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المؤلفون: Brian T. Campbell, Arup K. Ghose, Helen Hua, Ronald R. Nepomuceno, Joyce James, Mark A. Ator, Brian Struss, Torsten Herbertz, Ruwanthi N. Gunawardane, Mark W. Holladay, Michael Williams, Darren E. Insko, Eduardo Setti, Susan Jones-Bolin, Ianina Valenta, Julius L. Apuy, Sunny Abraham, Martin W. Rowbottom, Michael F. Gardner, Robert C. Armstrong, Merryl D. Cramer, Michael Gibney, Lan Tran, Kelly G. Sprankle, Maiko Ezawa, Bruce D. Dorsey, Raffaella Faraoni, Dana Gitnick, Shripad Bhagwat, Qi Chao, Andiliy G. Lai, Bruce Ruggeri
المصدر: Journal of medicinal chemistry. 55(3)
مصطلحات موضوعية: MAPK/ERK pathway, Male, Models, Molecular, Proto-Oncogene Proteins B-raf, Transplantation, Heterologous, Administration, Oral, Mice, Nude, Pharmacology, Binding, Competitive, Rats, Sprague-Dawley, chemistry.chemical_compound, Mice, Structure-Activity Relationship, Dogs, Cell Line, Tumor, Drug Discovery, Quinazoline, Structure–activity relationship, Animals, Humans, Protein kinase A, Cell Proliferation, Cell growth, Phenylurea Compounds, Stereoisomerism, Isoxazoles, digestive system diseases, Rats, Transplantation, Macaca fascicularis, chemistry, Mutation, Cancer research, Microsomes, Liver, Quinazolines, Molecular Medicine, Female, Signal transduction, Drug Screening Assays, Antitumor, V600E, Neoplasm Transplantation