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1
المؤلفون: Walter G. Smith, Suzanne H Kim, Doreen Villani-Price, Matthew W Mahoney, Nayereh S Ghoreishi-Haack, Helen Y. Chen, Thomas D. Penning, Stella Siu-Tzyy Yu, James W. Malecha, Leslie J Askonas, Chi-Dean Liang, Elizabeth I Harding, E.Yvonne Pyla, Maureen K Highkin, James K. Gierse, Julie M Miyashiro, Mark A Russell, James F Kachur, Chen Barbara B
المصدر: Journal of Medicinal Chemistry. 45:3482-3490
مصطلحات موضوعية: Epoxide Hydrolases, chemistry.chemical_classification, biology, Stereochemistry, Administration, Oral, Leukotriene A4, Chemical synthesis, Proinflammatory cytokine, Leukotriene-A4 hydrolase, Mice, Structure-Activity Relationship, Enzyme, chemistry, Enzyme inhibitor, In vivo, Drug Discovery, Hydrolase, beta-Alanine, biology.protein, Animals, Humans, Molecular Medicine, Structure–activity relationship, Enzyme Inhibitors
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2
المؤلفون: Leslie J Askonas, Mark A Russell, Walter G. Smith, James F. Kachur, Chi-Dean D. Liang, D Villani-Price
المصدر: Journal of Pharmacology and Experimental Therapeutics. 300:577-582
مصطلحات موضوعية: beta-Alanine, Enzyme-Linked Immunosorbent Assay, In Vitro Techniques, Pharmacology, Aminopeptidases, Substrate Specificity, Mice, chemistry.chemical_compound, Dogs, Species Specificity, In vivo, Hydrolase, Animals, Humans, Enzyme Inhibitors, Epoxide hydrolase, Chromatography, High Pressure Liquid, Epoxide Hydrolases, Leukotriene, Arachidonic Acid, Ionophores, Leukotriene A4, Macaca mulatta, Recombinant Proteins, Rats, Kinetics, chemistry, Biochemistry, Eicosanoids, Leukotriene Antagonists, Molecular Medicine, Arachidonic acid, Ex vivo
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::8a43488c1feb896fd592f6e43e83a9e0
https://doi.org/10.1124/jpet.300.2.577 -
3
المؤلفون: Thomas D. Penning, Nizal S. Chandrakumar, Barbara B. Chen, Helen Y. Chen, Bipin N. Desai, Stevan W. Djuric, Stephen H. Docter, Alan F. Gasiecki, Richard A. Haack, Julie M. Miyashiro, Mark A. Russell, Stella S. Yu, David G. Corley, Richard C. Durley, Brian F. Kilpatrick, Barry L. Parnas, Leslie J. Askonas, James K. Gierse, Elizabeth I. Harding, Maureen K. Highkin, James F. Kachur, Suzanne H. Kim, Gwen G. Krivi, Doreen Villani-Price, E. Yvonne Pyla, Walter G. Smith, Nayereh S. Ghoreishi-Haack
المصدر: Journal of Medicinal Chemistry. 43:721-735
مصطلحات موضوعية: Male, Pyrrolidines, Tertiary amine, Administration, Oral, In Vitro Techniques, Pharmacology, Leukotriene B4, Leukotriene-A4 hydrolase, Mice, Structure-Activity Relationship, Drug Discovery, Hydrolase, Animals, Humans, Structure–activity relationship, Enzyme Inhibitors, Epoxide Hydrolases, chemistry.chemical_classification, biology, In vitro, Enzyme, Biochemistry, chemistry, Enzyme inhibitor, biology.protein, Molecular Medicine, Ex vivo
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4
المؤلفون: Timothy S. Gaginella, James F. Kachur, C. P. Anglin, Suzanne Won-Kim
المصدر: Inflammation. 19:717-725
مصطلحات موضوعية: Male, medicine.medical_specialty, Guinea Pigs, Immunology, Complement C5a, Ileum, Tetrodotoxin, Histamine Release, Guinea pig, Electrolytes, chemistry.chemical_compound, Internal medicine, medicine, Animals, Immunology and Allergy, Intestinal Mucosa, Ussing chamber, Chemistry, Muscarinic antagonist, Recombinant Proteins, Electrophysiology, medicine.anatomical_structure, Endocrinology, Mechanism of action, Prostaglandin-Endoperoxide Synthases, Eicosanoids, Arachidonic acid, medicine.symptom, Histamine, medicine.drug
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5
المؤلفون: M M de las Alas, R Walsh, Ali Keshavarzian, T S Gaginella, James F. Kachur, M Doria, R Sundaresan
المصدر: Inflammation. 19:245-259
مصطلحات موضوعية: Anions, Male, Serotonin, medicine.medical_specialty, Patch-Clamp Techniques, Time Factors, Carbachol, Neutrophils, Mitomycin, Immunology, Bradykinin, Substance P, Inflammation, Second Messenger Systems, Rats, Sprague-Dawley, chemistry.chemical_compound, Theophylline, Internal medicine, medicine, Animals, Immunology and Allergy, Alprostadil, Intestinal Mucosa, Colitis, Receptor, Prostaglandin E1, Peroxidase, business.industry, medicine.disease, Epithelium, Rats, Endocrinology, medicine.anatomical_structure, chemistry, medicine.symptom, Secretory Rate, business, medicine.drug
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6
المؤلفون: D. Spangler, James F Kachur, C. P. Anglin, Snyder Jp, Stella Siu-Tzyy Yu, T. D. Penning, S. W. Djuric, R H Keith, D. J. Fretland, Julie M Miyashiro
المصدر: Journal of Medicinal Chemistry. 38:858-868
مصطلحات موضوعية: Azoles, Stereochemistry, medicine.drug_class, Guinea Pigs, Molecular Sequence Data, Receptors, Leukotriene B4, Intracolonic, Mice, Structure-Activity Relationship, In vivo, Drug Discovery, medicine, Animals, Humans, Benzopyrans, Amino Acid Sequence, Colitis, Leukotriene, Chemotactic Factors, Chemistry, Leukotriene B4 receptor, Antagonist, medicine.disease, Receptor antagonist, N-Formylmethionine Leucyl-Phenylalanine, Thiazoles, Molecular Medicine, Pharmacophore
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7
المؤلفون: Doreen Villani-Price, Suzanne H Kim, Walter G. Smith, Leslie J Askonas, Elizabeth I Harding, Maureen K Highkin, Thomas D. Penning, Alan F. Gasiecki, Nayereh S Ghoreishi-Haack, Nizal S Chandrakumar, E.Yvonne Pyla, Bipin N Desai, James F Kachur, Mark A Russell, Stevan W Djuric, James W. Malecha, James K. Gierse, Julie M Miyashiro
المصدر: Bioorganic & Medicinal Chemistry Letters. 13:1137-1139
مصطلحات موضوعية: Imidazopyridine, Pyridines, Clinical Biochemistry, Pharmaceutical Science, Purine analogue, In Vitro Techniques, Biochemistry, Chemical synthesis, Leukotriene-A4 hydrolase, Mice, Structure-Activity Relationship, Heterocyclic Compounds, Drug Discovery, Animals, Humans, Structure–activity relationship, Enzyme Inhibitors, Purine metabolism, Molecular Biology, Epoxide Hydrolases, biology, Chemistry, Organic Chemistry, Recombinant Proteins, stomatognathic diseases, Purines, Enzyme inhibitor, biology.protein, Molecular Medicine, Indicators and Reagents, Ex vivo
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8
المؤلفون: D. J. Fretland, D. L. Widomski, Timothy S. Gaginella, James F. Kachur, T.J. Maziasz, C. P. Anglin, B.S. Tsai, Stella S. Yu, Tadimeti S. Rao, R. E. Walsh, R H Keith, Stephen H Docter, Stevan W. Djuric, D Villani-Price
المصدر: Bioorganic & Medicinal Chemistry Letters. 4:811-816
مصطلحات موضوعية: Chemistry, Leukotriene B4, Organic Chemistry, Clinical Biochemistry, Leukotriene B4 receptor, Antagonist, Pharmaceutical Science, Biological activity, Pharmacology, Biochemistry, Chemical synthesis, chemistry.chemical_compound, Pharmacodynamics, Drug Discovery, Molecular Medicine, Potency, Structure–activity relationship, Molecular Biology
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9
المؤلفون: James F. Kachur, Suzanne Won-Kim, Timothy S. Gaginella
المصدر: Prostaglandins. 46:221-231
مصطلحات موضوعية: Male, medicine.medical_specialty, Colon, In Vitro Techniques, Biology, Biochemistry, Rats, Sprague-Dawley, Electrolytes, chemistry.chemical_compound, Endocrinology, In vivo, 16,16-Dimethylprostaglandin E2, Internal medicine, medicine, Animals, Intestinal Mucosa, Prostaglandin E1, Biological Transport, Stereoisomerism, In vitro, Rats, Atropine, Mechanism of action, Eicosanoid, chemistry, Tetrodotoxin, medicine.symptom, Misoprostol, Bumetanide, medicine.drug
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10
المؤلفون: Timothy S. Gaginella, M. W. Musch, Hiroshi Tamai, Matthew B. Grisham, James F. Kachur, E. B. Chang
المصدر: American Journal of Physiology-Cell Physiology. 265:C166-C170
مصطلحات موضوعية: Male, medicine.medical_specialty, Colon, Physiology, Ammonium Chloride, Rats, Sprague-Dawley, Electrolytes, chemistry.chemical_compound, Internal medicine, medicine, Animals, Secretion, Sulfhydryl Compounds, Ion transporter, Diamide, Cell Biology, Glutathione, Rats, Amiloride, Electrophysiology, Endocrinology, Mechanism of action, chemistry, Tetrodotoxin, Secretagogue, medicine.symptom, Oxidation-Reduction, Intracellular, medicine.drug
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::a13bed2bc40e61de5ff489e7729eea81
https://doi.org/10.1152/ajpcell.1993.265.1.c166