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1دورية أكاديميةOral Absorption of Middle-to-Large Molecules and Its Improvement, with a Focus on New Modality Drugs
المؤلفون: Daigo Asano, Hideo Takakusa, Daisuke Nakai
المصدر: Pharmaceutics, Vol 16, Iss 1, p 47 (2023)
مصطلحات موضوعية: middle-to-large molecule, absorption enhancer, new modality, Lipinski’s rule of five, cyclic peptide, antisense oligonucleotide, Pharmacy and materia medica, RS1-441
وصف الملف: electronic resource
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2دورية أكاديمية
المؤلفون: Kentaro Ito, Hideo Takakusa, Masayo Kakuta, Akira Kanda, Nana Takagi, Hiroyuki Nagase, Nobuaki Watanabe, Daigo Asano, Ryoya Goda, Takeshi Masuda, Akifumi Nakamura, Yoshiyuki Onishi, Toshio Onoda, Makoto Koizumi, Yasuhiro Takeshima, Masafumi Matsuo, Kiyosumi Takaishi
المصدر: Current Issues in Molecular Biology, Vol 43, Iss 3, Pp 1267-1281 (2021)
مصطلحات موضوعية: Duchenne muscular dystrophy, exon skipping, antisense oligonucleotide, dystrophin, 2′-O,4′-C-ethylene-bridged nucleic acid (ENA), renadirsen sodium, Biology (General), QH301-705.5
وصف الملف: electronic resource
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المؤلفون: Hideo Takakusa, Norihiko Iwazaki, Makiya Nishikawa, Tokuyuki Yoshida, Satoshi Obika, Takao Inoue
المصدر: Nucleic Acid Therapeutics. 33:83-94
مصطلحات موضوعية: Drug Discovery, Genetics, Molecular Medicine, Molecular Biology, Biochemistry
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_________::5895afa3c2e5946b692edfffdb2d8d96
https://doi.org/10.1089/nat.2022.0054 -
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المؤلفون: Daigo Asano, Koichi Nakamura, Yumi Nishiya, Hideyuki Shiozawa, Hideo Takakusa, Takahiro Shibayama, Shin-ichi Inoue, Tsuyoshi Shinozuka, Takakazu Hamada, Chizuko Yahara, Nobuaki Watanabe, Kouichi Yoshinari
المصدر: Drug Metabolism and Disposition. 51:67-80
مصطلحات موضوعية: Pharmacology, Pharmaceutical Science
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_________::b60456efe4bbedd2b0c9bab443faf822
https://doi.org/10.1124/dmd.122.001000 -
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المؤلفون: Akifumi Nakamura, Akira Kanda, Kiyosumi Takaishi, Nobuaki Watanabe, Hideo Takakusa, Toshio Onoda, Masayo Kakuta, Yasuhiro Takeshima, Hiroyuki Nagase, Daigo Asano, Ito Kentaro, Takeshi Masuda, Yoshiyuki Onishi, Makoto Koizumi, Masafumi Matsuo, Nana Takagi, Ryoya Goda
المصدر: Current Issues in Molecular Biology, Vol 43, Iss 90, Pp 1267-1281 (2021)
Current Issues in Molecular Biology
Volume 43
Issue 3
Pages 90-1281مصطلحات موضوعية: Duchenne muscular dystrophy, antisense oligonucleotide, musculoskeletal diseases, Microbiology (medical), congenital, hereditary, and neonatal diseases and abnormalities, cardiac muscle, QH301-705.5, Nonsense mutation, Microbiology, dystrophin, Exon, medicine, renadirsen sodium, Biology (General), Muscular dystrophy, Molecular Biology, 2′-O,4′-C-ethylene-bridged nucleic acid (ENA), biology, business.industry, Cardiac muscle, Skeletal muscle, General Medicine, medicine.disease, Exon skipping, medicine.anatomical_structure, biology.protein, Cancer research, business, Dystrophin, exon skipping
وصف الملف: application/pdf
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::39145bf396bf8da7e422b375dd43fe94
https://doi.org/10.3390/cimb43030090 -
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المؤلفون: Chie, Makino, Akiko, Watanabe, Manabu, Kato, Hideyuki, Shiozawa, Hideo, Takakusa, Daisuke, Nakai, Tomoyo, Honda, Nobuaki, Watanabe
المصدر: Drug metabolism and pharmacokinetics. 45
مصطلحات موضوعية: Cyclopropanes, Oxadiazoles, Administration, Oral, Rats, Receptors, G-Protein-Coupled, Rats, Sprague-Dawley, Feces, Macaca fascicularis, Species Specificity, Benzamides, Animals, Humans, Pharmacokinetics, Carbon Radioisotopes
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المؤلفون: Chie Makino, Akiko Watanabe, Manabu Kato, Hideyuki Shiozawa, Hideo Takakusa, Daisuke Nakai, Tomoyo Honda, Nobuaki Watanabe
المصدر: Drug Metabolism and Pharmacokinetics. 45:100459
مصطلحات موضوعية: Pharmacology, Pharmaceutical Science, Pharmacology (medical)
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المؤلفون: Hideo Takakusa, Osamu Ando, Jeanne Mendell, Takako Shimizu, Makiko Yamada
المصدر: Drug Metabolism and Disposition. 47:340-349
مصطلحات موضوعية: Pharmacology, medicine.medical_specialty, CYP3A, Chemistry, Glucuronidation, Pharmaceutical Science, Urine, 030226 pharmacology & pharmacy, Hydrolysate, Intestinal absorption, Excretion, 03 medical and health sciences, 0302 clinical medicine, Mineralocorticoid receptor, Endocrinology, Pharmacokinetics, 030220 oncology & carcinogenesis, Internal medicine, medicine
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_________::514cfbea3286e159d36d997827960b7c
https://doi.org/10.1124/dmd.118.084897 -
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المؤلفون: Nobuyuki Murayama, Takashi Izumi, Shin-ichi Inoue, Takuo Washio, Makiko Yamada, Hideo Takakusa, Eiko Suzuki, Masakatsu Kotsuma, Makoto Takei
المصدر: Xenobiotica. 47:1090-1103
مصطلحات موضوعية: Male, medicine.medical_specialty, Metabolic Clearance Rate, Health, Toxicology and Mutagenesis, Administration, Oral, Biological Availability, 030204 cardiovascular system & hematology, Pharmacology, Toxicology, 030226 pharmacology & pharmacy, Biochemistry, Non steroidal, Excretion, 03 medical and health sciences, 0302 clinical medicine, Mineralocorticoid receptor, Pharmacokinetics, Internal medicine, medicine, Animals, Distribution (pharmacology), Pyrroles, Tissue Distribution, Sulfones, Tissue distribution, Mineralocorticoid Receptor Antagonists, Chemistry, General Medicine, Metabolism, Disposition, Rats, Macaca fascicularis, Endocrinology, hormones, hormone substitutes, and hormone antagonists
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المؤلفون: Makiko, Yamada, Jeanne, Mendell, Hideo, Takakusa, Takako, Shimizu, Osamu, Ando
المصدر: Drug metabolism and disposition: the biological fate of chemicals. 47(3)
مصطلحات موضوعية: Adult, Male, ATP Binding Cassette Transporter, Subfamily B, Metabolic Clearance Rate, Administration, Oral, Middle Aged, Healthy Volunteers, Neoplasm Proteins, Receptors, Mineralocorticoid, Intestinal Absorption, ATP Binding Cassette Transporter, Subfamily G, Member 2, Cytochrome P-450 CYP3A, Humans, Pyrroles, Tissue Distribution, Sulfones, Caco-2 Cells, Glucuronosyltransferase, Mineralocorticoid Receptor Antagonists
URL الوصول: https://explore.openaire.eu/search/publication?articleId=pmid________::ebfc875e5513b239b270d85d40341133
https://pubmed.ncbi.nlm.nih.gov/30541878