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المؤلفون: Eric Goffin, Pierre Fraikin, Dayana Abboud, Pascal de Tullio, Caroline Beaufour, Iuliana Botez, Julien Hanson, Laurence Danober, Pierre Francotte, Bernard Pirotte
مصطلحات موضوعية: Pharmacology, Organic Chemistry, Drug Discovery, General Medicine
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::2dbce7893b489005fcc0c403b43869b6
https://doi.org/10.2139/ssrn.4329581 -
2
المؤلفون: Jerzy Dorosz, Thomas Colson, Jean-Yves Thomas, Pierre Francotte, Jette S. Kastrup, Laurence Danober, Iuliana Botez Pop, Koffi Senam Etse, Eric Goffin, Katrine McLain Christensen, Bernard Pirotte, Pierre Lestage
المصدر: ACS Chemical Neuroscience. 12:2679-2692
مصطلحات موضوعية: Physiology, Stereochemistry, Chemistry, Cognitive Neuroscience, Dimer, Allosteric regulation, Stereoisomerism, Cell Biology, General Medicine, AMPA receptor, Benzothiadiazines, Crystallography, X-Ray, Biochemistry, Cocrystal, In vitro, chemistry.chemical_compound, Allosteric Regulation, In vivo, Benzothiadiazine, Receptors, AMPA, Enantiomer, alpha-Amino-3-hydroxy-5-methyl-4-isoxazolepropionic Acid
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3دورية أكاديمية
المؤلفون: Rosse Marie ESPARZA-HUAMANCHUMO, Iuliana BOTEZAN, Rodrigo SANCHEZ-JIMENEZ, Klinge Orlando VILLALBA-CONDORI
المصدر: Geo Journal of Tourism and Geosites, Vol 54, Iss 2 supplement, Pp 953-966 (2024)
مصطلحات موضوعية: ecotourism, sustainable tourism, nature based tourism, bibliometric analysis, science mapping, Geography. Anthropology. Recreation, Geography (General), G1-922
وصف الملف: electronic resource
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المؤلفون: Vassili Prudhomme, Mélissa Cucca, Lionel Nauton, Elsa Andrieu, Mathilde Fereyrolles, Sylvain Lamoine, Clément Michelin, Khalil Bennis, Aurore Collin, Frédéric De Ceuninck, Iuliana Botez, Christophe Mallet, Sylvie Ducki
المساهمون: Institut de Chimie de Clermont-Ferrand (ICCF), Institut de Chimie du CNRS (INC)-Centre National de la Recherche Scientifique (CNRS)-Université Clermont Auvergne (UCA)-Institut national polytechnique Clermont Auvergne (INP Clermont Auvergne), Université Clermont Auvergne (UCA)-Université Clermont Auvergne (UCA), ANR-16-IDEX-0001,CAP 20-25,CAP 20-25(2016)
المصدر: European Journal of Medicinal Chemistry
European Journal of Medicinal Chemistry, 2022, 244, pp.114809. ⟨10.1016/j.ejmech.2022.114809⟩مصطلحات موضوعية: E7010, Pharmacology, History, Vascular-disrupting agents (VDA), Indoles, Polymers and Plastics, Organic Chemistry, Inhibition of tubulin assembly (ITA), Antineoplastic Agents, Angiogenesis Inhibitors, General Medicine, Industrial and Manufacturing Engineering, Tubulin Modulators, Tubulin, Cell Line, Tumor, Drug Discovery, [CHIM]Chemical Sciences, Business and International Management
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5دورية أكاديمية
لا يتم عرض هذه النتيجة على الضيوف.
تسجيل الدخول للوصول الكامل. -
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المؤلفون: Jette S. Kastrup, Bernard Pirotte, Lars Olsen, Pierre Lestage, Ann-Beth Nørholm, Eric Goffin, Laurence Danober, Chris Oostenbrink, Pierre Francotte, Iuliana Botez
المصدر: Journal of Chemical Information and Modeling. 54:3404-3416
مصطلحات موضوعية: Chemistry, Entropy, General Chemical Engineering, Enthalpy, Allosteric regulation, Thermodynamic integration, Isothermal titration calorimetry, General Chemistry, Plasma protein binding, Molecular Dynamics Simulation, Library and Information Sciences, Benzothiadiazines, Ligands, Protein Structure, Tertiary, Computer Science Applications, Molecular dynamics, Protein structure, Allosteric Regulation, Computational chemistry, Ionotropic glutamate receptor, Receptors, AMPA, Protein Binding
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المؤلفون: Pascal De Tullio, Pierre Fraikin, Fabrice Iop, Ann-Beth Nørholm, Taru Deva, Karla Frydenvang, Jean-Yves Thomas, Lars Olsen, Sylvie Challal, Caroline Louis, Bernard Pirotte, Pierre Lestage, Pierre Francotte, Iuliana Botez-Pop, Laurence Danober, Jette S. Kastrup, Eric Goffin
المصدر: Journal of Medicinal Chemistry. 57:9539-9553
مصطلحات موضوعية: chemistry.chemical_compound, chemistry, In vivo, Benzothiadiazine, Stereochemistry, Drug Discovery, Allosteric regulation, Molecular Medicine, Isothermal titration calorimetry, AMPA receptor, Potentiator, Receptor, Compound 32
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8
المؤلفون: Pierre Lestage, Ann-Beth Nørholm, Iuliana Botez-Pop, Sylvie Challal, Bernard Pirotte, Karla Frydenvang, Laurence Danober, Christian Krintel, Pierre Francotte, Eric Goffin, Jette S. Kastrup, Lars Olsen
المصدر: Journal of Medicinal Chemistry. 56:8736-8745
مصطلحات موضوعية: Models, Molecular, Allosteric modulator, Stereochemistry, Dimer, Allosteric regulation, Calorimetry, Benzothiadiazines, Crystallography, X-Ray, Structure-Activity Relationship, chemistry.chemical_compound, Allosteric Regulation, Drug Discovery, Animals, Structure–activity relationship, Receptors, AMPA, Neurons, Dose-Response Relationship, Drug, Molecular Structure, biology, Chemistry, Isothermal titration calorimetry, Cyclic S-Oxides, Rats, Allosteric enzyme, Benzothiadiazine, biology.protein, Thermodynamics, Molecular Medicine, Ionotropic effect
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9
المؤلفون: P. Lestage, B. Lesur, L. Danober, P. de Tullio, Pierre Francotte, Iuliana Botez, Bernard Pirotte, Eric Goffin, Pierre Fraikin, Daniel-Henri Caignard
المصدر: Current Medicinal Chemistry. 17:3575-3582
مصطلحات موضوعية: Pharmacology, Thiadiazines, Organic Chemistry, Allosteric regulation, Glutamate receptor, Long-term potentiation, AMPA receptor, Biology, Potentiator, Biochemistry, Glutamatergic, Allosteric Regulation, nervous system, Drug Discovery, Humans, Molecular Medicine, Receptors, AMPA, Nervous System Diseases, Receptor, Neuroscience, Ionotropic effect
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::2c92e8ae1e4c846c4fd6bd27d1f0ed0e
https://doi.org/10.2174/092986710792927859 -
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المؤلفون: Pierre, Francotte, Ann-Beth, Nørholm, Taru, Deva, Lars, Olsen, Karla, Frydenvang, Eric, Goffin, Pierre, Fraikin, Pascal, de Tullio, Sylvie, Challal, Jean-Yves, Thomas, Fabrice, Iop, Caroline, Louis, Iuliana, Botez-Pop, Pierre, Lestage, Laurence, Danober, Jette S, Kastrup, Bernard, Pirotte
المصدر: Journal of medicinal chemistry. 57(22)
مصطلحات موضوعية: Thiadiazines, Chemistry, Pharmaceutical, Temperature, Oxides, Calorimetry, Benzothiadiazines, Crystallography, X-Ray, Hippocampus, Cyclic S-Oxides, Rats, Electrophysiology, Kinetics, Mice, Drug Design, Animals, Humans, Thermodynamics, Receptors, AMPA, Propionates, Rats, Wistar, Dimerization, Allosteric Site, Hydrogen, Protein Binding