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1دورية أكاديمية
المؤلفون: Gregory D Ferguson, Mercedes Delgado, Veronique Plantevin-Krenitsky, Kristen Jensen-Pergakes, R J Bates, Sanaa Torres, Maria Celeridad, Heather Brown, Kelven Burnett, Lisa Nadolny, Lida Tehrani, Garrick Packard, Barbra Pagarigan, Jason Haelewyn, Trish Nguyen, Li Xu, Yang Tang, Matthew Hickman, Frans Baculi, Steven Pierce, Keiji Miyazawa, Pilgrim Jackson, Philip Chamberlain, Laurie LeBrun, Weilin Xie, Brydon Bennett, Kate Blease
المصدر: PLoS ONE, Vol 11, Iss 1, p e0145705 (2016)
وصف الملف: electronic resource
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المؤلفون: Mark A. Nagy, Robert Hilgraf, Deborah S. Mortensen, Jan Elsner, Stephen Norris, Jayashree Tikhe, Won Yoon, David Paisner, Mercedes Delgado, Paul Erdman, Jason Haelewyn, Godrej Khambatta, Li Xu, William J. Romanow, Kevin Condroski, Sogole Bahmanyar, Meg McCarrick, Brent Benish, Kate Blease, Laurie LeBrun, Mehran F. Moghaddam, Julius Apuy, Stacie S. Canan, Brydon L. Bennett, Yoshitaka Satoh
المصدر: Journal of Medicinal Chemistry. 64:18193-18208
مصطلحات موضوعية: Drug Discovery, Molecular Medicine
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المؤلفون: Philip W. Iversen, Jason Haelewyn, Jeffrey R. Weidner
المصدر: SLAS discovery : advancing life sciences RD. 26(10)
مصطلحات موضوعية: stomatognathic diseases, Statistics, Robust statistics, Molecular Medicine, Bioassay, Statistical analysis, Biological Assay, Biology, Biochemistry, Analytical Chemistry, Biotechnology
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::1cb2a9eaa1fa5a79ce70ff02a66e002f
https://pubmed.ncbi.nlm.nih.gov/34474612 -
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المؤلفون: Gregory D. Ferguson, Frans Baculi, Kristen Jensen-Pergakes, Maria Celeridad, Steven Pierce, Barbra Pagarigan, Garrick Packard, Matt Hickman, Brydon L. Bennett, Yang Tang, Li Xu, Veronique Plantevin-Krenitsky, Sanaa Torres, Lisa Nadolny, Lida Tehrani, R. J. Bates, Trish Nguyen, Jason Haelewyn, Kelven Burnett, Laurie LeBrun, Philip P Chamberlain, Weilin Xie, Kate Blease, Keiji Miyazawa, Mercedes Delgado, Pilgrim Jackson, Heather Brown
المصدر: PLoS ONE
PLoS ONE, Vol 11, Iss 1, p e0145705 (2016)مصطلحات موضوعية: 0301 basic medicine, Male, Neutrophils, Pyridines, lcsh:Medicine, Syk, Arthritis, Receptors, Fc, Crystallography, X-Ray, Rats, Sprague-Dawley, 0302 clinical medicine, Medicine, Edema, Kinome, lcsh:Science, Receptor, Skin, Multidisciplinary, Kinase, Intracellular Signaling Peptides and Proteins, hemic and immune systems, Protein-Tyrosine Kinases, Basophils, Hypertension, Female, Collagen, Tyrosine kinase, Research Article, Indazoles, Neutropenia, chemical and pharmacologic phenomena, Cell Line, 03 medical and health sciences, Inhibitory Concentration 50, Immune system, Animals, Humans, Syk Kinase, Inflammation, Dose-Response Relationship, Drug, business.industry, lcsh:R, Autoantibody, Janus Kinase 2, Triazoles, medicine.disease, Arthritis, Experimental, Vascular Endothelial Growth Factor Receptor-2, Rats, Eosinophils, 030104 developmental biology, HEK293 Cells, Rats, Inbred Lew, Immunology, Cancer research, lcsh:Q, business, 030215 immunology
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المؤلفون: Jason Haelewyn, Brian Dyck, Troy Vickers, Junko Tamiya, Mingzhu Zhang, Linh Nguyen, Martin W. Rowbottom, David A. Schwarz, Val S. Goodfellow, Monica S. Mistry, Christopher E. Heise, Jonathan Grey
المصدر: Bioorganic & Medicinal Chemistry Letters. 17:2535-2539
مصطلحات موضوعية: Pyrrolidines, Melanin-concentrating hormone, Stereochemistry, Chemistry, Pharmaceutical, Clinical Biochemistry, Molecular Conformation, Pharmaceutical Science, Plasma protein binding, Biochemistry, Chemical synthesis, Inhibitory Concentration 50, Mice, Structure-Activity Relationship, chemistry.chemical_compound, Cytochrome P-450 CYP2D6 Inhibitors, Drug Discovery, Animals, Humans, Urea, Structure–activity relationship, Receptors, Somatostatin, Molecular Biology, Bicyclic molecule, Organic Chemistry, In vitro, Melanin-concentrating hormone receptor, Kinetics, Models, Chemical, chemistry, Drug Design, Lactam, Molecular Medicine, Protein Binding
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المؤلفون: Graham Beaton, Aixia Sun, Jason Haelewyn, Susan K. Sullivan, Wilna J. Moree, Michael P. Hedrick, Mark Santos, Margaret J. Bradbury, Jenny Wen, Jinghua Yu, Said Zamani-Kord, Coon Timothy Richard, Paul D. Crowe, Lisa M. Hernández, Siobhan Malany, Robert E. Petroski, Bin-Feng Li, Samuel J. Hoare
المصدر: Bioorganicmedicinal chemistry letters. 19(15)
مصطلحات موضوعية: Benzimidazole, ERG1 Potassium Channel, medicine.medical_treatment, Chemistry, Pharmaceutical, Clinical Biochemistry, hERG, Histamine Antagonists, Pharmaceutical Science, Pharmacology, Biochemistry, Rats, Sprague-Dawley, chemistry.chemical_compound, Structure-Activity Relationship, Pharmacokinetics, In vivo, Sleep Initiation and Maintenance Disorders, Drug Discovery, medicine, Animals, Humans, Molecular Biology, biology, Electromyography, Organic Chemistry, Antagonist, Brain, Electroencephalography, Ether-A-Go-Go Potassium Channels, Rats, chemistry, Models, Chemical, Drug Design, biology.protein, Molecular Medicine, Antihistamine, Benzimidazoles, Histamine, Mizolastine, medicine.drug