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1
المؤلفون: Alessia Vesentini, Luigi Piero Stasi, Barbara Bertani, Matthew Hill, Jeannette M. Watson, Steven Mark Bromidge, Enrica Granci, Laura Zonzini, Valeria Zucchelli, Howard Robert Marshall, Stefania Faedo, Giancarlo Merlo, Laurie J. Gordon, Manuela Borriello
المصدر: Bioorganic & Medicinal Chemistry Letters. 18:5653-5656
مصطلحات موضوعية: Tertiary amine, Stereochemistry, Clinical Biochemistry, Pharmaceutical Science, Serotonin 5-HT1 Receptor Antagonists, Biochemistry, Piperazines, Drug Discovery, Animals, Humans, Receptor, Piperazine, Molecular Biology, 5-HT receptor, Benzoxazoles, Bicyclic molecule, Chemistry, Organic Chemistry, Antidepressive Agents, Rats, Liver, Models, Chemical, Drug Design, Molecular Medicine, Antidepressant, 5-HT1 receptor, Serotonin Antagonists, Serotonin, Reuptake inhibitor, Selective Serotonin Reuptake Inhibitors
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2
المؤلفون: Lee A. Dawson, Wyman Paul Adrian, Howard Robert Marshall, Gary W. Price, Paul W. Smith, Sean Thomas Flynn, Claire M. Scott, Mervyn Thompson, Ron J. King, Michael S. Hadley
المصدر: ChemInform. 37
مصطلحات موضوعية: Intrinsic activity, Stereochemistry, medicine.drug_class, Clinical Biochemistry, Pharmaceutical Science, Serotonin 5-HT1 Receptor Antagonists, Ligands, Biochemistry, Structure-Activity Relationship, chemistry.chemical_compound, Drug Discovery, medicine, Animals, Humans, Selective receptor modulator, Receptor, Molecular Biology, 5-HT receptor, Organic Chemistry, Antagonist, General Medicine, Receptor antagonist, Rats, HYDIA, Piperazine, chemistry, Competitive antagonist, Microsomes, Liver, Molecular Medicine, Serotonin Antagonists, Selectivity