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1
المؤلفون: Laura Vidal, Miriam Andrés, Marta Mir, Pilar Forns, Sara Sevilla, Bernat Vidal, Estrella Lozoya, Cristina Esteve, Mónica Bravo, Manel Ferrer, Paul R. Eastwood, Richard S. Roberts, Jordi Castro, Elena Gómez, Marta Calbet, Pere Vilaseca, Jacob González, Imma Moreno, Silvia Petit, J. A. Alonso, Maria Antonia Buil
المصدر: Bioorganic & Medicinal Chemistry Letters. 24:5127-5133
مصطلحات موضوعية: Steric effects, endocrine system diseases, Stereochemistry, Receptors, Prostaglandin, Clinical Biochemistry, Substituent, Pharmaceutical Science, Acetates, Kinetic energy, Biochemistry, Dissociation (chemistry), Bridged Bicyclo Compounds, Structure-Activity Relationship, chemistry.chemical_compound, Drug Discovery, Humans, Receptors, Immunologic, Receptor, Crth2 antagonist, Molecular Biology, Bicyclic molecule, Hydrogen bond, Organic Chemistry, nutritional and metabolic diseases, Hydrogen Bonding, Models, Chemical, chemistry, Molecular Medicine, Half-Life
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2
المؤلفون: Cristina Esteve, Jacob González, Pere Vilaseca, Marta Calbet, Imma Moreno, Marta Mir, Richard S. Roberts, Silvia Petit, Elena Gómez, Mónica Bravo, Miriam Zanuy, J. A. Alonso, Manel Ferrer, Sara Sevilla, Laura Vidal, Peter Eichhorn, Miriam Andrés, Paul R. Eastwood, Bernat Vidal
المصدر: Bioorganic & Medicinal Chemistry Letters. 24:5123-5126
مصطلحات موضوعية: Indoles, Stereochemistry, Receptors, Prostaglandin, Clinical Biochemistry, Substituent, Pharmaceutical Science, Acetates, Biochemistry, Dissociation (chemistry), Bridged Bicyclo Compounds, Structure-Activity Relationship, chemistry.chemical_compound, Drug Discovery, Animals, Humans, Molecule, Rats, Wistar, Receptors, Immunologic, Crth2 antagonist, Molecular Biology, Bicyclic molecule, Chemistry, Organic Chemistry, Rats, Injections, Intravenous, Molecular Medicine, Half-Life
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3
المؤلفون: Richard S. Roberts, Maria Antonia Buil, Peter Eichhorn, Paul R. Eastwood, Imma Moreno, Silvia Petit, Pilar Forns, Jordi Castro, Oscar Casado, Manel Ferrer, Miriam Andrés, Marta Calbet
المصدر: Bioorganic & Medicinal Chemistry Letters. 24:5111-5117
مصطلحات موضوعية: Cell Membrane Permeability, Stereochemistry, Receptors, Prostaglandin, Clinical Biochemistry, Kinetics, Administration, Oral, Pharmaceutical Science, Acetates, Biochemistry, Structure-Activity Relationship, Piperidines, Drug Discovery, Low permeability, Animals, Humans, Receptors, Immunologic, Crth2 antagonist, Receptor, Molecular Biology, Chemistry, Organic Chemistry, Prodrug, Rats, Bioavailability, Pyrazoles, Molecular Medicine, Caco-2 Cells, Half-Life
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4
المؤلفون: Richard S. Roberts, Maria Antonia Buil, Manel Ferrer, Marcos Castillo, Miriam Andrés, Mónica Bravo, Martin D. Lehner, Jordi Castro, Sara Sevilla, Peter Eichhorn, Marta Calbet, Imma Moreno
المصدر: European Journal of Medicinal Chemistry. 71:168-184
مصطلحات موضوعية: Pharmacology, Stereochemistry, Receptors, Prostaglandin, Organic Chemistry, Biological activity, General Medicine, Acetates, Pyrazole, In vitro, Structure-Activity Relationship, Acetic acid, chemistry.chemical_compound, chemistry, Biochemistry, In vivo, Drug Discovery, Homologous chromosome, Humans, Pyrazoles, Structure–activity relationship, Molecule, Receptors, Immunologic
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5
المؤلفون: Jordi Serrat, Jordi Gràcia, Judit Cabedo, Lluís Pagès, Dolors Vilella, Martin D. Lehner, Manel Ferrer, Montserrat Miralpeix, Peter Eichhorn, Jordi Castro, Begoña Hernández, Maria Antonia Buil, Victor Segarra, Elena Calama, Sara Sevilla, Carla Carcasona, Miriam Andrés, Joan Taltavull, Imma Moreno, Richard S. Roberts, Amadeu Gavaldà
المصدر: Journal of medicinal chemistry. 59(23)
مصطلحات موضوعية: 0301 basic medicine, Male, Models, Molecular, Pharmacology, Adenylyl cyclase, Rats, Sprague-Dawley, 03 medical and health sciences, Cyclic nucleotide, chemistry.chemical_compound, Structure-Activity Relationship, Drug Discovery, Animals, Humans, chemistry.chemical_classification, Cyclic nucleotide phosphodiesterase, Dose-Response Relationship, Drug, Molecular Structure, Biphenyl Compounds, Adenosine receptor, Cyclic Nucleotide Phosphodiesterases, Type 4, Rats, Pyridazines, 030104 developmental biology, Enzyme, chemistry, Biochemistry, Structural biology, Second messenger system, Molecular Medicine, Phosphodiesterase 4 Inhibitors, Intracellular
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6Discovery of a novel class of zwitterionic, potent, selective and orally active S1P1 direct agonists
المؤلفون: Gema Tarrasón, Nuria Godessart, Marta Mir, Clara Armengol, Mònica Córdoba, Dolors Vilella, Daniel Casals, Manel López, Victor Segarra, Teresa Doménech, Imma Moreno, M Sabate, Nuria Aguilar, Pedro M. Grima, María Domínguez, Laia Esteban
المصدر: Bioorganic & Medicinal Chemistry Letters. 22:7672-7676
مصطلحات موضوعية: Chemistry, Organic Chemistry, Clinical Biochemistry, Rat model, Pharmaceutical Science, Biochemistry, Combinatorial chemistry, Receptor subtype, Orally active, In vivo, Drug Discovery, Molecular Medicine, Homology modeling, Molecular Biology, Structural class
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7
المؤلفون: Jordi Sanahuja, Montse Erra, Nuria Godessart, Raquel F. Reinoso, Estrella Lozoya, Imma Moreno, Pilar Pizcueta, Julio C. Castro-Palomino, Miriam Andrés
المصدر: Bioorganic & Medicinal Chemistry Letters. 21:7268-7272
مصطلحات موضوعية: Oxidoreductases Acting on CH-CH Group Donors, Toluidines, Stereochemistry, Clinical Biochemistry, Dihydroorotate Dehydrogenase, Hydroxybutyrates, Pharmaceutical Science, Biochemistry, Peripheral blood mononuclear cell, Structure-Activity Relationship, chemistry.chemical_compound, In vivo, Nitriles, Drug Discovery, Teriflunomide, Animals, Humans, Computer Simulation, Enzyme Inhibitors, Molecular Biology, Binding Sites, Chemistry, Biphenyl Compounds, Organic Chemistry, Arthritis, Experimental, Protein Structure, Tertiary, Rats, Crotonates, Drug Design, Dihydroorotate dehydrogenase, Molecular Medicine
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8
المؤلفون: Angel F. Remacha, M. Arilla, Imma Moreno, Neus Boto, Adelaida Ramos, Jorge Sierra, Rodrigo Martino, Concepción Pastoret, P Madoz, Clara Martínez, E Muniz-Diaz, C. Canals
المصدر: Transfusion. 44:1603-1611
مصطلحات موضوعية: medicine.medical_specialty, business.industry, Immunology, Pure red cell aplasia, Hematology, medicine.disease, Gastroenterology, Hemolysis, Transplantation, Red blood cell, medicine.anatomical_structure, Platelet transfusion, hemic and lymphatic diseases, ABO blood group system, Internal medicine, parasitic diseases, medicine, Immunology and Allergy, Transplantation Conditioning, Progenitor cell, business
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9
المؤلفون: Martin D. Lehner, Teresa Doménech, Imma Moreno, Elena Gómez, Jordi Castro, Maria Antonia Buil, Manel Ferrer, Miriam Andrés, Sara Sevilla, Marta Calbet, Mónica Bravo, Peter Eichhorn, Richard S. Roberts
المصدر: Bioorganicmedicinal chemistry letters. 23(11)
مصطلحات موضوعية: Stereochemistry, High-throughput screening, Clinical Biochemistry, Receptors, Prostaglandin, Pharmaceutical Science, Plasma protein binding, Pyrazole, Acetates, Biochemistry, chemistry.chemical_compound, Structure-Activity Relationship, Drug Discovery, Animals, Receptors, Immunologic, Receptor, Molecular Biology, Chemistry, Organic Chemistry, Antagonist, High-Throughput Screening Assays, Rats, Molecular Medicine, Pyrazoles, Prostaglandin D2, Half-Life, Protein Binding
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10Discovery of a novel class of zwitterionic, potent, selective and orally active S1P₁ direct agonists
المؤلفون: Nuria, Aguilar, Marta, Mir, Pedro M, Grima, Manel, López, Victor, Segarra, Laia, Esteban, Imma, Moreno, Nuria, Godessart, Gema, Tarrasón, Teresa, Domenech, Dolors, Vilella, Clara, Armengol, Mònica, Córdoba, Mar, Sabaté, Daniel, Casals, Maria, Domínguez
المصدر: Bioorganicmedicinal chemistry letters. 22(24)
مصطلحات موضوعية: Models, Molecular, Encephalomyelitis, Autoimmune, Experimental, Dose-Response Relationship, Drug, Molecular Structure, Administration, Oral, Crystallography, X-Ray, Rats, Disease Models, Animal, Receptors, Lysosphingolipid, Structure-Activity Relationship, Lymphopenia, Drug Discovery, Thiadiazoles, Animals, Sphingosine-1-Phosphate Receptors