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1
المؤلفون: Rudolph G. Krause, Charles P. Sloan, Jingfang Qian-Cutrone, Thaddeus F. Molski, Joseph A. Cipollina, Gail K. Mattson, Matthew T. Taber, Qi Gao, Ronald J. Mattson, Jeffrey A. Deskus, James R. Epperson, Brett R. Beno, Baoqing Ma, Nicholas J. Lodge, Pierre Dextraze
المصدر: Bioorganic & Medicinal Chemistry Letters. 17:3099-3104
مصطلحات موضوعية: Indoles, Nitrile, Pyridines, Stereochemistry, Microdialysis, Clinical Biochemistry, Molecular Conformation, Substituent, Pharmaceutical Science, Biochemistry, chemistry.chemical_compound, Fluoxetine, Cyclohexenes, Drug Discovery, Animals, Humans, Serotonin Uptake Inhibitors, Molecular Biology, Serotonin transporter, Serotonin Plasma Membrane Transport Proteins, Indole test, biology, Organic Chemistry, Tryptamines, Rats, chemistry, biology.protein, Molecular Medicine, Serotonin, Reuptake inhibitor, Selective Serotonin Reuptake Inhibitors
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2
المؤلفون: Anthony J. Gentile, Jeffrey A. Deskus, Nathan S. Sarbin, James R. Epperson, Elaine Ryan, Lawrence G. Iben
المصدر: Bioorganic & Medicinal Chemistry Letters. 14:1023-1026
مصطلحات موضوعية: Agonist, medicine.drug_class, Stereochemistry, Clinical Biochemistry, Pharmaceutical Science, Carboxamide, Binding, Competitive, Biochemistry, Chemical synthesis, Melatonin, Structure-Activity Relationship, Drug Discovery, medicine, Humans, Anilides, Receptor, Molecular Biology, Molecular Structure, Receptor, Melatonin, MT2, Chemistry, Organic Chemistry, In vitro, Melatonergic, Molecular Medicine, Selectivity, medicine.drug
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3
المؤلفون: James R. Epperson, Clayton H. Heathcock, Robert W. Scott
المصدر: The Journal of Organic Chemistry. 63:5001-5012
مصطلحات موضوعية: Stereochemistry, Meso compound, Chemistry, Mannich condensation, Model study, Intramolecular force, Organic Chemistry, Diastereomer, Total synthesis, Model synthesis, Stereocenter
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4
المؤلفون: Jonathan L. Ditta, Derek J. Denhart, Gail K. Mattson, Zhaoxing Meng, Qi Gao, Mellissa A. LaPaglia, Jeffrey A. Deskus, Matthew T. Taber, Nicholas J. Lodge, John E. Macor, James R. Epperson, Thaddeus F. Molski, Ronald J. Mattson
المصدر: Bioorganicmedicinal chemistry letters. 23(10)
مصطلحات موضوعية: Indole test, Serotonin Plasma Membrane Transport Proteins, biology, Dose-Response Relationship, Drug, Molecular Structure, Chemistry, Organic Chemistry, Clinical Biochemistry, Molecular Conformation, Pharmaceutical Science, Pharmacology, Serotonin reuptake, Biochemistry, Methylamines, Structure-Activity Relationship, Drug Discovery, biology.protein, Molecular Medicine, Humans, Serotonin, Molecular Biology, Serotonin transporter, Selective Serotonin Reuptake Inhibitors
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5
المصدر: Synthesis. 1994:846-850
مصطلحات موضوعية: chemistry.chemical_compound, Bicyclic molecule, Chemistry, Organic Chemistry, Synthon, Organic chemistry, Aminoacylation, Isocyanate, Catalysis
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_________::7cfd0622b54ef427eda08ec6feae8d3f
https://doi.org/10.1055/s-1994-25587 -
6
المؤلفون: Piyasena Hewawasam, Debra J. Post-Munson, Christopher G. Boissard, James R. Epperson, Valentin K. Gribkoff, Nicholas A. Meanwell
المصدر: Bioorganic & Medicinal Chemistry Letters. 3:2801-2804
مصطلحات موضوعية: chemistry.chemical_classification, Organic Chemistry, Clinical Biochemistry, Glutamate receptor, Antagonist, Pharmaceutical Science, AMPA receptor, Pharmacology, Biochemistry, Chemical synthesis, Amino acid, nervous system, chemistry, Drug Discovery, Excitatory postsynaptic potential, Molecular Medicine, NMDA receptor, Antagonism, Molecular Biology
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7
المؤلفون: Piyasena Hewawasam, Valentin K. Gribkoff, Christopher G. Boissard, Debra J. Post-Munson, James R. Epperson, Nicholas A. Meanwell
المصدر: ChemInform. 25
مصطلحات موضوعية: chemistry.chemical_classification, nervous system, chemistry, Excitatory postsynaptic potential, NMDA receptor, General Medicine, AMPA receptor, Pharmacology, Antagonism, Amino acid, Functional antagonism
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8
المصدر: ChemInform. 26
مصطلحات موضوعية: chemistry.chemical_compound, Chemistry, Synthon, Organic chemistry, General Medicine, Isocyanate
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9
المؤلفون: Joyce E. Kung, Derek J. Denhart, Jeffrey A. Deskus, Nicholas J. Lodge, John E. Macor, Jonathan L. Ditta, Ronald J. Mattson, Mendi A. Higgins, James R. Epperson, Lawrence R. Marcin, Charles P. Sloan, Robert L. Bertekap, Thaddeus F. Molski, Dalton King, Rudolph G. Krause, Gail K. Mattson
المصدر: Bioorganicmedicinal chemistry letters. 17(20)
مصطلحات موضوعية: Steric effects, Tertiary amine, Stereochemistry, Serotonin reuptake inhibitor, Clinical Biochemistry, Molecular Conformation, Pharmaceutical Science, Biochemistry, Chemical synthesis, Inhibitory Concentration 50, Structure-Activity Relationship, Heterocyclic Compounds, Drug Discovery, Side chain, Humans, Molecular Biology, Serotonin transporter, Indole test, Dopamine Plasma Membrane Transport Proteins, Norepinephrine Plasma Membrane Transport Proteins, Bicyclic molecule, biology, Chemistry, Organic Chemistry, Tryptamines, biology.protein, Molecular Medicine, Selective Serotonin Reuptake Inhibitors
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10
المؤلفون: Nathan S. Sarbin, Anthony J. Gentile, Lawrence G. Iben, Jeffrey A. Deskus, Elaine Ryan, James R. Epperson
المصدر: ChemInform. 35
مصطلحات موضوعية: Melatonin, Chemistry, Stereochemistry, Mt1 receptor, medicine, General Medicine, Selectivity, Receptor, Melatonergic, medicine.drug