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1
المؤلفون: Matthew Jude Sharp, Will L. Canoy, Kae M. Bullock, Eric Eugene Boros, Xiao-ming M. Zhou, Richard T. Matsuoka, Greg A. Erickson, Vassil I. Elitzin, Mark B. Mitchell, Matthew C. Salmon, David H. Igo, Nicole M. Deschamps, Daniel W. Reynolds, Andrew D. Brown, Gregory E. Peckham, Istvan Kaldor, Jennifer F. Toczko, Shannon Condon, Carpenter Andrew J, Elie Amine Tabet, Jing M. Fang, Biren K. Joshi, Lianming Michael Wu, Jeremy D. Cobb
المصدر: Organic Process Research & Development. 20:1469-1475
مصطلحات موضوعية: 0301 basic medicine, 03 medical and health sciences, 030104 developmental biology, 0302 clinical medicine, GPR119, Chemistry, 030220 oncology & carcinogenesis, Organic Chemistry, Physical and Theoretical Chemistry, Receptor, Combinatorial chemistry
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2
المؤلفون: Eric E. Boros, Istvan Kaldor
المصدر: Journal of Heterocyclic Chemistry. 52:302-305
مصطلحات موضوعية: chemistry.chemical_compound, chemistry, Organic Chemistry, Thermal, Organic chemistry, Tributylamine, Isocyanate
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3
المصدر: Journal of Heterocyclic Chemistry. 50:863-867
مصطلحات موضوعية: chemistry.chemical_classification, Base (chemistry), Imidazolidinone, Organic Chemistry, Regioselectivity, 2-imidazolidinone, Medicinal chemistry, Hydroxyethyl Urea, chemistry.chemical_compound, chemistry, Yield (chemistry), Alkali carbonate, Urea, Organic chemistry
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4
المؤلفون: Eric E. Boros, Robert L. Dobbins, Maggie S. McIntyre, Ryan Klein, David J. Cowan, Xi Liang, Xiaozhou Yao, Andrew A. Young, Kristin M. Patterson, Paul L. Feldman, John Ray, Christine L. Merrill, Lindsey T. Harston, Jeff L. Ambroso, Jon L. Collins, Shane Roller, Michael J. Bishop, Judith S. Prescott, Christopher Joseph Aquino, Alan Cunningham, Don L. Anderson, Istvan Kaldor, Wu Yulin, Lihong Chen, Josephine Yuen
المصدر: Journal of Medicinal Chemistry. 56:5094-5114
مصطلحات موضوعية: Male, Thiazepines, Portal vein, Hepatic cholesterol, Organic Anion Transporters, Sodium-Dependent, Type 2 diabetes, Pharmacology, Bile Acids and Salts, Methylamines, Mice, Dogs, Animal model, Drug Stability, Clinical investigation, Drug Discovery, medicine, Animals, Humans, Hypoglycemic Agents, Bile acid transporter, Symporters, Chemistry, Apical sodium-dependent bile acid transporter, Metabolism, medicine.disease, Rats, HEK293 Cells, Diabetes Mellitus, Type 2, Solubility, Molecular Medicine
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5
المؤلفون: Christie Schulte, Curt D. Haffner, J. Chuck Poole, Eric E. Boros, John C. Ulrich, David J. Cowan, Tiffany Carpenter, Eugene L. Stewart, J. Darren Stuart, Frank Preugschat, David N. Deaton, Tara Renae Rheault, Todd W. Shearer, Barry G. Shearer, J. David Becherer, Michael R. Jeune, Istvan Kaldor, Lisa M. Shewchuk, Terrence L. Smalley
المصدر: Journal of medicinal chemistry. 58(17)
مصطلحات موضوعية: Models, Molecular, medicine.drug_class, Protein Conformation, Biological Availability, Carboxamide, CD38, Pharmacology, Crystallography, X-Ray, Permeability, chemistry.chemical_compound, Structure-Activity Relationship, In vivo, Drug Discovery, Hydrolase, medicine, Structure–activity relationship, Animals, Humans, Obesity, Muscle, Skeletal, chemistry.chemical_classification, Hydrolysis, Quinoline, Membranes, Artificial, Stereoisomerism, NAD, ADP-ribosyl Cyclase 1, Amides, Mice, Inbred C57BL, Enzyme, chemistry, Biochemistry, Liver, Aminoquinolines, Quinolines, Molecular Medicine, NAD+ kinase
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6
المؤلفون: Eric E. Boros, Philip Stewart Turnbull, Istvan Kaldor
المصدر: Journal of Heterocyclic Chemistry. 48:733-736
مصطلحات موضوعية: Indole test, chemistry.chemical_compound, Trifluoromethyl, chemistry, Yield (chemistry), Organic Chemistry, Convergent synthesis, Phenol, Organic chemistry, Cyanation, Trifluoromethanesulfonate
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7
المؤلفون: Lihong Chen, Jonathan Y. Bass, David N. Deaton, Aaron B. Miller, Justin A. Caravella, Istvan Kaldor, Robert B. McFadyen, Stacey A. Jones, Dan Todd, Paul Kenneth Spearing, Kevin P. Madauss, Adwoa Akwabi-Ameyaw, Derek J. Parks, Richard Dana Caldwell, Frank Navas, Yaping Liu, Katrina L. Creech, G. Bruce Wisely, Harry B. Marr, Shawn P. Williams
المصدر: Bioorganic & Medicinal Chemistry Letters. 18:4339-4343
مصطلحات موضوعية: Agonist, Molecular model, medicine.drug_class, Stereochemistry, Clinical Biochemistry, Carboxylic Acids, Molecular Conformation, Administration, Oral, Receptors, Cytoplasmic and Nuclear, Pharmaceutical Science, Naphthalenes, Crystallography, X-Ray, Biochemistry, Chemical synthesis, Mice, Structure-Activity Relationship, Dogs, Drug Discovery, medicine, Animals, Structure–activity relationship, Receptor, Molecular Biology, Cholestasis, Molecular Structure, Chemistry, Stomach, Organic Chemistry, Haplorhini, Isoxazoles, G protein-coupled bile acid receptor, Rats, DNA-Binding Proteins, Disease Models, Animal, Nuclear receptor, Gastric Mucosa, Molecular Medicine, Farnesoid X receptor, Transcription Factors
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8
المؤلفون: Eric E. Boros, Istvan Kaldor
المصدر: ChemInform. 46
مصطلحات موضوعية: chemistry.chemical_compound, Chemistry, Polymer chemistry, Thermal, General Medicine, Tributylamine
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9
المؤلفون: John C. Ulrich, Petrov Kimberly, Tiffany Carpenter, David J. Cowan, J. Darren Stuart, J. David Becherer, Eugene L. Stewart, Frank Preugschat, David N. Deaton, W. Wallace Harrington, Yu Guo, Naphtali Milliken, Barry G. Shearer, Michael R. Jeune, Istvan Kaldor, Terrence L. Smalley, Curt D. Haffner, Brad R. Henke, Rodolfo Cadilla, Todd W. Shearer, Eric E. Boros, Christie Schulte
المصدر: Journal of medicinal chemistry. 58(8)
مصطلحات موضوعية: Muscle tissue, Pharmacology, CD38, Quinolones, Cell Line, Dogs, Pharmacokinetics, Drug Discovery, medicine, Animals, Humans, Obesity, Chemistry, Drug discovery, Muscles, NAD, Small molecule, ADP-ribosyl Cyclase 1, Mice, Inbred C57BL, Molecular Docking Simulation, Thiazoles, medicine.anatomical_structure, Biochemistry, Liver, Cell culture, Molecular Medicine, NAD+ kinase, Diet-induced obese
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10
المؤلفون: Istvan Kaldor, Boggs Sharon Davis, David N. Deaton, Katrina L. Creech, Lihong Chen, Justin A. Caravella, Terrence L. Smalley, Derek J. Parks
المصدر: Bioorganicmedicinal chemistry letters. 25(2)
مصطلحات موضوعية: Agonist, Models, Molecular, Activity profile, Molecular Structure, medicine.drug_class, Chemistry, Organic Chemistry, Clinical Biochemistry, Drug Evaluation, Preclinical, Pharmaceutical Science, Receptors, Cytoplasmic and Nuclear, Isoxazoles, Pharmacology, Biochemistry, Farnesoid X Receptor Agonists, Structure-Activity Relationship, Drug Discovery, medicine, Fluorescence Resonance Energy Transfer, Molecular Medicine, Humans, Farnesoid X receptor, Molecular Biology, Oxazolidinones