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1
المؤلفون: Hiroshi Sai, Tsuyoshi Ogiku, Hiroshi Miyazaki, Hiroshi Ohmizu, Jun Murakami, Akio Ohtani
المصدر: Bioorganic & Medicinal Chemistry. 18:1968-1979
مصطلحات موضوعية: Serine Proteinase Inhibitors, Clinical Biochemistry, Molecular Conformation, Administration, Oral, Pharmaceutical Science, Crystallography, X-Ray, Biochemistry, Phenylbutyrate, Molecular conformation, Structure-Activity Relationship, chemistry.chemical_compound, Dogs, Fibrinolytic Agents, Bleeding time, Plasminogen Activator Inhibitor 1, Drug Discovery, Antithrombotic, Butadienes, medicine, Animals, Structure–activity relationship, Molecular Biology, Cells, Cultured, medicine.diagnostic_test, Chemistry, Organic Chemistry, Phenylbutyrates, Rats, Plasminogen activator inhibitor-1, Molecular Medicine, Fibrinolytic agent
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2
المؤلفون: Tsuyoshi Ogiku, Hiroshi Miyazaki, Hiroshi Ohmizu
المصدر: Organic Process Research & Development. 13:760-763
مصطلحات موضوعية: In situ, chemistry.chemical_compound, chemistry, Stereochemistry, Plasminogen activator inhibitor-1, Organic Chemistry, Physical and Theoretical Chemistry, Selectivity, Isomerization, Plasminogen activator, Derivative (chemistry)
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3
المؤلفون: Akio Ohtani, Hiroshi Miyazaki, Tsuyoshi Ogiku, Jun Murakami, Hiroshi Ohmizu, Hiroshi Sai
المصدر: Bioorganic & Medicinal Chemistry Letters. 18:6419-6422
مصطلحات موضوعية: Chemistry, Pharmaceutical, Clinical Biochemistry, Drug Evaluation, Preclinical, Administration, Oral, Biological Availability, Succinimides, Pharmaceutical Science, Benzylidene Compounds, Biochemistry, Chemical synthesis, chemistry.chemical_compound, Dogs, Oral administration, Plasminogen Activator Inhibitor 1, Drug Discovery, Antithrombotic, Animals, Humans, Molecular Biology, chemistry.chemical_classification, biology, Chemistry, Drug Administration Routes, Organic Chemistry, In vitro, Rats, Bioavailability, Enzyme, Models, Chemical, Solubility, Enzyme inhibitor, Drug Design, Plasminogen activator inhibitor-1, biology.protein, Molecular Medicine
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4
المؤلفون: Tsuyoshi Ogiku, Hiroshi Ohmizu, Hiroshi Sai
المصدر: Tetrahedron. 63:10345-10353
مصطلحات موضوعية: Reaction mechanism, Chemistry, Organic Chemistry, Biochemistry, Medicinal chemistry, chemistry.chemical_compound, Stereospecificity, Deprotonation, Dehydration reaction, Drug Discovery, Copper(II) chloride, Cinnamates, 1-Ethyl-3-(3-dimethylaminopropyl)carbodiimide, Stereoselectivity
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5
المؤلفون: Hiroshi Sai, Hiroshi Ohmizu, Tsuyoshi Ogiku
المصدر: Synthesis. :0201-0204
مصطلحات موضوعية: Stereochemistry, Chemistry, Organic Chemistry, General Medicine, medicine.disease, Medicinal chemistry, Catalysis, chemistry.chemical_compound, Stereospecificity, medicine, 1-Ethyl-3-(3-dimethylaminopropyl)carbodiimide, Stereoselectivity, Dehydration, Carbodiimide
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::d65d183a95ff8a51ff6b83bdeffcdbd0
https://doi.org/10.1055/s-2003-36817 -
6
المؤلفون: Keiko Saito, Toshikazu Suzuki, Hiroshi Ohmizu, Mikiko Yasuhara, Ryo Shimizu, Hitoshi Kubota, Kazuya Nakao
المصدر: Bioorganic & Medicinal Chemistry. 9:853-861
مصطلحات موضوعية: chemistry.chemical_classification, Antioxidant, biology, Stereochemistry, Carboxylic acid, medicine.medical_treatment, Organic Chemistry, Clinical Biochemistry, Sterol O-acyltransferase, Pharmaceutical Science, Biochemistry, chemistry.chemical_compound, Enzyme, chemistry, Enzyme inhibitor, Low-density lipoprotein, Drug Discovery, medicine, biology.protein, Molecular Medicine, Structure–activity relationship, lipids (amino acids, peptides, and proteins), Molecular Biology, Foam cell
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7
المؤلفون: Hiroshi Miyazaki, Yoshihiro Terakawa, Hiroshi Ohmizu, Akio Ohtani, Tsuyoshi Ogiku, Tsutomu Miyake
المصدر: Bioorganic & Medicinal Chemistry Letters. 20:546-548
مصطلحات موضوعية: Serine Proteinase Inhibitors, Stereochemistry, Clinical Biochemistry, Pharmaceutical Science, Biochemistry, Chemical synthesis, chemistry.chemical_compound, Fibrinolytic Agents, Plasminogen Activator Inhibitor 1, Drug Discovery, Humans, Molecular Biology, IC50, chemistry.chemical_classification, biology, Organic Chemistry, Biological activity, Pyrrolidinones, Enzyme, Acrylates, chemistry, Enzyme inhibitor, Drug Design, Plasminogen activator inhibitor-1, biology.protein, Lactam, Molecular Medicine, Plasminogen activator
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8
المصدر: Free Radical Research. 32:255-264
مصطلحات موضوعية: Male, Nitrilotriacetic Acid, Pyridines, Radical, medicine.medical_treatment, Intraperitoneal injection, Probucol, Pharmacology, Ferric Compounds, Thiobarbituric Acid Reactive Substances, Biochemistry, Antioxidants, Rats, Sprague-Dawley, Lipid peroxidation, chemistry.chemical_compound, Phenols, Superoxides, In vivo, TBARS, medicine, Animals, Urea, Vitamin E, Aspartate Aminotransferases, Molecular Structure, Hydroxyl Radical, Superoxide, Phenylurea Compounds, Brain, Alanine Transaminase, Free Radical Scavengers, General Medicine, Butylated Hydroxytoluene, Rats, Oxidative Stress, chemistry, Hydroxyl radical, Lipid Peroxidation, medicine.drug
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9
المؤلفون: Hiroshi Sai, Hiroshi Ohmizu
المصدر: Tetrahedron Letters. 40:5019-5022
مصطلحات موضوعية: chemistry.chemical_compound, chemistry, Dehydration reaction, Organic Chemistry, Drug Discovery, Cinnamates, 1-Ethyl-3-(3-dimethylaminopropyl)carbodiimide, Organic chemistry, Stereoselectivity, Biochemistry
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10
المؤلفون: Hiroshi Ohmizu, Shin-ichi Yoshida, Tameo Iwasaki, Tsuyoshi Ogiku
المصدر: Synthesis. 1997:1475-1480
مصطلحات موضوعية: Lignan, chemistry.chemical_compound, chemistry, Organic Chemistry, Organic chemistry, Catalysis
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_________::7ba1df18cfd42b2b36b3f70d320ee1e7
https://doi.org/10.1055/s-1997-1375