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1
المؤلفون: Zhi-Jie Ni, Qun Li, Martin John Slater, Wuxin Zou, Linos Lazarides, Yang Liu, Lois L. Wright, Paul Rowland, Liang Liao, Charles Z. Ding, Tadeusz Skarzynski, Jacob J. Plattner, Jackie E. Mordaunt, Don O. Somers, Xianfeng Li, Colin M. Edge, Yong-Kang Zhang, Gemma Victoria White, Malcolm Ellis, Jon Wright, Stephen J. Baker, Dazhong Fan, Wieslaw M. Kazmierski, Gary K. Smith, Pia Thommes, Lewis E. Pennicott, Julia A. Hubbard, Richard L. Jarvest, Bill McDowell, Yasheen Zhou, Xuelei Qian, Pamela Nassau, Richard Martin Grimes
المصدر: Bioorganic & Medicinal Chemistry Letters. 20:3550-3556
مصطلحات موضوعية: Stereochemistry, viruses, medicine.medical_treatment, Clinical Biochemistry, Pharmaceutical Science, Peptide, Hepacivirus, Viral Nonstructural Proteins, Biochemistry, Chemical synthesis, Structure-Activity Relationship, Catalytic Domain, Drug Discovery, Serine, medicine, Molecular Biology, chemistry.chemical_classification, Serine protease, NS3, Protease, Molecular Structure, biology, Organic Chemistry, virus diseases, Active site, Boronic Acids, digestive system diseases, Protease inhibitor (biology), chemistry, Enzyme inhibitor, Drug Design, biology.protein, Molecular Medicine, medicine.drug
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2
المؤلفون: Fabrizio Nerozzi, Shalia S Shabbir, Paul G. Wyatt, Mamta Patel, Michael Allen, Josie Chilcott, Christopher J. Gardner, Marion J. Perren, Jackie E. Mordaunt, Livermore David, Gordon G. Weingarten, Ping Zhou, Patrick M. Woollard
المصدر: Bioorganic & Medicinal Chemistry Letters. 12:1405-1411
مصطلحات موضوعية: Models, Molecular, endocrine system, medicine.drug_class, Clinical Biochemistry, Molecular Conformation, Pharmaceutical Science, Carboxamide, Pharmacology, Oxytocin, Biochemistry, Oxytocin Antagonist, Structure-Activity Relationship, Uterine Contraction, chemistry.chemical_compound, In vivo, Drug Discovery, medicine, Animals, Humans, Benzofuran, Molecular Biology, Benzofurans, Organic Chemistry, Antagonist, Oxytocin receptor, Rats, Kinetics, chemistry, Receptors, Oxytocin, Drug Design, Molecular Medicine, Female, hormones, hormone substitutes, and hormone antagonists, medicine.drug
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3
المؤلفون: Josie Chilcott, Paul Wyatt, Alison Foster, Jan Scicinski, Livermore David, Patrick M. Woollard, Michael J. Allen, Jackie E. Mordaunt
المصدر: Bioorganic & Medicinal Chemistry Letters. 12:1399-1404
مصطلحات موضوعية: Models, Molecular, Indoles, Pyrimidine, Stereochemistry, Clinical Biochemistry, Molecular Conformation, Biological Availability, Pharmaceutical Science, Oxytocin, Biochemistry, Oxytocin Antagonist, Structure-Activity Relationship, chemistry.chemical_compound, Dogs, Drug Discovery, Animals, Humans, Moiety, Benzofuran, Thiazole, Molecular Biology, Benzofurans, Indole test, Organic Chemistry, Antagonist, Oxytocin receptor, Kinetics, chemistry, Receptors, Oxytocin, Drug Design, Molecular Medicine, hormones, hormone substitutes, and hormone antagonists
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4
المؤلفون: Jackie E. Mordaunt, Paul Wyatt, Michael J. Allen, Alison Foster, Livermore David, Jan Scicinski, Josie Chilcott, Patrick M. Woollard
المصدر: ChemInform. 33
مصطلحات موضوعية: Indole test, Pyrimidine, Chemistry, Stereochemistry, General Medicine, Oxytocin Antagonist, chemistry.chemical_compound, Oxytocin, medicine, Moiety, Benzofuran, Thiazole, hormones, hormone substitutes, and hormone antagonists, medicine.drug, Benzoic acid
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5
المؤلفون: Paul G. Wyatt, Jackie E. Mordaunt, et al. et al.
المصدر: ChemInform. 33
مصطلحات موضوعية: chemistry.chemical_compound, chemistry, Oxytocin, Stereochemistry, medicine, Identification (biology), General Medicine, Benzofuran, medicine.drug
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6
المؤلفون: Matthew Campbell, Ping Zhou, Robert J. Young, Weston Helen Elisabeth, Savvas Kleanthous, David W. Brown, Champa Patel, Satish Dayal, Shah Gita Punjabhai, Alan D. Borthwick, N. Paul King, Cynthia L. Burns-Kurtis, Stefan Senger, Hawa Diallo, Máire A. Convery, Nigel S. Watson, Paul W. Smith, Henry Anderson Kelly, Miriam Crowe, Chuen Chan, Anthony J. Pateman, Jackie E. Mordaunt, Andrew M. Mason
المصدر: Bioorganicmedicinal chemistry letters. 16(23)
مصطلحات موضوعية: Models, Molecular, medicine.drug_mechanism_of_action, Molecular model, Stereochemistry, Clinical Biochemistry, Factor Xa Inhibitor, Antithrombin III, Substituent, Pharmaceutical Science, Crystallography, X-Ray, Biochemistry, Chemical synthesis, chemistry.chemical_compound, Structure-Activity Relationship, Amide, Drug Discovery, Hydrolase, medicine, Pyrroles, Molecular Biology, chemistry.chemical_classification, Alanine, Binding Sites, Molecular Structure, Organic Chemistry, Anticoagulants, Amides, Sulfonamide, chemistry, Drug Design, Lipophilicity, Factor Xa, Molecular Medicine