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1دورية أكاديمية
المؤلفون: Holger Scheible, Martin Dyroff, Annick Seithel‐Keuth, Eleanor Harrison‐Moench, Nadra Mammasse, Andreas Port, Angelika Bachmann, Jennifer Dong, Jan Jaap vanLier, William Tracewell, David Mitchell
المصدر: Clinical and Translational Science, Vol 14, Iss 6, Pp 2420-2430 (2021)
مصطلحات موضوعية: Therapeutics. Pharmacology, RM1-950, Public aspects of medicine, RA1-1270
وصف الملف: electronic resource
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المؤلفون: Eleanor Harrison-Moench, Jan J. van Lier, Jennifer Dong, Angelika Bachmann, David Mitchell, Andreas Port, Nadra Mammasse, Annick Seithel-Keuth, Martin Dyroff, William Tracewell, Holger Scheible
المصدر: Clinical and Translational Science, Vol 14, Iss 6, Pp 2420-2430 (2021)
Clinical and Translational Scienceمصطلحات موضوعية: Adult, Male, Drug, Adolescent, Metabolic Clearance Rate, medicine.drug_class, media_common.quotation_subject, Metabolite, Administration, Oral, RM1-950, Urine, Pharmacology, Article, General Biochemistry, Genetics and Molecular Biology, Tyrosine-kinase inhibitor, Excretion, Young Adult, chemistry.chemical_compound, Piperidines, Pharmacokinetics, medicine, Humans, General Pharmacology, Toxicology and Pharmaceutics, Protein Kinase Inhibitors, Biotransformation, Feces, media_common, business.industry, Research, General Neuroscience, Articles, General Medicine, Metabolism, Middle Aged, Protein-Tyrosine Kinases, Healthy Volunteers, Pyrimidines, chemistry, Therapeutics. Pharmacology, Public aspects of medicine, RA1-1270, business, Protein Kinases
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المؤلفون: Gloria Vendrell-Navarro, Piet Swart, Holger Scheible, Howard Burt, Christian Luepfert, Nada Abla, Floriane Lignet, Andreas Marx, Dominique Perrin
المصدر: Drug Metabolism and Disposition. 48:481-490
مصطلحات موضوعية: Chemistry, Pharmaceutical, Metabolite, Pharmaceutical Science, 030226 pharmacology & pharmacy, Praziquantel, Cell Line, 03 medical and health sciences, chemistry.chemical_compound, 0302 clinical medicine, Non-competitive inhibition, Cytochrome P-450 Enzyme System, Pharmacokinetics, parasitic diseases, Humans, Metabolomics, Drug Interactions, CYP2C9, Enzyme Assays, Pharmacology, biology, Chemistry, Cytochrome P450, Substrate (chemistry), Stereoisomerism, Metabolism, Recombinant Proteins, Kinetics, Biochemistry, 030220 oncology & carcinogenesis, Hepatocytes, Microsomes, Liver, biology.protein, Enantiomer, Oxidation-Reduction
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::0f175caf87d22f4a765237ec15c15215
https://doi.org/10.1124/dmd.119.089888 -
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المؤلفون: Cornelis E. C. A. Hop, Swapan Chowdhury, Douglas K. Spracklin, Simone Schadt, Christoph Funk, W. Griffith Humphreys, Angus N. R. Nedderman, Fumihiko Igarashi, Josh Yuan, Chandra Prakash, Frank Runge, Holger Scheible, Mark Kagan, S. Cyrus Khojasteh, Piet Swart, R. Scott Obach, Bojan Bister, Alexander David James, Susanna Tse
المصدر: BASE-Bielefeld Academic Search Engine
مصطلحات موضوعية: 0301 basic medicine, Drug Industry, Metabolite, Pharmaceutical Science, Human metabolism, Computational biology, 030226 pharmacology & pharmacy, Food and drug administration, 03 medical and health sciences, chemistry.chemical_compound, 0302 clinical medicine, Drug Discovery, Animals, Humans, Medicine, Drug Interactions, Safety testing, Pharmaceutical industry, Pharmacology, United States Food and Drug Administration, business.industry, United States, 030104 developmental biology, Pharmaceutical Preparations, chemistry, Drug development, Inactivation, Metabolic, Experimental methods, business, Drug metabolism
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::28c0739606a23742034a3be6254e08fa
https://doi.org/10.1124/dmd.117.079848 -
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المؤلفون: Friedrich Kraetzer, Holger Scheible, Andreas Marx, Andreas Johne, Elmar Wimmer
المصدر: Drug Metabolism and Disposition. 45:174-182
مصطلحات موضوعية: Adult, Male, Niacinamide, Adolescent, MAP Kinase Signaling System, Carboxylic acid, Metabolite, MAP Kinase Kinase 2, MAP Kinase Kinase 1, Deamination, Pharmaceutical Science, 030226 pharmacology & pharmacy, Young Adult, 03 medical and health sciences, chemistry.chemical_compound, 0302 clinical medicine, Biotransformation, Neoplasms, Humans, Tissue Distribution, Protein Kinase Inhibitors, Aged, Pharmacology, chemistry.chemical_classification, Chemistry, Primary metabolite, Metabolism, Middle Aged, Biochemistry, Ethanolamines, 030220 oncology & carcinogenesis, Cancer cell, Conjugate
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::3ded892c5f63e4cfe0663d2bb88dd54c
https://doi.org/10.1124/dmd.116.072934 -
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المصدر: British Journal of Clinical Pharmacology. 82:1498-1508
مصطلحات موضوعية: 0301 basic medicine, Pharmacology, Volume of distribution, medicine.medical_specialty, Metabolite, Coefficient of variation, Urology, Cancer, Urine, medicine.disease, 03 medical and health sciences, chemistry.chemical_compound, 030104 developmental biology, 0302 clinical medicine, chemistry, Pharmacokinetics, 030220 oncology & carcinogenesis, medicine, Pharmacology (medical), Geometric mean, Absolute bioavailability
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المؤلفون: Andreas Johne, Andreas Becker, Holger Scheible, Jan J. van Lier, Andreas Kovar, Oliver von Richter
المصدر: The Journal of Clinical Pharmacology. 55:815-824
مصطلحات موضوعية: Adult, Male, medicine.medical_specialty, medicine.drug_class, Cilengitide, Urine, Pharmacology, Excretion, Young Adult, chemistry.chemical_compound, Pharmacokinetics, Internal medicine, medicine, Humans, Receptors, Vitronectin, Pharmacology (medical), Infusions, Intravenous, Feces, Metabolism, Integrin alphaVbeta3, Receptor antagonist, Endocrinology, Renal Elimination, chemistry, Snake Venoms
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المؤلفون: Ana Javornik, Holger Scheible, Elmar Wimmer, Marc Laisney, Hugues Dolgos
المصدر: Xenobiotica. 43:1084-1094
مصطلحات موضوعية: Health, Toxicology and Mutagenesis, Metabolite, Glucuronidation, Administration, Oral, Biology, Pharmacology, Toxicology, Biochemistry, Mass Spectrometry, Feces, Mice, chemistry.chemical_compound, Dogs, Adenosine deaminase, Deoxyadenosine, In vivo, medicine, Animals, Humans, Cladribine, Chromatography, High Pressure Liquid, Whole blood, Haplorhini, General Medicine, In vitro, Rats, chemistry, Hepatocytes, Metabolome, biology.protein, Administration, Intravenous, Rabbits, Metabolic Networks and Pathways, medicine.drug
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المؤلفون: Hugues Dolgos, Friedrich Krätzer, Dieter Gallemann, Tetsuo Yamagata, Markus Fluck, Holger Scheible, Achim Freisleben, Elmar Wimmer
المصدر: Pharmacology Research & Perspectives
مصطلحات موضوعية: 0301 basic medicine, Integrin, Cilengitide, Pharmacology, Excretion, 03 medical and health sciences, chemistry.chemical_compound, sandwich‐cultured hepatocytes, 0302 clinical medicine, Pharmacokinetics, In vivo, Medicine, General Pharmacology, Toxicology and Pharmaceutics, biology, business.industry, Animals and human, Original Articles, In vitro, 030104 developmental biology, medicine.anatomical_structure, Neurology, chemistry, cilengitide, 030220 oncology & carcinogenesis, Hepatocyte, Renal physiology, biology.protein, Original Article, hepatobiliary, business, pharmacokinetics, in vitro and in vivo
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المؤلفون: Michael Meyring, J.J. Van Lier, Holger Scheible, Andreas Becker, Andreas Johne
المصدر: European Journal of Cancer. 51:S77
مصطلحات موضوعية: c-Met inhibitor, Cancer Research, Oncology, Chemistry, Phase (matter), Open label, Pharmacology, Single Center, Absolute bioavailability, Balance (ability)