protease, biology, Chemistry, medicine.medical_treatment, Organic Chemistry, Clinical Biochemistry, Pharmaceutical Science, Pharmacology, biology.organism_classification, Biochemistry, In vitro, Virus, Enzyme, Betaherpesvirinae, Enzyme inhibitor, Drug Discovery, medicine, biology.protein, Molecular Medicine, Protease inhibitor (pharmacology), Molecular Biology
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6
المؤلفون: Joselina G. Gorniak, Martin J. Parratt, Richard L. Jarvest, James E. Strickler, Christine Debouck, Halina T. Serafinowska, L.John Jennings
المصدر: Bioorganic & Medicinal Chemistry Letters. 6:2463-2466
مصطلحات موضوعية: Protease, Stereochemistry, Benzoxazinones, Chemistry, medicine.medical_treatment, Organic Chemistry, Clinical Biochemistry, Pharmaceutical Science, Mechanism based, HSL and HSV, Mass spectrometry, Biochemistry, Drug Discovery, medicine, Molecular Medicine, Molecular Biology
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7
المؤلفون: Michael Raymond Harnden, Halina T. Serafinowska
المصدر: Bioorganic & Medicinal Chemistry Letters. 6:2215-2218
مصطلحات موضوعية: chemistry.chemical_compound, Biochemistry, chemistry, Guanine, Organic Chemistry, Clinical Biochemistry, Drug Discovery, Pharmaceutical Science, Molecular Medicine, Purine metabolism, Molecular Biology, Peripheral blood
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8
المؤلفون: Michael Raymond Harnden, Halina T. Serafinowska
المصدر: Nucleosides and Nucleotides. 13:903-913
مصطلحات موضوعية: Ganciclovir, Chemistry, Guanine, Acyclic nucleoside, Biochemistry, Medicinal chemistry, Thiophosphate, Turn (biochemistry), chemistry.chemical_compound, Sodium thiophosphate, Penciclovir, Genetics, medicine, Organic chemistry, Hydroxymethyl, medicine.drug
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9
المؤلفون: Halina T. Serafinowska, Michael Raymond Harnden
المصدر: ChemInform. 28
مصطلحات موضوعية: chemistry.chemical_compound, Biochemistry, Chemistry, Guanine, Nucleic acid, General Medicine, Purine metabolism, Peripheral blood
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10
المصدر: ChemInform. 22
مصطلحات موضوعية: Solid-phase synthesis, Chemistry, Nucleic acid, Polyribonucleotides, General Medicine, Combinatorial chemistry