يعرض 1 - 10 نتائج من 14 نتيجة بحث عن '"JM Lacoste"', وقت الاستعلام: 1.56s تنقيح النتائج
  1. 1
    The antagonist properties of S 11978 on 5HT3receptors in N1E-115 neuroblastoma cells

    المؤلفون: M. Laubie, C. Malen, JM Lacoste, E. Giesen-Crouse, C. Abraham, P. Morain

    المصدر: Fundamental & Clinical Pharmacology. 7:205-208

    مصطلحات موضوعية: medicine.medical_specialty, Indoles, Tropisetron, Thiophenes, Biology, Tritium, Binding, Competitive, Mice, Neuroblastoma, Internal medicine, Tumor Cells, Cultured, medicine, Animals, Pharmacology (medical), Patch clamp, Receptor, Pharmacology, Quipazine, Antagonist, Biological activity, medicine.disease, Ligand (biochemistry), Ondansetron, Molecular biology, In vitro, Electrophysiology, Kinetics, Endocrinology, Serotonin Antagonists, medicine.drug

    URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::90d1727ce9568ae9d6415bcc5c156d5c
    https://doi.org/10.1111/j.1472-8206.1993.tb00233.x

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  2. 2
    S18616, a highly potent, spiroimidazoline agonist at alpha(2)-adrenoceptors: I. Receptor profile, antinociceptive and hypothermic actions in comparison with dexmedetomidine and clonidine

    المؤلفون: Mj, Millan, Dekeyne A, Newman-Tancredi A, Cussac D, Audinot V, Milligan G, Duqueyroix D, Girardon S, Mullot J, Jean Albert Boutin, Jp, Nicolas, Renouard-Try A, Jm, Lacoste, Cordi A

    المصدر: Europe PubMed Central

    مصطلحات موضوعية: Male, Receptors, Drug, Imidazoles, CHO Cells, Analgesics, Non-Narcotic, Clonidine, Body Temperature, Rats, Mice, Cricetinae, Adrenergic alpha-2 Receptor Agonists, Animals, Humans, Imidazoline Receptors, Rats, Wistar, Adrenergic alpha-Agonists, Oxazoles, Dexmedetomidine

    URL الوصول: https://explore.openaire.eu/search/publication?articleId=pmid_dedup__::3d3e195a812d3d20e0fe958f81e72a2f
    https://pubmed.ncbi.nlm.nih.gov/11082457

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  3. 3
    دورية أكاديمية
    Role of NADPH oxidase-mediated superoxide production in the regulation of E-selectin expression by endothelial cells subjected to anoxia/reoxygenation.

    المؤلفون: Rupin A; Division of Angiology, Servier Research Institute, 11 rue des Moulineaux, Suresnes 92150, France., Paysant J, Sansilvestri-Morel P, Lembrez N, Lacoste JM, Cordi A, Verbeuren TJ

    المصدر: Cardiovascular research [Cardiovasc Res] 2004 Aug 01; Vol. 63 (2), pp. 323-30.

    نوع المنشور: Journal Article

    بيانات الدورية: Publisher: Oxford Journals Country of Publication: England NLM ID: 0077427 Publication Model: Print Cited Medium: Print ISSN: 0008-6363 (Print) Linking ISSN: 00086363 NLM ISO Abbreviation: Cardiovasc Res Subsets: MEDLINE

    مواضيع طبية MeSH: E-Selectin/*metabolism , Endothelial Cells/*metabolism , Hypoxia/*metabolism , NADPH Oxidases/*metabolism , Superoxides/*metabolism, Blotting, Southern/methods ; Blotting, Western/methods ; Cells, Cultured ; Humans ; Membrane Transport Proteins/genetics ; NADPH Dehydrogenase/genetics ; Phosphoproteins/analysis ; Phosphoproteins/genetics ; RNA, Messenger/analysis ; Reverse Transcriptase Polymerase Chain Reaction

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  4. 4
    دورية أكاديمية
    Potential antidepressants displayed combined alpha(2)-adrenoceptor antagonist and monoamine uptake inhibitor properties.

    المؤلفون: Cordi AA; Institut de Recherches Servier, 11, rue des Moulineaux, F-92150 Suresnes, France. alex.cordi@fr.netgrs.com, Berque-Bestel I, Persigand T, Lacoste JM, Newman-Tancredi A, Audinot V, Millan MJ

    المصدر: Journal of medicinal chemistry [J Med Chem] 2001 Mar 01; Vol. 44 (5), pp. 787-805.

    نوع المنشور: Journal Article

    بيانات الدورية: Publisher: American Chemical Society Country of Publication: United States NLM ID: 9716531 Publication Model: Print Cited Medium: Print ISSN: 0022-2623 (Print) Linking ISSN: 00222623 NLM ISO Abbreviation: J Med Chem Subsets: MEDLINE

    مواضيع طبية MeSH: Adrenergic Uptake Inhibitors/*chemical synthesis , Adrenergic alpha-Antagonists/*chemical synthesis , Antidepressive Agents/*chemical synthesis , Imidazoles/*chemical synthesis , Indans/*chemical synthesis , Receptors, Adrenergic, alpha-2/*drug effects , Selective Serotonin Reuptake Inhibitors/*chemical synthesis, Adrenergic Uptake Inhibitors/chemistry ; Adrenergic Uptake Inhibitors/metabolism ; Adrenergic alpha-Antagonists/chemistry ; Adrenergic alpha-Antagonists/metabolism ; Animals ; Antidepressive Agents/chemistry ; Antidepressive Agents/metabolism ; Binding Sites ; Binding, Competitive ; CHO Cells ; Cerebral Cortex/metabolism ; Cricetinae ; Frontal Lobe/metabolism ; Imidazoles/chemistry ; Imidazoles/metabolism ; In Vitro Techniques ; Indans/chemistry ; Indans/metabolism ; Ligands ; Norepinephrine/antagonists & inhibitors ; Rats ; Receptors, Adrenergic, alpha-2/metabolism ; Selective Serotonin Reuptake Inhibitors/chemistry ; Selective Serotonin Reuptake Inhibitors/metabolism ; Structure-Activity Relationship

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  5. 5
    دورية أكاديمية
    S18616, a highly potent, spiroimidazoline agonist at alpha(2)-adrenoceptors: I. Receptor profile, antinociceptive and hypothermic actions in comparison with dexmedetomidine and clonidine.

    المؤلفون: Millan MJ; Psychopharmacology Department, Institut de Recherches Servier, Centre de Recherches de Croissy, Croissy/Seine, Paris, France., Dekeyne A, Newman-Tancredi A, Cussac D, Audinot V, Milligan G, Duqueyroix D, Girardon S, Mullot J, Boutin JA, Nicolas JP, Renouard-Try A, Lacoste JM, Cordi A

    المصدر: The Journal of pharmacology and experimental therapeutics [J Pharmacol Exp Ther] 2000 Dec; Vol. 295 (3), pp. 1192-205.

    نوع المنشور: Comparative Study; Journal Article

    بيانات الدورية: Publisher: American Society for Pharmacology and Experimental Therapeutics Country of Publication: United States NLM ID: 0376362 Publication Model: Print Cited Medium: Print ISSN: 0022-3565 (Print) Linking ISSN: 00223565 NLM ISO Abbreviation: J Pharmacol Exp Ther Subsets: MEDLINE

    مواضيع طبية MeSH: Adrenergic alpha-2 Receptor Agonists*, Adrenergic alpha-Agonists/*pharmacology , Analgesics, Non-Narcotic/*pharmacology , Body Temperature/*drug effects , Clonidine/*pharmacology , Dexmedetomidine/*pharmacology , Oxazoles/*pharmacology, Animals ; CHO Cells ; Cricetinae ; Humans ; Imidazoles/pharmacology ; Imidazoline Receptors ; Male ; Mice ; Rats ; Rats, Wistar ; Receptors, Drug/metabolism

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  6. 6
    دورية أكاديمية
    S18616, a highly potent spiroimidazoline agonist at alpha(2)-adrenoceptors: II. Influence on monoaminergic transmission, motor function, and anxiety in comparison with dexmedetomidine and clonidine.

    المؤلفون: Millan MJ; Psychopharmacology Department, Institut de Recherches Servier, Centre de Recherches de Croissy, Croissy/Seine, Paris, France., Lejeune F, Gobert A, Brocco M, Auclair A, Bosc C, Rivet JM, Lacoste JM, Cordi A, Dekeyne A

    المصدر: The Journal of pharmacology and experimental therapeutics [J Pharmacol Exp Ther] 2000 Dec; Vol. 295 (3), pp. 1206-22.

    نوع المنشور: Comparative Study; Journal Article

    بيانات الدورية: Publisher: American Society for Pharmacology and Experimental Therapeutics Country of Publication: United States NLM ID: 0376362 Publication Model: Print Cited Medium: Print ISSN: 0022-3565 (Print) Linking ISSN: 00223565 NLM ISO Abbreviation: J Pharmacol Exp Ther Subsets: MEDLINE

    مواضيع طبية MeSH: Adrenergic alpha-2 Receptor Agonists*, Adrenergic alpha-Agonists/*pharmacology , Anti-Anxiety Agents/*pharmacology , Biogenic Monoamines/*metabolism , Clonidine/*pharmacology , Dexmedetomidine/*pharmacology , Motor Activity/*drug effects , Oxazoles/*pharmacology, Animals ; Imidazoles/pharmacology ; Locus Coeruleus/drug effects ; Locus Coeruleus/physiology ; Male ; Mice ; Raphe Nuclei/drug effects ; Raphe Nuclei/physiology ; Rats ; Rats, Wistar ; Ventral Tegmental Area/drug effects ; Vocalization, Animal/drug effects

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  7. 7
    دورية أكاديمية
    Design, synthesis and structure-activity relationships of novel strychnine-insensitive glycine receptor ligands.

    المؤلفون: Cordi A; Institut de Recherches Servier, Suresnes, France. cordi@netgrs.com, Lacoste JM, Audinot V, Millan M

    المصدر: Bioorganic & medicinal chemistry letters [Bioorg Med Chem Lett] 1999 May 17; Vol. 9 (10), pp. 1409-14.

    نوع المنشور: Journal Article

    بيانات الدورية: Publisher: Elsevier Science Ltd Country of Publication: England NLM ID: 9107377 Publication Model: Print Cited Medium: Print ISSN: 0960-894X (Print) Linking ISSN: 0960894X NLM ISO Abbreviation: Bioorg Med Chem Lett Subsets: MEDLINE

    مواضيع طبية MeSH: Drug Design*, Glycine/*metabolism , Imidazoles/*chemistry , Imidazoles/*pharmacology , Receptors, N-Methyl-D-Aspartate/*metabolism , Strychnine/*pharmacology, Imidazoles/chemical synthesis ; Ligands ; Receptors, N-Methyl-D-Aspartate/chemistry ; Structure-Activity Relationship

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  8. 8
    دورية أكاديمية
    Recording of the saphenous vein compliance by an ultrasonic echo-tracking device in the dog: effects of S 18149.

    المؤلفون: Vayssettes-Courchay C; Division of Angiology, Servier Research Institute, Suresnes, France., Cordi AA, Lacoste JM, Laubie M, Verbeuren TJ

    المصدر: British journal of pharmacology [Br J Pharmacol] 1997 Dec; Vol. 122 (7), pp. 1361-6.

    نوع المنشور: Journal Article

    بيانات الدورية: Publisher: Wiley Country of Publication: England NLM ID: 7502536 Publication Model: Print Cited Medium: Print ISSN: 0007-1188 (Print) Linking ISSN: 00071188 NLM ISO Abbreviation: Br J Pharmacol Subsets: MEDLINE

    مواضيع طبية MeSH: Saphenous Vein/*drug effects , Tetrahydronaphthalenes/*pharmacology , Vasoconstrictor Agents/*pharmacology, Administration, Oral ; Anesthesia ; Animals ; Compliance/drug effects ; Dogs ; Female ; Infusions, Intravenous ; Male ; Phenylephrine/pharmacology ; Saphenous Vein/physiology

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  9. 9
    دورية أكاديمية
    (S)-spiro[(1,3-diazacyclopent-1-ene)-5,2'-(7'-methyl-1',2',3',4'- tetrahydronaphthalene)]: resolution, stereospecific synthesis, and preliminary pharmacological characterization as a partial alpha-adrenergic agonist.

    المؤلفون: Cordi AA; Institut de Recherches Servier, Suresnes, France., Lacoste JM, Le Borgne F, Herve Y, Vaysse-Ludot L, Descombes JJ, Courchay C, Laubie M, Verbeuren TJ

    المصدر: Journal of medicinal chemistry [J Med Chem] 1997 Aug 29; Vol. 40 (18), pp. 2931-5.

    نوع المنشور: Journal Article

    بيانات الدورية: Publisher: American Chemical Society Country of Publication: United States NLM ID: 9716531 Publication Model: Print Cited Medium: Print ISSN: 0022-2623 (Print) Linking ISSN: 00222623 NLM ISO Abbreviation: J Med Chem Subsets: MEDLINE

    مواضيع طبية MeSH: Adrenergic alpha-Agonists/*chemistry , Blood Pressure/*drug effects , Muscle, Smooth, Vascular/*physiology , Tetrahydronaphthalenes/*chemistry, Adrenergic alpha-Agonists/chemical synthesis ; Adrenergic alpha-Agonists/pharmacology ; Animals ; Crystallography, X-Ray ; Femoral Artery/drug effects ; In Vitro Techniques ; Magnetic Resonance Spectroscopy ; Models, Molecular ; Molecular Conformation ; Molecular Structure ; Muscle Contraction/drug effects ; Muscle, Smooth, Vascular/drug effects ; Phenylephrine/pharmacology ; Prazosin/pharmacology ; Rats ; Saphenous Vein/drug effects ; Saphenous Vein/pathology ; Stereoisomerism ; Structure-Activity Relationship ; Tetrahydronaphthalenes/chemical synthesis ; Tetrahydronaphthalenes/pharmacology ; Yohimbine/pharmacology

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  10. 10
    دورية أكاديمية
    Design, synthesis, and structure-activity relationships of a new series of alpha-adrenergic agonists: spiro[(1,3-diazacyclopent-1-ene)-5,2'-(1',2',3',4'- tetrahydronaphthalene)].

    المؤلفون: Cordi AA; Institut de Recherches Servier, Suresnes, France., Lacoste JM, Descombes JJ, Courchay C, Vanhoutte PM, Laubie M, Verbeuren TJ

    المصدر: Journal of medicinal chemistry [J Med Chem] 1995 Sep 29; Vol. 38 (20), pp. 4056-69.

    نوع المنشور: Journal Article

    بيانات الدورية: Publisher: American Chemical Society Country of Publication: United States NLM ID: 9716531 Publication Model: Print Cited Medium: Print ISSN: 0022-2623 (Print) Linking ISSN: 00222623 NLM ISO Abbreviation: J Med Chem Subsets: MEDLINE

    مواضيع طبية MeSH: Adrenergic alpha-Agonists/*chemical synthesis , Imidazoles/*chemical synthesis, Adrenergic alpha-Agonists/pharmacology ; Animals ; Dogs ; Imidazoles/pharmacology ; In Vitro Techniques ; Male ; Rats ; Rats, Sprague-Dawley ; Structure-Activity Relationship ; Vasoconstriction/drug effects

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