-
1
المؤلفون: Ivo Vranesic, Peter Ertl, Manuel Koller, Grit Laue, Dirk Behnke, David Orain, Sandrine Desrayaud, David Carcache
المصدر: Bioorganic & Medicinal Chemistry Letters. 22:6454-6459
مصطلحات موضوعية: Pyridones, Stereochemistry, Metabotropic glutamate receptor 5, Chemistry, Receptor, Metabotropic Glutamate 5, Organic Chemistry, Clinical Biochemistry, Allosteric regulation, Pharmaceutical Science, Receptors, Metabotropic Glutamate, Amides, Biochemistry, Inhibitory Concentration 50, chemistry.chemical_compound, Allosteric Regulation, Solubility, Drug Discovery, Aqueous solubility, Pyridine, Humans, Molecular Medicine, Pyrroles, Metabotropic glutamate receptor 2, Molecular Biology
-
2
المؤلفون: Ivo Vranesic, Markus Fendt, Ralf Glatthar, Troxler Thomas J, David Orain, Carsten Spanka, Sandrine Desrayaud
المصدر: Bioorganic & Medicinal Chemistry Letters. 20:184-188
مصطلحات موضوعية: medicine.drug_class, Receptor, Metabotropic Glutamate 5, Clinical Biochemistry, Administration, Oral, Aminopyridines, Pharmaceutical Science, Carboxamide, Pharmacology, Receptors, Metabotropic Glutamate, Biochemistry, Rats, Sprague-Dawley, Structure-Activity Relationship, chemistry.chemical_compound, Drug Discovery, medicine, Animals, Humans, Structure–activity relationship, Receptor, Molecular Biology, Nicotinamide, Metabotropic glutamate receptor 5, Organic Chemistry, Antagonist, Amides, Rats, Metabotropic receptor, Anti-Anxiety Agents, chemistry, Metabotropic glutamate receptor, Microsomes, Liver, Molecular Medicine, Peptides
-
3
المؤلفون: Stephan Urwyler, Samuel Hintermann, Daniel Hoyer, Thomas Moenius, Steven Whitebread, Michel Lemaire, Ivo Vranesic, Hans Allgeier, Armin Brülisauer, Yves Auberson, Fabrizio Gasparini
المصدر: Bioorganic & Medicinal Chemistry. 15:903-914
مصطلحات موضوعية: Male, Biodistribution, Chemical Phenomena, Pyridines, Clinical Biochemistry, Pharmaceutical Science, In Vitro Techniques, Ligands, Phosphatidylinositols, Binding, Competitive, Biochemistry, Mass Spectrometry, Cell Line, Rats, Sprague-Dawley, Receptors, Kainic Acid, Pharmacokinetics, Cricetinae, Mglu5 receptors, Oximes, Drug Discovery, Excitatory Amino Acid Agonists, Animals, Humans, Tissue Distribution, Rats, Wistar, Receptor, Molecular Biology, Chemistry, Physical, Chemistry, Metabotropic glutamate receptor 5, Organic Chemistry, Quisqualic Acid, Blood Proteins, Rats, In vitro pharmacology, Metabotropic glutamate receptor, Positron-Emission Tomography, Injections, Intravenous, Microsomes, Liver, Autoradiography, Molecular Medicine, Indicators and Reagents, Radiopharmaceuticals, Preclinical imaging, Protein Binding
-
4
المؤلفون: M. Maj, Zorica Dragic, Fabrizio Gasparini, Rainer Kuhn, Peter J. Flor, Valeria Bruno, T. Stein, Giuseppe Battaglia, Ivo Vranesic, R. Yamamoto, F. Nicoletti, Werner Inderbitzin, Natacha Stoehr
المصدر: Neuropharmacology. 45:895-906
مصطلحات موضوعية: Agonist, N-Methylaspartate, Allosteric modulator, medicine.drug_class, Excitatory Amino Acids, Pharmacology, Biology, Receptors, Metabotropic Glutamate, Neuroprotection, Cell Line, Cellular and Molecular Neuroscience, Cyclic AMP, Excitatory Amino Acid Agonists, medicine, Humans, Benzopyrans, Cloning, Molecular, Cerebral Cortex, Neurons, Amyloid beta-Peptides, Dose-Response Relationship, Drug, Cell Membrane, Antagonist, Neuroprotective Agents, Metabotropic receptor, Guanosine 5'-O-(3-Thiotriphosphate), Metabotropic glutamate receptor, Metabotropic glutamate receptor 1, Calcium, Metabotropic glutamate receptor 2, Neuroglia
-
5
المؤلفون: Will P.J.M Spooren, Andrzej Pilc, Ivo Vranesic, Natacha Stoehr, Peter J. Flor, Kurt Lingenhöhl, Annick Vassout, Adriana Pagano, Fabrizio Gasparini, Rainer Kuhn, Conrad Gentsch
المصدر: Amino Acids. 23:207-211
مصطلحات موضوعية: Binding Sites, Allosteric modulator, Pyridines, Metabotropic glutamate receptor 5, Chemistry, Receptor, Metabotropic Glutamate 5, Metabotropic glutamate receptor 4, Organic Chemistry, Clinical Biochemistry, Metabotropic glutamate receptor 7, Brain, Pain, Class C GPCR, Anxiety, Pharmacology, Ligands, Receptors, Metabotropic Glutamate, Biochemistry, Anti-Anxiety Agents, Metabotropic glutamate receptor, Animals, Metabotropic glutamate receptor 1, Metabotropic glutamate receptor 2, Excitatory Amino Acid Antagonists
-
6
المؤلفون: Ivo Vranesic, Kevin H. McAllister, Peter J. Flor, Fabrizio Gasparini, Rainer Kuhn, Albert Enz, Sandrine Desrayaud, Graeme Bilbe, Silvio Ofner, Rochdi Bouhelal
المصدر: Bioorganicmedicinal chemistry. 22(21)
مصطلحات موضوعية: Male, Dyskinesia, Drug-Induced, Indoles, medicine.drug_class, Pyridines, Receptor, Metabotropic Glutamate 5, Clinical Biochemistry, Pharmaceutical Science, Pharmacology, Biochemistry, Levodopa, Rats, Sprague-Dawley, chemistry.chemical_compound, Mice, Structure-Activity Relationship, In vivo, mental disorders, Drug Discovery, medicine, Mavoglurant, Animals, Humans, Receptor, Molecular Biology, IC50, Metabotropic glutamate receptor 5, Organic Chemistry, Antagonist, Brain, Hyperthermia, Induced, Receptor antagonist, High-Throughput Screening Assays, Rats, chemistry, Metabotropic glutamate receptor, Molecular Medicine, Half-Life, Protein Binding
-
7
المؤلفون: Ivo Vranesic, Markus Fendt, Silvio Ofner, Kaspar Zimmermann, Ralf Glatthar, Grit Laue, Daniel Peterlik, Klemens Kaupmann, Dominik Feuerbach, Christine E. Gee, Rochdi Bouhelal, Peter J. Flor, Herman van der Putten, Christoph Neuhäuser, Nicole Uschold-Schmidt, John F. Cryan
المصدر: The Journal of biological chemistry. 289(16)
مصطلحات موضوعية: Agonist, medicine.drug_class, Long-Term Potentiation, CHO Cells, Biology, Anxiety, Receptors, Metabotropic Glutamate, Biochemistry, Amygdala, Mice, Cricetulus, L Cells, Neurobiology, Cricetinae, medicine, Animals, Fear conditioning, Molecular Biology, Behavior, Animal, Metabotropic glutamate receptor 7, Metabotropic glutamate receptor 6, Long-term potentiation, Cell Biology, Mice, Mutant Strains, Protein Structure, Tertiary, medicine.anatomical_structure, Metabotropic glutamate receptor, Metabotropic glutamate receptor 1, Neuroscience, Stress, Psychological
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::35d470b156affce7a8cb2c77a1868896
https://pubmed.ncbi.nlm.nih.gov/24596089 -
8
المؤلفون: Christine Stierlin, Peter J. Flor, Werner Inderbitzin, Natacha Stoehr, Fabrizio Gasparini, David Ott, Rainer Kuhn, Philipp Floersheim, Micheline Heinrich, Adriana Pagano, Ivo Vranesic
المصدر: Il Farmaco. 56:95-99
مصطلحات موضوعية: Models, Molecular, Binding Sites, Stereochemistry, Chemistry, Glutamate receptor, Pharmaceutical Science, Receptors, Metabotropic Glutamate, Metabotropic receptor, Non-competitive inhibition, Mechanism of action, Biochemistry, Docking (molecular), Metabotropic glutamate receptor, mental disorders, Drug Discovery, medicine, medicine.symptom, Binding site, Receptor
-
9
المؤلفون: Adam Kesingland, Natacha Stoehr, Katharine Walker, Adriana Pagano, Will P.J.M Spooren, Fabrizio Gasparini, Clive Gentry, Andrew J. Davis, Kurt Lingenhoehl, Mark A. Varney, Rainer Kuhn, Ivo Vranesic, Edwin C. Johnson, Moh Panesar, Laszlo Urban, M Bowes, Peter J. Flor
المصدر: Neuropharmacology. 40:1-9
مصطلحات موضوعية: Pharmacology, medicine.medical_specialty, business.industry, Analgesic, Chronic pain, Glutamate receptor, medicine.disease, Cellular and Molecular Neuroscience, Metabotropic receptor, Endocrinology, Metabotropic glutamate receptor, Internal medicine, mental disorders, Neuropathic pain, medicine, Noxious stimulus, business, Ionotropic effect
-
10
المؤلفون: Peter J. Flor, Ivo Vranesic, Roberto Pellicciari, Gabriele Costantino, Fabrizio Gasparini, Rainer Kuhn, Laura Amori, Maura Marinozzi
المصدر: Bioorganic & Medicinal Chemistry Letters. 10:1447-1450
مصطلحات موضوعية: Agonist, Molecular model, Stereochemistry, medicine.drug_class, Carboxylic acid, Clinical Biochemistry, Pharmaceutical Science, CHO Cells, Cyclopentanes, Receptors, Metabotropic Glutamate, Biochemistry, chemistry.chemical_compound, Cricetinae, Drug Discovery, Excitatory Amino Acid Agonists, medicine, Animals, Humans, Cyclopentene, Receptor, Molecular Biology, chemistry.chemical_classification, Molecular Structure, Colforsin, Organic Chemistry, HYDIA, chemistry, Metabotropic glutamate receptor, Molecular Medicine, Biological Assay, Pharmacophore