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1
المؤلفون: Susan K. Yagel, Ellen E. Codd, Sui-Po Zhang, Jack A. Kauffman
المصدر: SLAS Discovery. 11:672-677
مصطلحات موضوعية: Ziconotide, Voltage-dependent calcium channel, medicine.drug_class, Chemistry, Calcium channel, Ligand binding assay, Drug Evaluation, Preclinical, Brain, Calcium channel blocker, N-type calcium channel, Pharmacology, Calcium Channel Blockers, Ligand (biochemistry), Biochemistry, Rats, Analytical Chemistry, Calcium Channels, N-Type, Scintillation proximity assay, medicine, Animals, Scintillation Counting, Molecular Medicine, Biotechnology, medicine.drug
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::0c2c57b65e7d939461f0844fe01085b3
https://doi.org/10.1177/1087057106289210 -
2
المؤلفون: Annette J. Eckardt, Enrico Di Cera, Jack A. Kauffman, Edward C. Giardino, Thomas W. Corcoran, Michael N. Greco, Bruce E. Maryanoff, Lawrence de Garavilla, Claudia K. Derian, Narayanasami Sukumar, Barbara J. Haertlein, Zhi-wei Chen, Bruce P. Damiano, Grace I. Wells, Patricia Andrade-Gordon, F. Scott Mathews, Agustin O. Pineda
المصدر: Journal of Biological Chemistry. 280:18001-18007
مصطلحات موضوعية: Proteases, Chymase, Cell Biology, Cathepsin G, Biochemistry, Molecular biology, Cathepsin B, Nitric oxide, Serine, chemistry.chemical_compound, chemistry, Cathepsin O, Cathepsin L1, Molecular Biology
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_________::2bb41a9acbf419e02cb964ca95c9e201
https://doi.org/10.1074/jbc.m501302200 -
3
المؤلفون: Patricia Andrade-Gordon, Frank A. Amato, Sergey E. Ilyin, Albert Pinhasov, Douglas E. Brenneman, Jack A. Kauffman, Dhammika Amaratunga, Dana L. Johnson, Hong Lu, Jay Mei, Hong Xin
المصدر: Combinatorial Chemistry & High Throughput Screening. 7:133-140
مصطلحات موضوعية: Biomarker identification, Reverse Transcriptase Polymerase Chain Reaction, Drug discovery, Gene Expression Profiling, High-throughput screening, Organic Chemistry, General Medicine, Computational biology, Biology, Molecular biology, Computer Science Applications, High throughput analysis, Gene expression profiling, Drug Design, Drug Discovery, Gene expression, TaqMan, Taq Polymerase, RNA, Messenger, Throughput (business)
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::cf5d498b1eb3a0bc165f2acb728bde2a
https://doi.org/10.2174/138620704773120810 -
4
المؤلفون: Jack A. Kauffman, Michael J. Costanzo, William A. Kinney, Rosemary J. Santulli, Stephen C. Yabut, Brett A. Tounge, Patricia Andrade-Gordon, Edward C. Lawson, Diane K. Luci, Hoekstra William J
المصدر: Letters in Drug Design & Discovery. 1:14-18
مصطلحات موضوعية: chemistry.chemical_compound, chemistry, biology, Stereochemistry, Drug Discovery, Structure function, biology.protein, Pharmaceutical Science, Molecular Medicine, Vitronectin, Ligand (biochemistry), Receptor, Quinazolinone
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_________::4cebab9524db6475d2791ace4a2e054a
https://doi.org/10.2174/1570180043485644 -
5
المؤلفون: Jack A. Kauffman, Joseph J. Salata, Ramesh M. Kanojia
المصدر: Bioorganic & Medicinal Chemistry Letters. 10:2819-2823
مصطلحات موضوعية: chemistry.chemical_classification, Chemistry, medicine.drug_class, Stereochemistry, medicine.medical_treatment, Aryl, Organic Chemistry, Clinical Biochemistry, Nitro compound, Pharmaceutical Science, Carboxamide, macromolecular substances, Class iii, Antiarrhythmic agent, Biochemistry, Chemical synthesis, In vitro, chemistry.chemical_compound, Drug Discovery, medicine, Molecular Medicine, Piperidine, Molecular Biology
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6
المؤلفون: Quan Sheng Li, Michael J. Costanzo, Edward C. Giardino, Jack A. Kauffman, Patricia Andrade-Gordon, Bruce E. Maryanoff
المصدر: Thrombosis Research. 98:83-93
مصطلحات موضوعية: Blood Platelets, Platelet Aggregation, Pharmacology, Guanidines, Hemostatics, Dogs, Thrombin, Fibrinolytic Agents, Bleeding time, Antithrombotic, medicine, Animals, Humans, Platelet, medicine.diagnostic_test, biology, Chemistry, Hematology, Thiazoles, Coagulation, Enzyme inhibitor, Anesthesia, biology.protein, Platelet aggregation inhibitor, Rabbits, Platelet Aggregation Inhibitors, Fibrinolytic agent, medicine.drug
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7
المؤلفون: Barbara J. Haertlein, Jack A. Kauffman, Judith H. Cohen, Patricia Andrade-Gordon, John A. Mitchell, Patricia Keane, Hoekstra William J, Michael J. Costanzo, David F. McComsey, Rekha D. Shah, Bruce P. Damiano, Becky L. Hulshizer, Bruce E. Maryanoff, Stephen C. Yabut, Leonard R. Hecker, Lorraine Scott
المصدر: Journal of Medicinal Chemistry. 42:5254-5265
مصطلحات موضوعية: Magnetic Resonance Spectroscopy, Proline, Pyridines, Fibrinogen receptor, Nipecotic Acids, Administration, Oral, Biological Availability, Platelet Glycoprotein GPIIb-IIIa Complex, Pharmacology, Fibrinogen, Mass Spectrometry, Structure-Activity Relationship, Dogs, In vivo, Oral administration, Drug Discovery, medicine, Animals, Potency, Platelet, Chemistry, Biochemistry, Area Under Curve, Molecular Medicine, Platelet aggregation inhibitor, Platelet Aggregation Inhibitors, Ex vivo, medicine.drug
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8
المؤلفون: Joan M. Lewis, Jack A. Kauffman, Patricia Andrade-Gordon, Venkatapathy Ganesh, Michael N. Greco, Bruce E. Maryanoff, Leonard R. Hecker, Powell Eugene, Alexander Tulinsky
المصدر: Bioorganic & Medicinal Chemistry Letters. 6:2947-2952
مصطلحات موضوعية: Stereochemistry, Chemistry, Organic Chemistry, Clinical Biochemistry, Pharmaceutical Science, Tripeptide, Biochemistry, In vitro, Ring size, Enzyme inhibition, Thrombin, Drug Discovery, medicine, Molecular Medicine, Bovine trypsin, Molecular Biology, Ternary complex, medicine.drug, Discovery and development of direct thrombin inhibitors
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9
المؤلفون: Bruce D. Harris, Frank J. Villani, Jack A. Kauffman, Hoekstra William J, Patricia Andrade-Gordon, Michael J. Costanzo, Judith H. Cohen, Bruce P. Damiano, Stephen C. Yabut, David F. McComsey, Bruce E. Maryanoff, Barbara J. Haertlein, Patricia Keane
المصدر: Bioorganic & Medicinal Chemistry Letters. 6:2371-2376
مصطلحات موضوعية: chemistry.chemical_classification, Gpiib iiia antagonist, Fibrinogen receptor, Stereochemistry, Organic Chemistry, Clinical Biochemistry, Antagonist, Pharmaceutical Science, Peptide, Fibrinogen, Biochemistry, Combinatorial chemistry, In vitro, chemistry.chemical_compound, chemistry, Drug Discovery, Nipecotic acid, medicine, Molecular Medicine, Potency, Molecular Biology, medicine.drug
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10
المؤلفون: Michael N. Greco, Kyriacos C. Nicolaou, Aijun Liu, Patricia Andrade-Gordon, Jack A. Kauffman, Bruce E. Maryanoff, Han-Cheng Zhang, Peter H. Brungs
المصدر: Journal of the American Chemical Society. 117:1225-1239
مصطلحات موضوعية: Proteases, Primary (chemistry), Chemistry, Late stage, Total synthesis, General Chemistry, Biochemistry, Catalysis, Serine, Colloid and Surface Chemistry, Thrombin, medicine, Amine gas treating, MASP1, medicine.drug