-
1
المؤلفون: David G. Tew, Alfonso Rivera-Sagredo, Paloma Perez, Cheryl A. Janson, Nestor O. Concha, Martin Gilpin, Juan A. Hueso-Rodríguez, Michael Rees, John H. Bateson, Jesús Ángel de la Fuente, Helen F. Boyd, Niconovich Nancy, Stewart C. Pearson, Christy Cheever, David J. Payne, E. Diez, Stephen Rittenhouse
المصدر: Antimicrobial Agents and Chemotherapy. 46:1880-1886
مصطلحات موضوعية: Models, Molecular, medicine.drug_class, Klebsiella pneumoniae, Antibiotics, Bacillus, Microbial Sensitivity Tests, Chaetomium, medicine.disease_cause, beta-Lactamases, Microbiology, Bacillus cereus, polycyclic compounds, medicine, Pharmacology (medical), Enzyme Inhibitors, Antibacterial agent, Pharmacology, chemistry.chemical_classification, Binding Sites, biology, Pseudomonas aeruginosa, Drug Synergism, Meropenem, Chemistry, Biosynthesis, biochemical phenomena, metabolism, and nutrition, bacterial infections and mycoses, biology.organism_classification, Kinetics, Infectious Diseases, Enzyme, Biochemistry, chemistry, Enzyme inhibitor, Fermentation, Serratia marcescens, biology.protein, bacteria, Thienamycins, Bacteroides fragilis, beta-Lactamase Inhibitors, Heterocyclic Compounds, 3-Ring
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::e9aa937c16cee0ca888b0a557de1cdef
https://doi.org/10.1128/aac.46.6.1880-1886.2002 -
2
المؤلفون: Andrew Keith Forrest, Murray J. B. Brown, Martin Hibbs, Valerie Berry, Robert J. Sheppard, Deborah Dee Jaworski, John S. Elder, Courtney Slater-Radosti, Peter J. O'Hanlon, Helen F. Boyd, John M. Berge, Richard L. Jarvest, Andrew J. Pope, Angela Worby, Andrew P. Fosberry, Daniel R. Gentry, Stephen Rittenhouse
المصدر: Journal of Medicinal Chemistry. 45:1959-1962
مصطلحات موضوعية: Staphylococcus aureus, Micrococcaceae, medicine.drug_class, Staphylococcus, Antibiotics, Methionine-tRNA Ligase, Quinolones, medicine.disease_cause, Microbiology, Rats, Sprague-Dawley, Structure-Activity Relationship, Staphylococcus epidermidis, Drug Resistance, Bacterial, Drug Discovery, medicine, Animals, Enzyme Inhibitors, Antibacterial agent, biology, Chemistry, Biological activity, biology.organism_classification, Abscess, Anti-Bacterial Agents, Rats, Biochemistry, Molecular Medicine, Antibacterial activity, Enterococcus, Bacteria
-
3
المؤلفون: Deirdre M. B. Hickey, Ian Stansfield, Leach Colin Andrew, Caroline M. Whittaker, Ivan Leo Pinto, Stephen A. Smith, Stephen Christopher Martin Fell, Sean Thomas Flynn, Kitty Moores, Helen F. Boyd, Colin J. Theobald, David G. Tew, Roderick A. Porter, Robert John Ife, Kevin J. Milliner, Colin H. Macphee, D. Anthony Rawlings
المصدر: Bioorganic & Medicinal Chemistry Letters. 10:2557-2561
مصطلحات موضوعية: medicine.drug_class, Stereochemistry, Lipoproteins, Clinical Biochemistry, Administration, Oral, Pharmaceutical Science, Carboxamide, Pyrimidinones, Biochemistry, Chemical synthesis, Phospholipases A, chemistry.chemical_compound, Phospholipase A2, Oral administration, Drug Discovery, medicine, Animals, Enzyme Inhibitors, Molecular Biology, chemistry.chemical_classification, Molecular Structure, biology, Chemistry, Lipoprotein-associated phospholipase A2, Organic Chemistry, Phospholipases A2, Enzyme, Enzyme inhibitor, biology.protein, Lactam, Molecular Medicine, Rabbits
-
4
المؤلفون: Martin Jones, Colin J. Theobald, Leach Colin Andrew, Sean Thomas Flynn, Deirdre M. B. Hickey, Ian Stansfield, David G. Tew, Brian Peter Slingsby, Helen F. Boyd, Stephen A. Smith, Kevin J. Milliner, Colin H. Macphee, Robert John Ife, D. Anthony Rawlings
المصدر: Bioorganic & Medicinal Chemistry Letters. 10:395-398
مصطلحات موضوعية: Stereochemistry, High-throughput screening, Clinical Biochemistry, Drug Evaluation, Preclinical, Pharmaceutical Science, Pyrimidinones, Biochemistry, Chemical synthesis, Phospholipases A, Substrate Specificity, Inhibitory Concentration 50, Structure-Activity Relationship, Phospholipase A2, Drug Discovery, Humans, Enzyme Inhibitors, Molecular Biology, chemistry.chemical_classification, biology, Chemistry, Lipoprotein-associated phospholipase A2, Organic Chemistry, Substrate (chemistry), Phospholipases A2, Enzyme, Enzyme inhibitor, Drug Design, 1-Alkyl-2-acetylglycerophosphocholine Esterase, biology.protein, Molecular Medicine, Selectivity
-
5
المؤلفون: Helen F. Boyd, Deirdre M. B. Hickey, Kitty Moores, Kevin J. Milliner, Colin H. Macphee, Dash Dhanak, Keith E. Suckling, Leach Colin Andrew, Rebecca A. Patterson, Robert John Ife, David S. Leake, David G. Tew
المصدر: Biochemical Journal. 338:479-487
مصطلحات موضوعية: chemistry.chemical_classification, biology, Lipoprotein-associated phospholipase A2, Fatty acid, Cell Biology, 1-Alkyl-2-acetylglycerophosphocholine Esterase, Biochemistry, chemistry.chemical_compound, Phospholipase A2, Lysophosphatidylcholine, chemistry, Low-density lipoprotein, biology.protein, lipids (amino acids, peptides, and proteins), Chemoattractant activity, Molecular Biology, Lipoprotein
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_________::fbda5ac7d34f8ba6f99f2e2fc0fda486
https://doi.org/10.1042/bj3380479 -
6
المؤلفون: David G. Tew, Patrick Camilleri, Patricia Sweeney, Nigel J. Pearce, Anthony N. Shaw, Theo A. Berkhout, John W. Yates, Brian Jackson, Helen F. Boyd, Pieter H. E. Groot, Andrew Derrick Gribble
المصدر: Biochemical Journal. 334:113-119
مصطلحات موضوعية: medicine.medical_specialty, Very low-density lipoprotein, ATP citrate lyase, Triglyceride, Cholesterol, ATP Citrate (pro-S)-Lyase, Lipid metabolism, Cell Biology, Biology, Biochemistry, chemistry.chemical_compound, Endocrinology, chemistry, Internal medicine, medicine, lipids (amino acids, peptides, and proteins), Molecular Biology, Fatty acid synthesis, Lipoprotein
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_________::07b90e7279f49fc3d28bbc236f1d1907
https://doi.org/10.1042/bj3340113 -
7
المصدر: Biochemistry. 37:10087-10093
مصطلحات موضوعية: Lactams, Stereochemistry, Kinetics, beta-Lactams, Biochemistry, Phospholipases A, Substrate Specificity, Hydrolysis, Phospholipase A2, Peptide bond, Lipase, Chromatography, High Pressure Liquid, biology, Chemistry, Spectrum Analysis, Stereoisomerism, Enzyme Activation, Lipoproteins, LDL, Phospholipases A2, Burst kinetics, Covalent bond, 1-Alkyl-2-acetylglycerophosphocholine Esterase, biology.protein, Azetidines, Enantiomer
-
8
المؤلفون: Helen F. Boyd, Stephen Christopher Martin Fell, Stephen A. Smith, Deirdre Mary Bernadette Hickey, Colin A. Leach, Colin J. Theobald, Colin H. Macphee, Caroline M. Whittaker, D. Anthony Rawlings, Ivan Leo Pinto, Ian Stansfield, Steven J. Stanway, Kevin J. Milliner, Robert J. Ife
المصدر: Bioorganicmedicinal chemistry letters. 12(1)
مصطلحات موضوعية: Clinical Biochemistry, Drug Evaluation, Preclinical, Pharmaceutical Science, Administration, Oral, Pyrimidinones, Biochemistry, Phospholipases A, law.invention, Inhibitory Concentration 50, Structure-Activity Relationship, Phospholipase A2, In vivo, law, Drug Discovery, Potency, Animals, Humans, Enzyme Inhibitors, Molecular Biology, chemistry.chemical_classification, Phospholipase A, biology, Chemistry, Lipoprotein-associated phospholipase A2, Organic Chemistry, Kinetics, Enzyme, Enzyme inhibitor, Drug Design, 1-Alkyl-2-acetylglycerophosphocholine Esterase, biology.protein, Recombinant DNA, Molecular Medicine, Rabbits
-
9
المؤلفون: Maxine A. Taylor, Robert J. Ife, Colin H. Macphee, Kevin J. Milliner, Ivan Leo Pinto, Jackie C. Bloomer, Steven J. Stanway, Colin A. Leach, D. Anthony Rawlings, Stephen A. Smith, Ian Stansfield, Caroline M. Whittaker, Helen F. Boyd, Colin J. Theobald, Deirdre Mary Bernadette Hickey
المصدر: Bioorganicmedicinal chemistry letters. 11(14)
مصطلحات موضوعية: medicine.drug_class, Metabolic Clearance Rate, Clinical Biochemistry, Pharmaceutical Science, Administration, Oral, Carboxamide, Pyrimidinones, Biochemistry, Phospholipases A, Piperazines, law.invention, Inhibitory Concentration 50, Phospholipase A2, law, Drug Discovery, medicine, Potency, Animals, Humans, Enzyme Inhibitors, Molecular Biology, chemistry.chemical_classification, Phospholipase A, biology, Organic Chemistry, In vitro, Rats, Enzyme, chemistry, Enzyme inhibitor, 1-Alkyl-2-acetylglycerophosphocholine Esterase, biology.protein, Recombinant DNA, Microsomes, Liver, Molecular Medicine, Rabbits
-
10
المؤلفون: Colin A. Leach, Colin H. Macphee, V.Ann Lewis, Kevin J. Milliner, Ivan Leo Pinto, Ian Stansfield, Robert J. Ife, Caroline M. Whittaker, Beverley Hammond, Helen F. Boyd, Deirdre Mary Bernadette Hickey, Stephen A. Smith, Colin J. Theobald
المصدر: Bioorganicmedicinal chemistry letters. 11(5)
مصطلحات موضوعية: Male, medicine.drug_class, Arteriosclerosis, Clinical Biochemistry, Pharmaceutical Science, Carboxamide, Pyrimidinones, Biochemistry, Phospholipases A, chemistry.chemical_compound, Phospholipase A2, Drug Discovery, medicine, Potency, Animals, Humans, Pyrimidone, Enzyme Inhibitors, Molecular Biology, chemistry.chemical_classification, biology, Molecular Structure, Chemistry, Lipoprotein-associated phospholipase A2, Drug Administration Routes, Organic Chemistry, Water, In vitro, Rats, Phospholipases A2, Enzyme, Solubility, Enzyme inhibitor, biology.protein, Molecular Medicine, Rabbits