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المؤلفون: Molly A. McGlynn, Matthew Frank Brown, Stacie P. O'Sullivan, Anthony Marfat, John B. Cheng, Theodore E. Liston, John W. Watson, J.S. Pillar, David B. Damon, J.T. Shirley, R. J. Chambers, Gerard Antognoli, Brian S. Owens
المصدر: Bioorganic & Medicinal Chemistry Letters. 8:2451-2456
مصطلحات موضوعية: Indoles, Leukotriene D4, Stereochemistry, Guinea Pigs, Clinical Biochemistry, Phenylcarbamates, Pharmaceutical Science, Biochemistry, Chemical synthesis, Tosyl Compounds, chemistry.chemical_compound, Drug Discovery, medicine, Animals, Humans, Potency, Zafirlukast, Imide, Receptor, Molecular Biology, Receptors, Leukotriene, Indole test, Sulfonamides, Chemistry, Organic Chemistry, Antagonist, Membrane Proteins, Haplorhini, respiratory system, Rats, Models, Chemical, Leukotriene Antagonists, Molecular Medicine, lipids (amino acids, peptides, and proteins), medicine.drug
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المصدر: Journal of Biological Chemistry. 273:15559-15564
مصطلحات موضوعية: Phosphodiesterase Inhibitors, Molecular Sequence Data, Allosteric regulation, Biology, Biochemistry, Isozyme, Catalysis, Mice, chemistry.chemical_compound, FLAG-tag, 3',5'-Cyclic-GMP Phosphodiesterases, Cyclic AMP, Animals, Humans, Tissue Distribution, Amino Acid Sequence, Cloning, Molecular, Cyclic GMP, Molecular Biology, chemistry.chemical_classification, Binding Sites, Base Sequence, Sequence Homology, Amino Acid, C-terminus, Phosphodiesterase, Cell Biology, Molecular biology, Amino acid, Kinetics, Enzyme, chemistry, Zaprinast, Sequence Alignment
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::815b48beb6a6c2a476da7e68bb28cba3
https://doi.org/10.1074/jbc.273.25.15559 -
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المؤلفون: Peter F. Moore, A. Nagahisa, Saul B. Kadin, Francis J. Sweeney, Thomas J. Carty, P. P. Pazoles, M. J. Ernest, J. D. Cheng, J.S. Pillar, Leland D. Loose, P. A. Joseph, R. J. Griffiths, S. Murase, James D. Eskra
المصدر: Inflammation Research. 46:168-179
مصطلحات موضوعية: Erythrocytes, Indoles, Neutrophils, Intracellular pH, Immunology, Radioimmunoassay, 6-Ketoprostaglandin F1 alpha, Leukotriene B4, Neutrophil Activation, Cyclooxygenase pathway, Immunoenzyme Techniques, Rats, Sprague-Dawley, chemistry.chemical_compound, In vivo, Hydroxyeicosatetraenoic Acids, medicine, Animals, Humans, Cyclooxygenase Inhibitors, Lipoxygenase Inhibitors, Calcimycin, Chromatography, High Pressure Liquid, Leukotriene E4, Pharmacology, Leukotriene, Arachidonate 5-Lipoxygenase, Arachidonic Acid, Chemotactic Factors, Ionophores, biology, Chemistry, Anti-Inflammatory Agents, Non-Steroidal, Zymosan, Oxindoles, Rats, Thromboxane B2, Cytosol, Leukemia, Basophilic, Acute, Biochemistry, Arachidonate 5-lipoxygenase, biology.protein, Arachidonic acid, Rabbits, Tenidap, medicine.drug
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المؤلفون: G.W. Antognoli, J.T. Shirley, A. Marfat, C.F. Wright, Thomas J. Carty, Frank W. Rusek, J. W. Watson, J. Delehunt, B. A. Naclerio, James F. Eggler, J.S. Pillar, Herbert Sherman, E.G. Andrews, Francis J. Sweeney, K. W. Freiert, R. Breslow, C. J. Mularski, V. L. Cohan, C J Pazoles, Lawrence S. Melvin, L.A. Rappach, John B. Cheng, David B. Damon, Jeanene E. Tickner, Judith L. Collins, P. Reiche, Hiroko Masamune, M. P. Carta, James D. Eskra, Hada William Andrew, R. J. Chambers
المصدر: Bioorganic & Medicinal Chemistry Letters. 5:1365-1370
مصطلحات موضوعية: LTD4 receptor, Chemistry, Organic Chemistry, Clinical Biochemistry, Drug Discovery, Antagonist, Pharmaceutical Science, Molecular Medicine, Pharmacology, Receptor, Molecular Biology, Biochemistry, First generation
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المؤلفون: Hiroko Masamune, J.T. Shirley, A. Marfat, John B. Cheng, Henry J. Showell, James F. Eggler, J.S. Pillar, Maryrose J. Conklyn, Jeanene E. Tickner, Lawrence S. Melvin, R. Breslow
المصدر: Bioorganic & Medicinal Chemistry Letters. 5:887-892
مصطلحات موضوعية: chemistry.chemical_compound, Chemistry, Organic Chemistry, Clinical Biochemistry, Drug Discovery, Quinoline, Pharmaceutical Science, Molecular Medicine, Pharmacology, Molecular Biology, Biochemistry, Combinatorial chemistry, In vitro
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المؤلفون: Kelvin Cooper, M. Zdankiewicz, James F. Eggler, J.S. Pillar, John B. Cheng, L. M. Hanak
المصدر: Journal of Labelled Compounds and Radiopharmaceuticals. 34:1147-1156
مصطلحات موضوعية: chemistry.chemical_classification, biology, Chemistry, Ligand binding assay, Organic Chemistry, Radiosynthesis, Biochemistry, eye diseases, In vitro, Analytical Chemistry, Enzyme, Enzyme inhibitor, Drug Discovery, Arachidonate 5-lipoxygenase, biology.protein, Radioligand, Radiology, Nuclear Medicine and imaging, 5-lipoxygenase-activating protein, Spectroscopy
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المؤلفون: John W. Watson, Anthony Marfat, John B. Cheng, J.T. Shirley, R. J. Chambers, G.W. Antognoli, J.S. Pillar
المصدر: ChemInform. 29
مصطلحات موضوعية: chemistry.chemical_compound, Leukotriene D4, chemistry, medicine, Potency, lipids (amino acids, peptides, and proteins), General Medicine, respiratory system, Zafirlukast, Pharmacology, Pranlukast, medicine.drug
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المؤلفون: T.C. Liston, Anthony Marfat, G.W. Antognoli, John B. Cheng, J.S. Pillar, Alexander V. Kuperman, J.T. Shirley, R. J. Chambers, Brian S. Owens, John W. Watson
المصدر: ChemInform. 30
مصطلحات موضوعية: Chemistry, medicine, General Medicine, Zafirlukast, Pharmacology, Receptor, Pranlukast, medicine.drug, Cyslt1 receptor
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المؤلفون: G.W. Antognoli, C. Mebus, T.C. Liston, David B. Damon, R. J. Chambers, J. W. Watson, J.T. Shirley, A. Marfat, John B. Cheng, J.S. Pillar, Alexander V. Kuperman
المصدر: Bioorganicmedicinal chemistry letters. 9(18)
مصطلحات موضوعية: Clinical Biochemistry, Guinea Pigs, Pharmaceutical Science, Biological Availability, Pharmacology, Biochemistry, Pranlukast, Pharmacokinetics, In vivo, Oral administration, Drug Discovery, medicine, Animals, Benzopyrans, Zafirlukast, Receptor, Molecular Biology, Receptors, Leukotriene, Leukotriene, Sulfonamides, Chemistry, Organic Chemistry, Membrane Proteins, Haplorhini, Rats, Liver, Drug Design, Toxicity, Molecular Medicine, Leukotriene Antagonists, medicine.drug, Half-Life
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المؤلفون: R. J. Chambers, Brian S. Owens, G.W. Antognoli, T.C. Liston, J.S. Pillar, Anthony Marfat, J.T. Shirley, John B. Cheng, Alexander V. Kuperman, John W. Watson
المصدر: Bioorganicmedicinal chemistry letters. 8(24)
مصطلحات موضوعية: Leukotriene D4, Magnetic Resonance Spectroscopy, Clinical Biochemistry, Guinea Pigs, Pharmaceutical Science, Biological Availability, Pharmacology, Biochemistry, Pranlukast, Cyslt1 receptor, chemistry.chemical_compound, In vivo, Drug Discovery, medicine, Animals, Humans, Anti-Asthmatic Agents, Zafirlukast, Receptor, Molecular Biology, Receptors, Leukotriene, Leukotriene, Chemistry, Organic Chemistry, Antagonist, Membrane Proteins, Stereoisomerism, U937 Cells, Rats, Thiazoles, Quinolines, Molecular Medicine, Leukotriene Antagonists, medicine.drug